Structures of Kibdelomycin Bound to Staphylococcus aureus GyrB and ParE Showed a Novel U‑Shaped Binding Mode von Lu, Jun, Patel, Sangita, Sharma, Nandini, Soisson, Stephen M, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Lumb, Kevin J, Singh, Sheo B

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Kibdelomycin is a bactericidal broad-spectrum aerobic antibacterial agent von Singh, Sheo B, Dayananth, Priya, Balibar, Carl J, Garlisi, Charles G, Lu, Jun, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi, Ha, Sookhee, Young, Katherine

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Synthesis and Antibacterial Activity of Novel Pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic Acid Derivatives Carrying the 3-Cyclopropylaminomethyl-4-substituted-1-pyrrolidinyl Grou... von Asahina, Yoshikazu, Takei, Masaya, Kimura, Tetsuya, Fukuda, Yasumichi

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Stereoselective Synthesis of cis-2-Fluorocyclopropanecarboxylic Acid von Shibue, Taku, Fukuda, Yasumichi

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Efficient synthesis of cyclopropylhydrazine salts von Shibue, Taku, Fukuda, Yasumichi

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Structure activity relationship of N-1 substituted 1,5-naphthyrid-2-one analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial... von Singh, Sheo B., Tan, Christopher M., Kaelin, David, Meinke, Peter T., Miesel, Lynn, Olsen, David B., Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Ohata, Kohei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi

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Synthesis and Structure−Activity Relationship Studies of Highly Potent Novel Oxazolidinone Antibacterials von Komine, Takashi, Kojima, Akihiko, Asahina, Yoshikazu, Saito, Tatsuhiro, Takano, Hisashi, Shibue, Taku, Fukuda, Yasumichi

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In Vitro and In Vivo Characterization of the Novel Oxabicyclooctane-Linked Bacterial Topoisomerase Inhibitor AM-8722, a Selective, Potent Inhibitor of Bacterial DNA Gyrase von Tan, Christopher M, Gill, Charles J, Wu, Jin, Toussaint, Nathalie, Yin, Jingjun, Tsuchiya, Takayuki, Garlisi, Charles G, Kaelin, David, Meinke, Peter T, Miesel, Lynn, Olsen, David B, Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Oohata, Kouhei, Takeuchi, Tomoko, Shibue, Taku, Takano, Hisashi, Nishimura, Akinori, Fukuda, Yasumichi, Singh, Sheo B

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Oxabicyclooctane-Linked Novel Bacterial Topoisomerase Inhibitors as Broad Spectrum Antibacterial Agents von Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Meinke, Peter T, Olsen, David, Lagrutta, Armando, Bradley, Prudence, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Wei, Changqing, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Fukuda, Yasumichi

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Tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of left-hand-side moiety (Part-2) von Singh, Sheo B, Kaelin, David E, Wu, Jin, Miesel, Lynn, Tan, Christopher M, Black, Todd, Nargund, Ravi, Meinke, Peter T, Olsen, David B, Lagrutta, Armando, Lu, Jun, Patel, Sangita, Rickert, Keith W, Smith, Robert F, Soisson, Stephen, Sherer, Edward, Joyce, Leo A, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takano, Hisashi, Shibasaki, Mitsuhito, Yajima, Masanobu, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi

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Structure activity relationship of pyridoxazinone substituted RHS analogs of oxabicyclooctane-linked 1,5-naphthyridinyl novel bacterial topoisomerase inhibitors as broad-spectrum a... von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Yajima, Masanobu, Shibue, Taku, Shibata, Takeshi, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi

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Hydroxy tricyclic 1,5-naphthyridinone oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents-SAR of RHS moiety (Part-3) von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Gill, Charles, Black, Todd, Nargund, Ravi, Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Shibue, Taku, Ohata, Kohei, Takano, Hisashi, Ban, Shizuka, Nishimura, Akinori, Fukuda, Yasumichi

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Structure activity relationship of C-2 ether substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacteri... von Singh, Sheo B., Kaelin, David E., Meinke, Peter T., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Olsen, David B., Lagrutta, Armando, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Takeuchi, Tomoko, Takano, Hisashi, Ohata, Kohei, Kurasaki, Haruaki, Nishimura, Akinori, Shibata, Takeshi, Fukuda, Yasumichi

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Structure activity relationship of substituted 1,5-naphthyridine analogs of oxabicyclooctane-linked novel bacterial topoisomerase inhibitors as broad-spectrum antibacterial agents... von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Shibata, Takeshi, Ohata, Kohei, Takano, Hisashi, Kurasaki, Haruaki, Takeuchi, Tomoko, Nishimura, Akinori, Fukuda, Yasumichi

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Synthetic studies on duocarmycin. 1. Total synthesis of dl-duocarmycin A and its 2-epimer von Fukuda, Yasumichi, Itoh, Yoshio, Nakatani, Kazuhiko, Shiro, Terashima

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Synthetic studies on duocarmycin. 2. Synthesis and cytotoxicity of natural (+)-duocarmycin A and its three possible stereoisomers von Fukuda, Yasumichi, Nakatani, Kazuhiko, Terashima, Shiro

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Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups von Fukuda, Yasumichi, Furuta, Hirosuke, Shiga, Futoshi, Oomori, Yasuo, Kusama, Yoshie, Ebisu, Hiroyuki, Terashima, Shiro

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The novel cyclopropapyrroloindole(CPI) bisalkylators bearing methoxycarbonyl and trifluoromethyl groups von FUKUDA, Y, FURUTA, H, KUSAMA, Y, EBISU, H, OOMORI, Y, TERASHIMA, S

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C1–C2-linker substituted 1,5-naphthyridine analogues of oxabicyclooctane-linked NBTIs as broad-spectrum antibacterial agents (part 7) von Singh, Sheo B., Kaelin, David E., Wu, Jin, Miesel, Lynn, Tan, Christopher M., Meinke, Peter T., Olsen, David B., Lagrutta, Armando, Wei, Changqing, Liao, Yonggang, Peng, Xuanjia, Wang, Xiu, Fukuda, Hideyuki, Kishii, Ryuta, Takei, Masaya, Shibata, Takeshi, Takeuchi, Tomoko, Ohata, Kohei, Nishimura, Akinori, Fukuda, Yasumichi

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Synthesis and cytotoxicity of enantiomeric pairs of duocarmycin a and its 2-epimer von Fukuda, Yasumichi, Nakatani, Kazuhiko, Terashima, Shiro

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