Agouti protein is an antagonist of the melanocyte-stimulating-hormone receptor von Lu, Dongsi, Willard, Derril, Patel, Indravadan R, Kadwell, Sue, Overton, Laurie, Kost, Tom, Luther, Michael, Chen, Wenbiao, Woychik, Richard P, Wilkison, William O, Cone, Roger D

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Design of Potent, Selective, and Orally Bioavailable Inhibitors of Cysteine Protease Cathepsin K von Tavares, Francis X, Boncek, Virginia, Deaton, David N, Hassell, Anne M, Long, Stacey T, Miller, Aaron B, Payne, Alan A, Miller, Larry R, Shewchuk, Lisa M, Wells-Knecht, Kevin, Willard, Derril H, Wright, Lois L, Zhou, Hui-Qiang

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Acyclic cyanamide-based inhibitors of cathepsin K von Barrett, David G., Deaton, David N., Hassell, Anne M., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Shewchuk, Lisa M., Willard, Derril H., Wright, Lois L.

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Novel and potent cyclic cyanamide-based cathepsin K inhibitors von Deaton, David N., Hassell, Anne M., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Shewchuk, Lisa M., Tavares, Francis X., Willard, Derril H., Wright, Lois L.

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Melanocortin receptor-mediated mobilization of intracellular free calcium in HEK293 cells von MOUNTJOY, KATHLEEN G, KONG, PHILIP L, TAYLOR, JOHN A, WILLARD, DERRIL H, WILKISON, WILLIAM O

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Semicarbazone-based inhibitors of cathepsin K, are they prodrugs for aldehyde inhibitors? von Adkison, Kim K., Barrett, David G., Deaton, David N., Gampe, Robert T., Hassell, Anne M., Long, Stacey T., McFadyen, Robert B., Miller, Aaron B., Miller, Larry R., Payne, J. Alan, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.

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Agouti structure and function: characterization of a potent .alpha.-melanocyte stimulating hormone receptor antagonist von Willard, Derril H, Bodnar, Wanda, Harris, Cole, Kiefer, Laura, Nichols, James S, Blanchard, Steven, Hoffman, Christine, Moyer, Mary, Burkhart, William

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Hydration Changes Implicated in the Remarkable Temperature-Dependent Membrane Permeation of Cyclosporin A von Augustijns, Patrick F, Brown, Stephen C, Willard, Derril H, Consler, Thomas G, Annaert, Pieter P, Hendren, R. Wayne, Bradshaw, Timothy P

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Novel, potent P2–P3 pyrrolidine derivatives of ketoamide-based cathepsin K inhibitors von Barrett, David G., Catalano, John G., Deaton, David N., Hassell, Anne M., Long, Stacey T., Miller, Aaron B., Miller, Larry R., Ray, John A., Samano, Vicente, Shewchuk, Lisa M., Wells-Knecht, Kevin J., Willard, Derril H., Wright, Lois L.

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Agouti Antagonism of Melanocortin-4 Receptor: Greater Effect with Desacetyl-α-Melanocyte-Stimulating Hormone (MSH) than withα -MSH von Mountjoy, Kathleen G, Willard, Derril H, Wilkison, William O

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Functional Dissection of Osteoprotegerin and Its Interaction with Receptor Activator of NF-κB Ligand von Schneeweis, Lumelle A., Willard, Derril, Milla, Marcos E.

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P2-P3 conformationally constrained ketoamide-based inhibitors of cathepsin K von BARRETT, David G, BONCEK, Virginia M, PAYNE, J. Alan, RAY, John A, SAMANO, Vicente, SHEWCHUK, Lisa M, TAVARES, Francis X, WELLS-KNECHT, Kevin J, WILLARD, Derril H, WRIGHT, Lois L, ZHOU, Hui-Qiang Q, CATALANO, John G, DEATON, David N, HASSELL, Anne M, JURGENSEN, Cynthia H, LONG, Stacey T, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R

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Potent and selective P2-P3 ketoamide inhibitors of cathepsin K with good pharmacokinetic properties via favorable P1', P1, and/or P3 substitutions von BARRETT, David G, CATALANO, John G, WRIGHT, Lois L, DEATON, David N, HASSELL, Anne M, LONG, Stacey T, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WELLS-KNECHT, Kevin J, WILLARD, Derril H

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Exploration of the P1 SAR of aldehyde cathepsin K inhibitors von CATALANO, John G, DEATON, David N, FURFINE, Eric S, HASSELL, Annie M, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R, SHEWCHUK, Lisa M, WILLARD, Derril H, WRIGHT, Lois L

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Human Recombinant Phosphodiesterase 4B2B Binds (R)-Rolipram at a Single Site with Two Affinities von Rocque, Warren J, Tian, Gaochao, Wiseman, Jeffrey S, Holmes, William D, Zajac-Thompson, Irene, Willard, Derril H, Patel, Indravaden R, Wisely, G. Bruce, Clay, William C, Kadwell, Sue H, Hoffman, Christine R, Luther, Michael A

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Mutations in the Carboxyl Terminus of the Agouti Protein Decrease Agouti Inhibition of Ligand Binding to the Melanocortin Receptors von Kiefer, Laura L, Ittoop, Olivia R. R, Bunce, Keith, Truesdale, Anne T, Willard, Derril H, Nichols, James S, Blanchard, Steven G, Mountjoy, Kathleen, Chen, Wen-Ji, Wilkison, William O

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Solution Studies of Recombinant Human Stromal-Cell-Derived Factor-1 von Holmes, William D., Consler, Thomas G., Dallas, Walter S., Rocque, Warren J., Willard, Derril H.

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Cloning of a disintegrin metalloproteinase that processes precursor tumour-necrosis factor-α von Moss, Marcia L, Jin, S.-L. Catherine, Milla, Marcos E, Burkhart, William, Carter, H. Luke, Chen, Wen-Ji, Clay, William C, Didsbury, John R, Hassler, Daniel, Hoffman, Christine R, Kost, Thomas A, Lambert, Millard H, Leesnitzer, M. Anthony, McCauley, Philip, McGeehan, Gerard, Mitchell, Justin, Moyer, Mary, Pahel, Gregory, Rocque, Warren, Overton, Laurie K, Schoenen, Frank, Seaton, Theresa, Su, Jui-Lan, Warner, Janet, Willard, Derril, Becherer, J. David

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Exploration of the P2-P3 SAR of aldehyde cathepsin K inhibitors von BORES, Eric E, DEATON, David N, WRIGHT, Lois L, HASSELL, Anne M, MCFADYEN, Robert B, MILLER, Aaron B, MILLER, Larry R, PAULICK, Margot G, SHEWCHUK, Lisa M, THOMPSON, James B, WILLARD, Derril H

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Functional Dissection of Osteoprotegerin and Its Interaction with Receptor Activator of NF-κB Ligand von Lumelle A. Schneeweis, Derril Willard, Marcos E. Milla

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