Novel Modes of Inhibition of Wild-Type Isocitrate Dehydrogenase 1 (IDH1): Direct Covalent Modification of His315 von Jakob, Clarissa G, Upadhyay, Anup K, Donner, Pamela L, Nicholl, Emily, Addo, Sadiya N, Qiu, Wei, Ling, Christopher, Gopalakrishnan, Sujatha M, Torrent, Maricel, Cepa, Steven P, Shanley, Jason, Shoemaker, Alexander R, Sun, Chaohong C, Vasudevan, Anil, Woller, Kevin R, Shotwell, J. Brad, Shaw, Bailin, Bian, Zhiguo, Hutti, Jessica E

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CRISPR Screen Reveals BRD2/4 Molecular Glue-like Degrader via Recruitment of DCAF16 von Shergalis, Andrea G., Marin, Violeta L., Rhee, David Y., Senaweera, Sameera, McCloud, Rebecca L., Ronau, Judith A., Hutchins, Charles W., McLoughlin, Shaun, Woller, Kevin R., Warder, Scott E., Vasudevan, Anil, Reitsma, Justin M.

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Targeting IRAK3 for Degradation to Enhance IL-12 Pro-inflammatory Cytokine Production von Rowley, Ann, Brown, Brian S., Stofega, Mary, Hoh, Hana, Mathew, Rebecca, Marin, Violeta, Ding, Rong-Xian, McClure, Ryan A., Bittencourt, Fabiola M., Chen, Jun, Gururaja, Tarikere, Kinoshita, Taisei, Wang, Xueqing, Rivkin, Alexey, Woller, Kevin R.

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Quantitative Measurement of Rate of Targeted Protein Degradation von Lynch, Thomas L., Marin, Violeta L., McClure, Ryan A., Phipps, Colin, Ronau, Judith A., Rouhimoghadam, Milad, Adams, Ashley M., Kandi, Soumya, Wolke, Malerie L., Shergalis, Andrea G., Potts, Gregory K., Nacham, Omprakash, Richardson, Paul, Kakavas, Stephan J., Chhor, Gekleng, Jenkins, Gary J., Woller, Kevin R., Warder, Scott E., Vasudevan, Anil, Reitsma, Justin M.

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Singlet Oxygenation/Radical Rearrangement as an Approach to 1,4-Dioxygenated Peroxides:  Asymmetric Total Syntheses of Plakorin and enantio-Chondrillin von Dussault, Patrick H, Woller, Kevin R

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( S) -N-(5-Chlorothiophene-2-sulfonyl)-β,β-diethylalaninol a Notch-1-sparing γ-secretase inhibitor von Cole, Derek C., Stock, Joseph R., Kreft, Anthony F., Antane, Madelene, Aschmies, Suzan H., Atchison, Kevin P., Casebier, David S., Comery, Thomas A., Diamantidis, George, Ellingboe, John W., Harrison, Boyd L., Hu, Yun, Jin, Mei, Kubrak, Dennis M., Lu, Peimin, Mann, Charles W., Martone, Robert L., Moore, William J., Oganesian, Aram, Riddell, David R., Sonnenberg-Reines, June, Sun, Shaiu-Ching, Wagner, Erik, Wang, Zheng, Woller, Kevin R., Xu, Zheng, Zhou, Hua, Jacobsen, J. Steven

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Total Synthesis of the Alkoxydioxines (+)- and (−)-Chondrillin and (+)- and (−)-Plakorin via Singlet Oxygenation/Radical Rearrangement von Dussault, Patrick H, Eary, C. Todd, Woller, Kevin R

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Approaches to Stereoselective Dioxygenation of Alkenes:  Chiral Phosphite Ozonides von Dussault, Patrick H, Woller, Kevin R

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The Reduction of Aryl Diethyl Phosphate Esters with Lithium Di-tert-butylbiphenylide Radical Anion: Aromatic Hydrocarbons via the Deoxygenation of Phenols von Lusch, Michael J., Woller, Kevin R., Keller, Anthony M., Turk, Michael C.

