Synthesis of 35-Deoxy Amphotericin B Methyl Ester: A Strategy for Molecular Editing von Szpilman, Alex M, Cereghetti, Damiano M, Wurtz, Nicholas R, Manthorpe, Jeffrey M, Carreira, Erick M

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Synthesis and Biophysical Studies on 35-Deoxy Amphotericin B Methyl Ester von Szpilman, Alex M., Cereghetti, Damiano M., Manthorpe, Jeffrey M., Wurtz, Nicholas R., Carreira, Erick M.

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Discovery of BMS-986235/LAR-1219: A Potent Formyl Peptide Receptor 2 (FPR2) Selective Agonist for the Prevention of Heart Failure von Asahina, Yoshikazu, Wurtz, Nicholas R, Arakawa, Kazuto, Carson, Nancy, Fujii, Kiyoshi, Fukuchi, Kazunori, Garcia, Ricardo, Hsu, Mei-Yin, Ishiyama, Junichi, Ito, Bruce, Kick, Ellen, Lupisella, John, Matsushima, Shingo, Ohata, Kohei, Ostrowski, Jacek, Saito, Yoshifumi, Tsuda, Kosuke, Villarreal, Francisco, Yamada, Hitomi, Yamaoka, Toshikazu, Wexler, Ruth, Gordon, David, Kohno, Yasushi

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Formyl peptide receptor 2 and heart disease von Lupisella, John A., Shirude, Pravin S., Wurtz, Nicholas R., Garcia, Ricardo A.

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Fmoc Solid Phase Synthesis of Polyamides Containing Pyrrole and Imidazole Amino Acids von Wurtz, Nicholas R, Turner, James M, Baird, Eldon E, Dervan, Peter B

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Atropisomer Control in Macrocyclic Factor VIIa Inhibitors von Glunz, Peter W, Mueller, Luciano, Cheney, Daniel L, Ladziata, Vladimir, Zou, Yan, Wurtz, Nicholas R, Wei, Anzhi, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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Discovery and Optimization of Aryl Piperidinone Ureas as Selective Formyl Peptide Receptor 2 Agonists von Wurtz, Nicholas R, Shirude, Pravin S, Cheney, Daniel L, Lupisella, John A, Chattopadhyay, Amit Kumar, Baligar, Vishweshwaraiah, Seshadri, Balaji, Anjanappa, Prakash, Viet, Andrew, Valente, Meriah N, Hsu, Mei-Yin, Abousleiman, Mojgan, Sarodaya, Sanket, Tagore, Debarati M, Dudhgaonkar, Shailesh, Putlur, Sivaprasad, Dierks, Elizabeth A, Ostrowski, Jacek, Wexler, Ruth R, Garcia, Ricardo, Kick, Ellen K

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Discovery of Heteroaryl Urea Isosteres for Formyl Peptide Receptor 2 Agonists von Wurtz, Nicholas R., Johnson, James A., Viet, Andrew, Shirude, Pravin S., Baligar, Vishweshwaraiah, Madduri, Sudhakara, Cheney, Daniel L., Park, Hyunsoo, Lupisella, John A., Hsu, Mei-Yin, Abousleiman, Mojgan, Galella, Michael A., Aulakh, Darpandeep, Dierks, Elizabeth A., Garcia, Ricardo A., Ostrowski, Jacek, Kick, Ellen K., Wexler, Ruth R.

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Selective FPR2 Agonism Promotes a Proresolution Macrophage Phenotype and Improves Cardiac Structure-Function Post Myocardial Infarction von García, Ricardo A., Lupisella, John A., Ito, Bruce R., Hsu, Mei-Yin, Fernando, Gayani, Carson, Nancy L., Allocco, John J., Ryan, Carol S., Zhang, Rongan, Wang, Zhaoqing, Heroux, Madeleine, Carrier, Marilyn, St.-Onge, Stéphane, Bouvier, Michel, Dudhgaonkar, Shailesh, Nagar, Jignesh, Bustamante-Pozo, Moises M., Garate-Carrillo, Alejandra, Chen, Jian, Ma, Xiuying, Search, Debra J., Dierks, Elizabeth A., Kick, Ellen K., Wexler, Ruth R., Gordon, David A., Ostrowski, Jacek, Wurtz, Nicholas R., Villarreal, Francisco

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Discovery of a Highly Potent, Selective, and Orally Bioavailable Macrocyclic Inhibitor of Blood Coagulation Factor VIIa–Tissue Factor Complex von Zhang, Xiaojun, Glunz, Peter W, Johnson, James A, Jiang, Wen, Jacutin-Porte, Swanee, Ladziata, Vladimir, Zou, Yan, Phillips, Monique S, Wurtz, Nicholas R, Parkhurst, Brandon, Rendina, Alan R, Harper, Timothy M, Cheney, Daniel L, Luettgen, Joseph M, Wong, Pancras C, Seiffert, Dietmar, Wexler, Ruth R, Priestley, E. Scott

