Small-Molecule Kinase Inhibitors for the Treatment of Nononcologic Diseases von Xie, Zhouling, Yang, Xiaoxiao, Duan, Yajun, Han, Jihong, Liao, Chenzhong

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Design, synthesis and anticancer activities of novel dual poly(ADP-ribose) polymerase-1/histone deacetylase-1 inhibitors von Tian, Yongbin, Xie, Zhouling, Liao, Chenzhong

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An Overview of Naphthylimide as Specific Scaffold for New Drug Discovery von Ruan, Wei, Xie, Zhouling, Wang, Ying, Xia, Lulu, Guo, Yuping, Qiao, Dan

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Synthesis and biological evaluation of 6-fluoro-3-phenyl-7-piperazinyl quinolone derivatives as potential topoisomerase I inhibitors von Ge, Raoling, Zhao, Qian, Xie, Zhouling, Lu, Lu, Guo, Qinglong, Li, Zhiyu, Zhao, Li

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Identification of novel PARP-1 inhibitors: Drug design, synthesis and biological evaluation von Xie, Zhouling, Zhou, Youli, Zhao, Wei, Jiao, He, Chen, Yu, Yang, Yong, Li, Zhiyu

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Lycopene inhibits carrageenan-induced thrombi by regulating AKT/FoxO3a and TLR4/NF-κB pathways von Huang, Rong, Liang, Yingquan, Feng, Jiukang, Xie, Zhouling, Li, Qingshan, Chen, Yuanli, Duan, Yajun, Liu, Hui, Zhang, Buchun, Liao, Chenzhong, Yang, Xiaoxiao

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Design, synthesis, and biological evaluation of novel highly selective polo-like kinase 2 inhibitors based on the tetrahydropteridin chemical scaffold von Zhan, Mei-Miao, Yang, Yang, Luo, Jinfeng, Zhang, Xing-Xing, Xiao, Xuan, Li, Shiyu, Cheng, Kai, Xie, Zhouling, Tu, Zhengchao, Liao, Chenzhong

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LX0702, a novel snake venom peptide derivative, inhibits thrombus formation via affecting the binding of fibrinogen with GPIIb/IIIa von Kong, Yi, Wang, Ying, Yang, Wei, Xie, Zhouling, Li, Zhiyu

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Apigenin ameliorates imiquimod-induced psoriasis in C57BL/6J mice by inactivating STAT3 and NF-κB von Meng, Xianshe, Zheng, Shihong, Yin, Zequn, Wang, Xuerui, Yang, Daigang, Zou, Tingfeng, Li, Huaxin, Chen, Yuanli, Liao, Chenzhong, Xie, Zhouling, Fan, Xiaodong, Han, Jihong, Duan, Yajun, Yang, Xiaoxiao

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Lessons Learned from Past Cyclin-Dependent Kinase Drug Discovery Efforts von Xie, Zhouling, Hou, Shuzeng, Yang, Xiaoxiao, Duan, Yajun, Han, Jihong, Wang, Qin, Liao, Chenzhong

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Discovery and development of plasma kallikrein inhibitors for multiple diseases von Xie, Zhouling, Li, Zhen, Shao, Yanruisheng, Liao, Chenzhong

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Selective factor XI/XIa inhibitors: a beacon of hope in anticoagulation therapy von Xie, Zhouling, Wang, Qin, Liao, Chenzhong

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Thiazole-based analogs as potential antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA) and their SAR elucidation von Guo, Jiaojiao, Xie, Zhouling, Ruan, Wei, Tang, Qidong, Qiao, Dan, Zhu, Wufu

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Zinc enzymes in medicinal chemistry von Hou, Rui, He, Yan, Yan, Guangwei, Hou, Shuzeng, Xie, Zhouling, Liao, Chenzhong

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Factor XIa Inhibitors in Anticoagulation Therapy: Recent Advances and Perspectives von Xie, Zhouling, Meng, Zhiwei, Yang, Xiaoxiao, Duan, Yajun, Wang, Qin, Liao, Chenzhong

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Developing polo-like kinase 1 inhibitors von Huang, Xufeng, Xie, Zhouling, Liao, Chenzhong

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Design and synthesis of indoline thiohydantoin derivatives based on enzalutamide as antiproliferative agents against prostate cancer von Zuo, Minzan, Xu, Xi, Xie, Zhouling, Ge, Raoling, Zhang, Ziyu, Li, Zhiyu, Bian, Jinlei

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Discovery of Highly Selective, Potent, Covalent, and Orally Bioavailable Factor XIIa Inhibitors for the Treatment of Thrombo-Inflammation von Meng, Zhiwei, Wang, Shengnan, Chen, Fangrong, Zhang, Zhenzhen, Zhang, Yajing, Yin, Zequn, Duan, Yajun, Zheng, Nan, Wang, Qin, Liao, Chenzhong, Chen, Yuanli, Xie, Zhouling

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Novel 1-(prop-2-yn-1-ylamino)-2,3-dihydro-1H-indene-4-thiol derivatives as potent selective human monoamine oxidase B inhibitors: Design, SAR development, and biological evaluation von Kong, Haiyan, Meng, Xianshe, Hou, Rui, Yang, Xiaoxiao, Han, Jihong, Xie, Zhouling, Duan, Yajun, Liao, Chenzhong

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Targeting the S2 Subsite Enables the Structure-Based Discovery of Novel Highly Selective Factor XIa Inhibitors von Yao, Ningning, Jia, Zhiping, Tian, Yongbin, Hou, Shuzeng, Yang, Xiaoxiao, Han, Jihong, Duan, Yajun, Liao, Chenzhong, Kong, Yi, Xie, Zhouling

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