Choose and Use Your Chemical Probe Wisely to Explore Cancer Biology von Blagg, Julian, Workman, Paul

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Combinatorial drug therapy for cancer in the post-genomic era von Al-Lazikani, Bissan, Banerji, Udai, Workman, Paul

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Inhibitors of cyclin-dependent kinases as cancer therapeutics von Whittaker, Steven R, Mallinger, Aurélie, Workman, Paul, Clarke, Paul A

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Critical Parameters in Targeted Drug Development: The Pharmacological Audit Trail von Banerji, Udai, PhD, Workman, Paul, PhD

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Discovery of small molecule cancer drugs: Successes, challenges and opportunities von Hoelder, Swen, Clarke, Paul A., Workman, Paul

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Drugging PI3K in cancer: refining targets and therapeutic strategies von Yap, Timothy A, Bjerke, Lynn, Clarke, Paul A, Workman, Paul

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The Hsp90 molecular chaperone: an open and shut case for treatment von Pearl, Laurence H, Prodromou, Chrisostomos, Workman, Paul

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Fadraciclib (CYC065), a novel CDK inhibitor, targets key pro-survival and oncogenic pathways in cancer von Frame, Sheelagh, Saladino, Chiara, MacKay, Craig, Atrash, Butrus, Sheldrake, Peter, McDonald, Edward, Clarke, Paul A., Workman, Paul, Blake, David, Zheleva, Daniella

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Maximizing the Therapeutic Potential of HSP90 Inhibitors von Butler, Lisa M, Ferraldeschi, Roberta, Armstrong, Heather K, Centenera, Margaret M, Workman, Paul

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Inhibitors of the heat shock response: Biology and pharmacology von Powers, Marissa V., Workman, Paul

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Dual Targeting of HSC70 and HSP72 Inhibits HSP90 Function and Induces Tumor-Specific Apoptosis von Powers, Marissa V., Clarke, Paul A., Workman, Paul

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The NCI-60 Human Tumor Cell Line Screen: A Catalyst for Progressive Evolution of Models for Discovery and Development of Cancer Drugs von Workman, Paul

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HSP90 inhibition: two-pronged exploitation of cancer dependencies von Travers, Jon, Sharp, Swee, Workman, Paul

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Chemical biology approaches to target validation in cancer von Blagg, Julian, Workman, Paul

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Targeting of multiple signalling pathways by heat shock protein 90 molecular chaperone inhibitors von Powers, Marissa V, Workman, Paul

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Small-molecule targeting of brachyury transcription factor addiction in chordoma von Sharifnia, Tanaz, Wawer, Mathias J., Chen, Ting, Huang, Qing-Yuan, Weir, Barbara A., Sizemore, Ann, Lawlor, Matthew A., Goodale, Amy, Cowley, Glenn S., Vazquez, Francisca, Ott, Christopher J., Francis, Joshua M., Sassi, Slim, Cogswell, Patricia, Sheppard, Hadley E., Zhang, Tinghu, Gray, Nathanael S., Clarke, Paul A., Blagg, Julian, Workman, Paul, Sommer, Josh, Hornicek, Francis, Root, David E., Hahn, William C., Bradner, James E., Wong, Kwok K., Clemons, Paul A., Lin, Charles Y., Kotz, Joanne D., Schreiber, Stuart L.

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ATP-competitive inhibitors block protein kinase recruitment to the Hsp90-Cdc37 system von Polier, Sigrun, Samant, Rahul S, Clarke, Paul A, Workman, Paul, Prodromou, Chrisostomos, Pearl, Laurence H

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Hsp90 molecular chaperone inhibitors: are we there yet? von Neckers, Len, Workman, Paul

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MIR21 Drives Resistance to Heat Shock Protein 90 Inhibition in Cholangiocarcinoma von Lampis, Andrea, Carotenuto, Pietro, Vlachogiannis, Georgios, Cascione, Luciano, Hedayat, Somaieh, Burke, Rosemary, Clarke, Paul, Bosma, Else, Simbolo, Michele, Scarpa, Aldo, Yu, Sijia, Cole, Rebecca, Smyth, Elizabeth, Mateos, Javier Fernández, Begum, Ruwaida, Hezelova, Blanka, Eltahir, Zakaria, Wotherspoon, Andrew, Fotiadis, Nicos, Bali, Maria Antonietta, Nepal, Chirag, Khan, Khurum, Stubbs, Mark, Hahne, Jens C., Gasparini, Pierluigi, Guzzardo, Vincenza, Croce, Carlo M., Eccles, Suzanne, Fassan, Matteo, Cunningham, David, Andersen, Jesper B., Workman, Paul, Valeri, Nicola, Braconi, Chiara

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Drugging the PI3 Kinome: From Chemical Tools to Drugs in the Clinic von WORKMAN, Paul, CLARKE, Paul A, RAYNAUD, Florence I, VAN MONTFORT, Rob L. M

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