Pharmacological and immunohistochemical characterization of the APJ receptor and its endogenous ligand apelin von Medhurst, Andrew D., Jennings, Carol A., Robbins, Melanie J., Davis, Robert P., Ellis, Catherine, Winborn, Kim Y., Lawrie, Kenneth W. M., Hervieu, Guillaume, Riley, Graham, Bolaky, Jane E., Herrity, Nicole C., Murdock, Paul, Darker, John G.

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Design and Synthesis of trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1H-3-benzazepine (SB-414796): ... von Macdonald, Gregor J, Branch, Clive L, Hadley, Michael S, Johnson, Christopher N, Nash, David J, Smith, Alexander B, Stemp, Geoffrey, Thewlis, Kevin M, Vong, Antonio K. K, Austin, Nigel E, Jeffrey, Phillip, Winborn, Kim Y, Boyfield, Izzy, Hagan, Jim J, Middlemiss, Derek N, Reavill, Charlie, Riley, Graham J, Watson, Jeannette M, Wood, Martyn, Parker, Steve G, Ashby, Charles R

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Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1 von Westaway, Susan M., Thompson, Mervyn, Rami, Harshad K., Stemp, Geoffrey, Trouw, Leontine S., Mitchell, Darren J., Seal, Jon T., Medhurst, Stephen J., Lappin, Sarah C., Biggs, James, Wright, James, Arpino, Sandra, Jerman, Jeffrey C., Cryan, Jennifer E., Holland, Vicky, Winborn, Kim Y., Coleman, Tanya, Stevens, Alexander J., Davis, John B., Gunthorpe, Martin J.

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SAR of biphenyl carboxamide ligands of the human melanin-concentrating hormone receptor 1 (MCH R1): Discovery of antagonist SB-568849 von Witty, David R., Bateson, John H., Hervieu, Guillaume J., Jeffrey, Phillip, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin M., Wilson, Shelagh, Winborn, Kim Y.

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Discovery of potent and stable conformationally constrained analogues of the MCH R1 antagonist SB-568849 von Witty, David R., Bateson, John, Hervieu, Guillaume J., Al-Barazanji, Kamal, Jeffrey, Phillip, Hamprecht, Dieter, Haynes, Andrea, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin, Winborn, Kim Y.

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N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1 von Westaway, Susan M., Chung, Ying-Kit, Davis, John B., Holland, Vicky, Jerman, Jeffrey C., Medhurst, Stephen J., Rami, Harshad K., Stemp, Geoffrey, Stevens, Alexander J., Thompson, Mervyn, Winborn, Kim Y., Wright, James

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Design and Synthesis of trans -3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1 H -3-benzazepine (SB-414796... von Macdonald, Gregor J., Branch, Clive L., Hadley, Michael S., Johnson, Christopher N., Nash, David J., Smith, Alexander B., Stemp, Geoffrey, Thewlis, Kevin M., Vong, Antonio K. K., Austin, Nigel E., Jeffrey, Phillip, Winborn, Kim Y., Boyfield, Izzy, Hagan, Jim J., Middlemiss, Derek N., Reavill, Charlie, Riley, Graham J., Watson, Jeannette M., Wood, Martyn, Parker, Steve G., Ashby, Charles R.

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Design and synthesis of trans-3-2-4-3-(3-(5-methyl-1,2,4-oxadiazolyl))-phenylcarboxamidocyclohexyl ethyl-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine (SB-414796): A potent... von MACDONALD, Gregor J, BRANCH, Clive L, JEFFREY, Phillip, WINBORN, Kim Y, BOYFIELD, Izzy, HAGAN, Jim J, MIDDLEMISS, Derek N, REAVILL, Charlie, RILEY, Graham J, WATSON, Jeannette M, WOOD, Martyn, PARKER, Steve G, HADLEY, Michael S, ASHBY, Charles R, JOHNSON, Christopher N, NASH, David J, SMITH, Alexander B, STEMP, Geoffrey, THEWLIS, Kevin M, VONG, Antonio K. K, AUSTIN, Nigel E

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