Creating and screening natural product libraries von Wilson, Brice A. P, Thornburg, Christopher C, Henrich, Curtis J, Grkovic, Tanja, O'Keefe, Barry R

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Sinularamides A–G, Terpenoid-Derived Spermidine and Spermine Conjugates with Casitas B‑Lineage Lymphoma Proto-Oncogene B (Cbl-b) Inhibitory Activities from a Sinularia sp. Soft Cor... von Jiang, Wei, Wang, Dongdong, Wilson, Brice A. P, Voeller, Donna, Bokesch, Heidi R, Smith, Emily A, Lipkowitz, Stanley, O’Keefe, Barry R, Gustafson, Kirk R

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Recifin A, Initial Example of the Tyr-Lock Peptide Structural Family, Is a Selective Allosteric Inhibitor of Tyrosyl-DNA Phosphodiesterase I von Krumpe, Lauren R. H, Wilson, Brice A. P, Marchand, Christophe, Sunassee, Suthananda N, Bermingham, Alun, Wang, Wenjie, Price, Edmund, Guszczynski, Tad, Kelley, James A, Gustafson, Kirk R, Pommier, Yves, Rosengren, K. Johan, Schroeder, Christina I, O’Keefe, Barry R

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Agelasine Diterpenoids and Cbl-b Inhibitory Ageliferins from the Coralline Demosponge Astrosclera willeyana von Jiang, Wei, Wang, Dongdong, Wilson, Brice A. P., Kang, Unwoo, Bokesch, Heidi R., Smith, Emily A., Wamiru, Antony, Goncharova, Ekaterina I., Voeller, Donna, Lipkowitz, Stanley, O'Keefe, Barry R., Gustafson, Kirk R.

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Suberitamides A-C, Aryl Alkaloids from a Pseudosuberites sp. Marine Sponge that Inhibit Cbl-b Ubiquitin Ligase Activity von Kim, Chang-Kwon, Wang, Dongdong, Wilson, Brice A. P., Sauri, Josep, Voeller, Donna, Lipkowitz, Stanley, O'Keefe, Barry R., Gustafson, Kirk R.

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Secondary Metabolites from the Fungus Dictyosporium sp. and Their MALT1 Inhibitory Activities von Tran, Trong D, Wilson, Brice A. P, Henrich, Curtis J, Staudt, Louis M, Krumpe, Lauren R. H, Smith, Emily A, King, Jarrod, Wendt, Karen L, Stchigel, Alberto M, Miller, Andrew N, Cichewicz, Robert H, O’Keefe, Barry R, Gustafson, Kirk R

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Rare Caulamidine Hexacyclic Alkaloids from the Marine Ascidian Polyandrocarpa sp von Tian, Xiangrong, Wang, Dongdong, Jiang, Wei, Bokesch, Heidi R., Wilson, Brice A. P., O’Keefe, Barry R., Gustafson, Kirk R.

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Photochemical Dimerization of Plakinidine B Leads to Potent Inhibition of the E3 Ubiquitin-Protein Ligase CBL‑B von Khong, Quan T., Li, Donghao, Wilson, Brice A. P., Ranguelova, Kalina, Dalilian, Masoumeh, Smith, Emily A., Wamiru, Antony, Goncharova, Ekaterina I., Grkovic, Tanja, Voeller, Donna, Lipkowitz, Stanley, Schnermann, Martin J., O’Keefe, Barry R., Du, Lin

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Discovery and Synthesis of a Naturally Derived Protein Kinase Inhibitor that Selectively Inhibits Distinct Classes of Serine/Threonine Kinases von Du, Lin, Wilson, Brice A. P., Li, Ning, Shah, Rohan, Dalilian, Masoumeh, Wang, Dongdong, Smith, Emily A., Wamiru, Antony, Goncharova, Ekaterina I., Zhang, Ping, O’Keefe, Barry R.

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Discovery and Characterization of a Biologically Active Non–ATP-Competitive p38 MAP Kinase Inhibitor von Wilson, Brice A.P., Alam, Muhammad S., Guszczynski, Tad, Jakob, Michal, Shenoy, Shilpa R., Mitchell, Carter A., Goncharova, Ekaterina I., Evans, Jason R., Wipf, Peter, Liu, Gang, Ashwell, Jonathan D., O’Keefe, Barry R.

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Acroamine A, a 2‑Amino Adenine Alkaloid from the Marine Soft Coral Acrozoanthus australiae and Its Semisynthetic Derivatives That Inhibit cAMP-Dependent Protein Kinase A Catalytic... von Senadeera, Sarath P. D., Wang, Dongdong, Wilson, Brice A. P., Smith, Emily A., Wamiru, Antony, Martinez Fiesco, Juliana A., Du, Lin, Zhang, Ping, O’Keefe, Barry R., Beutler, John A.

