Binding Kinetics and Pathways of Ligands to GPCRs von Strasser, Andrea, Wittmann, Hans-Joachim, Seifert, Roland

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Competitive association binding kinetic assays: a new tool to detect two different binding orientations of a ligand to its target protein under distinct conditions? von Wittmann, Hans-Joachim, Strasser, Andrea

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Binding pathway of histamine to the hH4R, observed by unconstrained molecular dynamics von Wittmann, Hans-Joachim, Strasser, Andrea

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Aminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors and hCB2R Ligands To Combat Neurodegenerative Disorders von Dolles, Dominik, Nimczick, Martin, Scheiner, Matthias, Ramler, Jacqueline, Stadtmüller, Patricia, Sawatzky, Edgar, Drakopoulos, Antonios, Sotriffer, Christoph, Wittmann, Hans-Joachim, Strasser, Andrea, Decker, Michael

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The First Photochromic Affinity Switch for the Human Cannabinoid Receptor 2 von Dolles, Dominik, Strasser, Andrea, Wittmann, Hans‐Joachim, Marinelli, Oliviero, Nabissi, Massimo, Pertwee, Roger G., Decker, Michael

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Cover Picture: Aminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors and hCB2R Ligands To Combat Neurodegenerative Disorders (Che... von Dolles, Dominik, Nimczick, Martin, Scheiner, Matthias, Ramler, Jacqueline, Stadtmüller, Patricia, Sawatzky, Edgar, Drakopoulos, Antonios, Sotriffer, Christoph, Wittmann, Hans-Joachim, Strasser, Andrea, Decker, Michael

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Structure–Activity Relationships and Computational Investigations into the Development of Potent and Balanced Dual-Acting Butyrylcholinesterase Inhibitors and Human Cannabinoid Rec... von Dolles, Dominik, Hoffmann, Matthias, Gunesch, Sandra, Marinelli, Oliviero, Möller, Jan, Santoni, Giorgio, Chatonnet, Arnaud, Lohse, Martin J, Wittmann, Hans-Joachim, Strasser, Andrea, Nabissi, Massimo, Maurice, Tangui, Decker, Michael

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Species-dependent activities of G-protein-coupled receptor ligands: lessons from histamine receptor orthologs von Strasser, Andrea, Wittmann, Hans-Joachim, Buschauer, Armin, Schneider, Erich H, Seifert, Roland

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Conformational Restriction and Enantioseparation Increase Potency and Selectivity of Cyanoguanidine-Type Histamine H4 Receptor Agonists von Geyer, Roland, Nordemann, Uwe, Strasser, Andrea, Wittmann, Hans-Joachim, Buschauer, Armin

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Modulation of GPCRs by monovalent cations and anions von Strasser, Andrea, Wittmann, Hans-Joachim, Schneider, Erich H., Seifert, Roland

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New insights into the cross-linking and degradation mechanism of Diels-Alder hydrogels von Kirchhof, Susanne, Strasser, Andrea, Wittmann, Hans-Joachim, Messmann, Viktoria, Hammer, Nadine, Goepferich, Achim M, Brandl, Ferdinand P

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3D-QSAR CoMFA Study to Predict Orientation of Suprahistaprodifens and Phenoprodifens in the Binding-Pocket of Four Histamine H1-Receptor Species von Straßer, Andrea, Wittmann, Hans-Joachim

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Sodium binding to hH3R and hH4R — a molecular modeling study von Wittmann, Hans-Joachim, Seifert, Roland, Strasser, Andrea

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Dibenzo[b,f][1,4]oxazepines and dibenzo[b,e]oxepines: Influence of the chlorine substitution pattern on the pharmacology at the H1R, H4R, 5-HT2AR and other selected GPCRs von Naporra, Franziska, Gobleder, Susanne, Wittmann, Hans-Joachim, Spindler, Julia, Bodensteiner, Michael, Bernhardt, Günther, Hübner, Harald, Gmeiner, Peter, Elz, Sigurd, Strasser, Andrea

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2,4-Diaminopyrimidines as dual ligands at the histamine H1 and H4 receptor—H1/H4-receptor selectivity von Hammer, Sebastian G., Gobleder, Susanne, Naporra, Franziska, Wittmann, Hans-Joachim, Elz, Sigurd, Heinrich, Markus R., Strasser, Andrea

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Molecular modeling studies give hint for the existence of a symmetric hβ2R-Gαβγ-homodimer von Straßer, Andrea, Wittmann, Hans-Joachim

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Contribution of Binding Enthalpy and Entropy to Affinity of Antagonist and Agonist Binding at Human and Guinea Pig Histamine H1-Receptor von Hans-Joachim Wittmann, Roland Seifert, Andrea Strasser

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Sodium binding to hH3R and hH 4R--a molecular modeling study von Wittmann, Hans-Joachim, Seifert, Roland, Strasser, Andrea

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Pharmacological profile of astemizole-derived compounds at the histamine H1 and H4 receptor—H1/H4 receptor selectivity von Wagner, Eva, Wittmann, Hans-Joachim, Elz, Sigurd, Strasser, Andrea

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Nanofibers Resulting from Cooperative Electrostatic and Hydrophobic Interactions between Peptides and Polyelectrolytes of Opposite Charge von Ferstl, Matthias, Strasser, Andrea, Wittmann, Hans-Joachim, Drechsler, Markus, Rischer, Matthias, Engel, Jürgen, Goepferich, Achim

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