Novel tetrahydropyran analogs as dipeptidyl peptidase IV inhibitors: Profile of clinical candidate (2R,3S,5R)-2-(2,5-difluorophenyl)-5-[2-(methylsulfonyl)-2,6-dihydropyrrolo[3,4-c]... von Biftu, Tesfaye, Qian, Xiaoxia, Chen, Ping, Feng, Dennis, Scapin, Giovanna, Gao, Ying-Duo, Cox, Jason, Sinha Roy, Ranabir, Eiermann, George, He, Huabing, Lyons, Kathy, Salituro, Gino, Patel, Sangita, Petrov, Alexander, Xu, Feng, Xu, Shiyao Sherrie, Zhang, Bei, Caldwell, Charles, Wu, Joseph K., Weber, Ann E.

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Structure–activity-relationship of amide and sulfonamide analogs of omarigliptin von Chen, Ping, Feng, Dennis, Qian, Xiaoxia, Apgar, James, Wilkening, Robert, Kuethe, Jeffrey T., Gao, Ying-Duo, Scapin, Giovanna, Cox, Jason, Doss, George, Eiermann, George, He, Huaibing, Li, Xiaohua, Lyons, Kathryn A., Metzger, Joseph, Petrov, Aleksandr, Wu, Joseph K., Xu, Shiyao, Weber, Ann E., Yan, Youwei, Roy, Ranabir Sinha, Biftu, Tesfaye

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Catalytic properties and inhibition of proline-specific dipeptidyl peptidases II, IV and VII von Leiting, Barbara, Pryor, KellyAnn D, Wu, Joseph K, Marsilio, Frank, Patel, Reshma A, Craik, Charles S, Ellman, Jonathan A, Cummings, Richard T, Thornberry, Nancy A

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Discovery of potent and selective phenylalanine based dipeptidyl peptidase IV inhibitors von Xu, Jinyou, Wei, Lan, Mathvink, Robert, He, Jiafang, Park, You-Jung, He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.

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Dipeptidyl peptidase IV inhibition for the treatment of type 2 diabetes : Potential importance of selectivity over dipeptidyl peptidases 8 and 9 von LANKAS, George R, LEITING, Barbara, IPPOLITO, Dawn E, KIM, Dooseop, LYONS, Kathryn A, OK, Hyun O, PATEL, Reshma A, PETROV, Aleksandr N, PRYOR, Kelly Ann, XIAOXIA QIAN, REIGLE, Leah, WOODS, Andrea, ROY, Ranabir Sinha, WU, Joseph K, ZALLER, Dennis, XIAOPING ZHANG, LAN ZHU, WEBER, Ann E, THORNBERRY, Nancy A, EIERMANN, George J, BECONI, Maria G, BIFTU, Tesfaye, CHAN, Chi-Chung, EDMONDSON, Scott, FEENEY, William P, HUAIBING HE

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Towards a More Complete Efficiency Wage Theory von Wu, Joseph S. K., Ho, Chi Pui

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Discovery of potent, selective, and orally bioavailable oxadiazole-based dipeptidyl peptidase IV inhibitors von Xu, Jinyou, Wei, Lan, Mathvink, Robert J., Edmondson, Scott D., Eiermann, George J., He, Huaibing, Leone, Joseph F., Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Patel, Sangita B., Petrov, Aleksandr, Scapin, Giovanna, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.

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The discovery of novel 5,6,5- and 5,5,6-tricyclic pyrrolidines as potent and selective DPP-4 inhibitors von Cox, Jason M., Chu, Hong D., Kuethe, Jeffrey T., Gao, Ying-Duo, Scapin, Giovanna, Eiermann, George, He, Huaibing, Li, Xiaohua, Lyons, Kathryn A., Metzger, Joseph, Petrov, Aleksandr, Wu, Joseph K., Xu, Shiyao, Sinha-Roy, Ranabir, Weber, Ann E., Biftu, Tesfaye

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A comparative study of the binding properties, dipeptidyl peptidase‐4 (DPP‐4) inhibitory activity and glucose‐lowering efficacy of the DPP‐4 inhibitors alogliptin, linagliptin, sax... von Berger, Joel P., SinhaRoy, Ranabir, Pocai, Alessandro, Kelly, Theresa M., Scapin, Giovanna, Gao, Ying‐Duo, Pryor, Kelly Ann D., Wu, Joseph K., Eiermann, George J., Xu, Shiyao S., Zhang, Xiaoping, Tatosian, Daniel A., Weber, Ann E., Thornberry, Nancy A., Carr, Richard D.