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Potent Triazolopyridine Myeloperoxidase Inhibitors von Wurtz, Nicholas R, Viet, Andrew, Shaw, Scott A, Dilger, Andrew, Valente, Meriah N, Khan, Javed A, Jusuf, Sutjano, Narayanan, Rangaraj, Fernando, Gayani, Lo, Fred, Liu, Xiaoqin, Locke, Gregory A, Kopcho, Lisa, Abell, Lynn M, Sleph, Paul, Basso, Michael, Zhao, Lei, Wexler, Ruth R, Duclos, Franck, Kick, Ellen K

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Correction to “Atropisomer Control in Macrocyclic Factor VIIa Inhibitors” von Glunz, Peter W, Mueller, Luciano, Cheney, Daniel L, Ladziata, Vladimir, Zou, Yan, Wurtz, Nicholas R, Wei, Anzhi, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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Discovery of Novel P1 Groups for Coagulation Factor VIIa Inhibition Using Fragment-Based Screening von Cheney, Daniel L, Bozarth, Jeffrey M, Metzler, William J, Morin, Paul E, Mueller, Luciano, Newitt, John A, Nirschl, Alexandra H, Rendina, Alan R, Tamura, James K, Wei, Anzhi, Wen, Xiao, Wurtz, Nicholas R, Seiffert, Dietmar A, Wexler, Ruth R, Priestley, E. Scott

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Neutral macrocyclic factor VIIa inhibitors von Wurtz, Nicholas R., Parkhurst, Brandon L., DeLucca, Indawati, Glunz, Peter W., Jiang, Wen, Zhang, Xiaojun, Cheney, Daniel L., Bozarth, Jeffrey M., Rendina, Alan R., Wei, Anzhi, Harper, Tim, Luettgen, Joseph M., Wu, Yiming, Wong, Pancras C., Seiffert, Dietmar A., Wexler, Ruth R., Priestley, E. Scott

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Preservation of Post-Infarction Cardiac Structure and Function via Long-Term Oral Formyl Peptide Receptor Agonist Treatment von García, Ricardo A., Ito, Bruce R., Lupisella, John A., Carson, Nancy A., Hsu, Mei-Yin, Fernando, Gayani, Heroux, Madeleine, Bouvier, Michel, Dierks, Elizabeth, Kick, Ellen K., Gordon, David A., Chen, Jian, Mintier, Gabe, Carrier, Marilyn, St-Onge, Stéphane, Shah, Himanshu, Towne, Jordan, Bucardo, Marcela Sotelo, Ma, Xiuying, Ryan, Carol S., Wurtz, Nicholas R., Ostrowski, Jacek, Villarreal, Francisco J.

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Molecular Mechanisms of Desensitization Underlying the Differential Effects of Formyl Peptide Receptor 2 Agonists on Cardiac Structure–Function Post Myocardial Infarction von Lupisella, John, St-Onge, Stéphane, Carrier, Marilyn, Cook, Erica M., Wang, Tao, Sum, Chi, Fernando, Gayani, Apgar, Kendra, Zhang, Rongan, Carson, Nancy, Snyder, Bradley J., Ryan, Carol S., Ma, Xiuying, Dierks, Elizabeth A., Little, Sean, Kick, Ellen K., Wurtz, Nicholas R., Bouvier, Michel, Héroux, Madeleine, Garcia, Ricardo A.

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Triazolopyrimidines identified as reversible myeloperoxidase inhibitors von Duclos, Franck, Abell, Lynn M, Harden, David G, Pike, Kristen, Nowak, Kimberly, Locke, Gregory A, Duke, Gerald J, Liu, Xiaoqin, Fernando, Gayani, Shaw, Scott A, Vokits, Benjamin P, Wurtz, Nicholas R, Viet, Andrew, Valente, Meriah N, Stachura, Sylwia, Sleph, Paul, Khan, Javed A, Gao, Ji, Dongre, Ashok R, Zhao, Lei, Wexler, Ruth R, Gordon, David A, Kick, Ellen K

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Discovery of Phenylglycine Lactams as Potent Neutral Factor VIIa Inhibitors von Wurtz, Nicholas R, Parkhurst, Brandon L, Jiang, Wen, DeLucca, Indawati, Zhang, Xiaojun, Ladziata, Vladimir, Cheney, Daniel L, Bozarth, Jeffrey R, Rendina, Alan R, Wei, Anzhi, Luettgen, Joseph M, Wu, Yiming, Wong, Pancras C, Seiffert, Dietmar A, Wexler, Ruth R, Priestley, E. Scott

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Inhibition of major groove DNA binding bZIP proteins by positive patch polyamides von Bremer, Ryan E, Wurtz, Nicholas R, Szewczyk, Jason W, Dervan, Peter B

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Design and Synthesis of Phenylpyrrolidine Phenylglycinamides As Highly Potent and Selective TF-FVIIa Inhibitors von Zhang, Xiaojun, Jiang, Wen, Jacutin-Porte, Swanee, Glunz, Peter W, Zou, Yan, Cheng, Xuhong, Nirschl, Alexandra H, Wurtz, Nicholas R, Luettgen, Joseph M, Rendina, Alan R, Luo, Gang, Harper, Timothy M, Wei, Anzhi, Anumula, Rushith, Cheney, Daniel L, Knabb, Robert M, Wong, Pancras C, Wexler, Ruth R, Priestley, E. Scott

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