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Structure elucidation and absolute configuration of metabolites from the soil-derived fungus Dictyosporium digitatum using spectroscopic and computational methods von Tran, Trong D., Wilson, Brice A.P., Henrich, Curtis J., Wendt, Karen L., King, Jarrod, Cichewicz, Robert H., Stchigel, Alberto M., Miller, Andrew N., O'Keefe, Barry R., Gustafson, Kirk R.

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Biochemical Discovery, Intracellular Evaluation, and Crystallographic Characterization of Synthetic and Natural Product Adenosine 3′,5′-Cyclic Monophosphate-Dependent Protein Kinas... von Wilson, Brice A. P., Li, Ning, Martinez Fiesco, Juliana A., Dalilian, Masoumeh, Wang, Dongdong, Smith, Emily A., Wamiru, Antony, Shah, Rohan, Goncharova, Ekaterina I., Beutler, John A., Grkovic, Tanja, Zhang, Ping, O’Keefe, Barry R.

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High-throughput screen identifies novel inhibitors of cancer biomarker α-methylacyl coenzyme A racemase (AMACR/P504S) von Wilson, Brice A P, Wang, Haofan, Nacev, Benjamin A, Mease, Ronnie C, Liu, Jun O, Pomper, Martin G, Isaacs, William B

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In Vitro Ubiquitination Platform Identifies Methyl Ellipticiniums as Ubiquitin Ligase Inhibitors von Wilson, Brice A.P., Voeller, Donna, Smith, Emily A., Wamiru, Antony, Goncharova, Ekaterina I., Liu, Gang, Lipkowitz, Stanley, O’Keefe, Barry R.

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Resolving the fibrotic niche of human liver cirrhosis at single-cell level von Ramachandran, P., Dobie, R., Wilson-Kanamori, J. R., Dora, E. F., Henderson, B. E. P., Luu, N. T., Portman, J. R., Matchett, K. P., Brice, M., Marwick, J. A., Taylor, R. S., Efremova, M., Vento-Tormo, R., Carragher, N. O., Kendall, T. J., Fallowfield, J. A., Harrison, E. M., Mole, D. J., Wigmore, S. J., Newsome, P. N., Weston, C. J., Iredale, J. P., Tacke, F., Pollard, J. W., Ponting, C. P., Marioni, J. C., Teichmann, S. A., Henderson, N. C.

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Multifunctional opioid receptor agonism and antagonism by a novel macrocyclic tetrapeptide prevents reinstatement of morphine‐seeking behaviour von Brice‐Tutt, Ariana C., Wilson, Lisa L., Eans, Shainnel O., Stacy, Heather M., Simons, Chloe A., Simpson, Grant G., Coleman, Jeremy S., Ferracane, Michael J., Aldrich, Jane V., McLaughlin, Jay P.

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Interleukin-27 Regulates the Function of the Gastrointestinal Epithelial Barrier in a Human Tissue-Derived Organoid Model von Brice, Daniel P, Murray, Graeme I, Wilson, Heather M, Porter, Ross J, Berry, Susan, Durum, Scott K, McLean, Mairi H

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Multimodal decoding of human liver regeneration von Matchett, K. P., Wilson-Kanamori, J. R., Portman, J. R., Kapourani, C. A., Fercoq, F., May, S., Zajdel, E., Beltran, M., Sutherland, E. F., Mackey, J. B. G., Brice, M., Wilson, G. C., Wallace, S. J., Kitto, L., Younger, N. T., Dobie, R., Mole, D. J., Oniscu, G. C., Wigmore, S. J., Ramachandran, P., Vallejos, C. A., Carragher, N. O., Saeidinejad, M. M., Quaglia, A., Jalan, R., Simpson, K. J., Kendall, T. J., Rule, J. A., Lee, W. M., Hoare, M., Weston, C. J., Marioni, J. C., Teichmann, S. A., Bird, T. G., Carlin, L. M., Henderson, N. C.

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Lyophilized Kratom Tea as a Therapeutic Option for Opioid Dependence von Wilson, Lisa L., Harris, Hannah M., Eans, Shainnel O., Brice-Tutt, Ariana C., Cirino, Thomas J., Stacy, Heather M., Simons, Chloe A., León, Francisco, Sharma, Abhisheak, Boyer, Edward W., Avery, Bonnie A., McLaughlin, Jay P., McCurdy, Christopher R.

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