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Quantitative easing in an open economy—Not a liquidity but a reserve trap von Herbst, Anthony F., Wu, Joseph S.K., Ho, Chi Pui

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Diastereoselective synthesis and configuration-dependent activity of (3-substituted-cycloalkyl)glycine pyrrolidides and thiazolidides as dipeptidyl peptidase IV inhibitors von ASHTON, Wallace T, HONG DONG, SISCO, Rosemary M, DOSS, George A, LEITING, Barbara, PATEL, Reshma A, WU, Joseph K, MARSILIO, Frank, THOMBERRY, Nancy A, WEBER, Ann E

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Synthesis and evaluation of [(1 R)-1-amino-2-(2,5-difluorophenyl)ethyl]cyclohexanes and 4-[(1 R)-1-amino-2-(2,5-difluorophenyl)ethyl]piperidines as DPP-4 inhibitors von Chen, Ping, Caldwell, Charles G., Ashton, Wallace, Wu, Joseph K., He, Huaibing, Lyons, Kathryn A., Thornberry, Nancy A., Weber, Ann E.

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Substituted piperazines as novel dipeptidyl peptidase IV inhibitors von Brockunier, Linda L., He, Jiafang, Colwell, Lawrence F., Habulihaz, Bahanu, He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Marsilio, Frank, Patel, Reshma A., Teffera, Yohannes, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E., Parmee, Emma R.

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Relationship between risk attitude and economic recovery in optimal growth theory von Herbst, Anthony F., Wu, Joseph S.K., Ho, Chi Pui

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Design, synthesis, and biological evaluation of triazolopiperazine-based β-amino amides as potent, orally active dipeptidyl peptidase IV (DPP-4) inhibitors von Kowalchick, Jennifer E., Leiting, Barbara, Pryor, KellyAnn D., Marsilio, Frank, Wu, Joseph K., He, Huaibing, Lyons, Kathryn A., Eiermann, George J., Petrov, Aleksandr, Scapin, Giovanna, Patel, Reshma A., Thornberry, Nancy A., Weber, Ann E., Kim, Dooseop

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(2S,3S)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-N,N-dimethyl-4-oxo-2-(4-[1,2,4]triazolo[1,5-a]- pyridin-6-ylphenyl)butanamide:  A Selective α-Amino Amide Dipeptidyl Peptidase IV In... von Edmondson, Scott D, Mastracchio, Anthony, Mathvink, Robert J, He, Jiafang, Harper, Bart, Park, You-Jung, Beconi, Maria, Di Salvo, Jerry, Eiermann, George J, He, Huaibing, Leiting, Barbara, Leone, Joseph F, Levorse, Dorothy A, Lyons, Kathryn, Patel, Reshma A, Patel, Sangita B, Petrov, Aleksandr, Scapin, Giovanna, Shang, Jackie, Roy, Ranabir Sinha, Smith, Aaron, Wu, Joseph K, Xu, Shiyao, Zhu, Bing, Thornberry, Nancy A, Weber, Ann E

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Modeling assisted rational design of novel, potent, and selective pyrrolopyrimidine DPP-4 inhibitors von Gao, Ying-Duo, Feng, Dennis, Sheridan, Robert P., Scapin, Giovanna, Patel, Sangita B., Wu, Joseph K., Zhang, Xiaoping, Sinha-Roy, Ranabir, Thornberry, Nancy A., Weber, Ann E., Biftu, Tesfaye

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Fluoroolefins as amide bond mimics in dipeptidyl peptidase IV inhibitors von Edmondson, Scott D., Wei, Lan, Xu, Jinyou, Shang, Jackie, Xu, Shiyao, Pang, Jianmei, Chaudhary, Ashok, Dean, Dennis C., He, Huaibing, Leiting, Barbara, Lyons, Kathryn A., Patel, Reshma A., Patel, Sangita B., Scapin, Giovanna, Wu, Joseph K., Beconi, Maria G., Thornberry, Nancy A., Weber, Ann E.

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Discovery of potent and selective orally bioavailable β-substituted phenylalanine derived dipeptidyl peptidase IV inhibitors von Edmondson, Scott D., Mastracchio, Anthony, Duffy, Joseph L., Eiermann, George J., He, Huaibing, Ita, Ida, Leiting, Barbara, Leone, Joseph F., Lyons, Kathryn A., Makarewicz, Amanda M., Patel, Reshma A., Petrov, Aleksandr, Wu, Joseph K., Thornberry, Nancy A., Weber, Ann E.

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(2R)-4-Oxo-4-[3-(Trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin- 7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-amine:  A Potent, Orally Active Dipeptidyl Peptidase IV Inhib... von Kim, Dooseop, Wang, Liping, Beconi, Maria, Eiermann, George J, Fisher, Michael H, He, Huaibing, Hickey, Gerard J, Kowalchick, Jennifer E, Leiting, Barbara, Lyons, Kathryn, Marsilio, Frank, McCann, Margaret E, Patel, Reshma A, Petrov, Aleksandr, Scapin, Giovanna, Patel, Sangita B, Roy, Ranabir Sinha, Wu, Joseph K, Wyvratt, Matthew J, Zhang, Bei B, Zhu, Lan, Thornberry, Nancy A, Weber, Ann E

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