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PYRIMIDINES FOR DEGRADING BRUTON'S TYROSINE KINASE von Jia, Zhaozhong J, Rivkin, Alexey A, Biannic, Berenger, Noey, Elizabeth L, Adams, Ashley M, Mortezaei, Shahab, Katcher, Matthew H, Zablocki, Jeffery A, Okano, Akinori, Burke, Jason P, Jiang, Xingyu, Marin, Violeta L, Mali, Venkat Reddy, Payette, Joshua N, Woller, Kevin R, Bian, Zhiguo, Zhao, Xianrui, Scholz, Spencer O

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NAMPT INHIBITORS von CURTIN, Michael L, WOLLER, Kevin R, VASUDEVAN, Anil

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NOVEL TRICYCLIC COMPOUNDS von FRANK, Kristine E, VOSS, Jeffrey W, ARGIRIADI, Maria A, WISHART, Neil, FIAMENGO, Bryan A, WOLLER, Kevin R, Ericsson, Anna M, GEORGE, Dawn M, STEWART, Kent D, JOSEPHSOHN, Nathan S, FRIEDMAN, Michael M, LI, Biqin C, WALLACE, Grier A, MORYTKO, Michael J, WANG, Lu, CALDERWOOD, David J, GOEDKEN, Eric R

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Anti-Viral Compounds von Sarris, Kathy, Wagaw, Seble H, Hutchins, Charles W, Carroll, William A, Li, Wenke, Randolph, John T, Jinkerson, Tammie K, Patel, Sachin V, Califano, Jean-Christophe C, Krueger, Allan C, Matulenko, Mark A, Betebenner, David A, Liu, Dachun, Tufano, Michael D, Kati, Warren M, Keddy, Ryan G, Flentge, Charles A, Maring, Clarence J, Bellizzi, Mary E, Pratt, John K, Hutchinson, Douglas K, Wagner, Rolf, Caspi, Daniel D, Rockway, Todd W, Donner, Pamela L, DeGoey, David A, Motter, Christopher E, Gao, Yi, Woller, Kevin R, Nelson, Lissa T

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Stereoselective dioxygenation of enoates von DUSSAULT, P. H, WOLLER, K. R, HILIER, M. C

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NOVEL TRICYCLIC COMPOUNDS von LI, Biqin, C, JOSEPHSOHN, Nathan, S, WISHART, Neil, VOSS, Jeffrey, W, MORYTKO, Michael, J, CALDERWOOD, David, J, WALLACE, Grier, A, WOLLER, Kevin, R, ERICSSON, Anna, M, GOEDKEN, Eric, R, ARGIRIADI, Maria, A, GEORGE, Dawn, M, FRANK, Kristine, E, FRIEDMAN, Michael, STEWART, Kent, D, WANG, Lu, FIAMENGO, Bryan, A

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NAMPT And Rock Inhibitors von CURTIN, Michael L, HEYMAN, Howard R, WOLLER, Kevin R, SHAH, Omar J, SWEIS, Ramzi, VASUDEVAN, Anil, SORENSEN, Bryan K, HANSEN, Todd M, CLARK, Richard F, PLIUSHCHEV, Marina A, MICHAELIDES, Michael, TSE, Chris, MACK, Helmut

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NAMPT INHIBITORS von VASUDEVAN, ANIL, CURTIN, MICHAEL L, WOLLER, KEVIN R

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NOVEL TRICYCLIC COMPOUNDS von FRANK, Kristine E, VOSS, Jeffrey W, ARGIRIADI, Maria A, WISHART, Neil, FIAMENGO, Bryan A, WOLLER, Kevin R, GEORGE, Dawn M, STEWART, Kent D, JOSEPHSOHN, Nathan S, FRIEDMAN, Michael M, ERICSSON, Anna M, LI, Biqin C, WALLACE, Grier A, MORYTKO, Michael J, WANG, Lu, CALDERWOOD, David J, GOEDKEN, Eric R

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inibidores de nampt e rock von MARINA A. PLIUSHCHEV, ANIL VASUDEVAN, RICHARD F. CLARK, TODD .M HANSEN, OMAR J. SHAH, CHRIS TSE, HOWARD R. HEYMAN, MICHAEL L. CURTIN, MICHAEL MICHAELIDES, HELMUT MACK, RAMZI SWEIS, BRYAN K. SORENSEN, KEVIN R. WOLLER

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NAMPT INHIBITORS von CURTIN, Michael L, WOLLER, Kevin R, VASUDEVAN, Anil

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