Development of Highly Potent Inhibitors of Ras Farnesyltransferase Possessing Cellular and in Vivo Activity von Leftheris, Katerina, Kline, Toni, Vite, Gregory D, Cho, Young H, Bhide, Rajeev S, Patel, Dinesh V, Patel, Manorama M, Schmidt, Robert J, Weller, Harold N, Andahazy, Mary L, Carboni, Joan M, Gullo-Brown, Johnni L, Lee, Francis Y. F, Ricca, Carol, Rose, William C, Yan, Ning, Barbacid, Mariano, Hunt, John T, Meyers, Chester A, Seizinger, Bernd R, Zahler, Robert, Manne, Veeraswamy

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Quinoxaline N-oxide containing potent angiotensin II receptor antagonists: synthesis, biological properties, and structure-activity relationships von Kim, Kyoung Soon, Qian, Ligang, Bird, J. Eileen, Dickinson, Kenneth E. J, Moreland, Suzanne, Schaeffer, Thomas R, Waldron, Thomas L, Delaney, Carol L, Weller, Harold N, Miller, Arthur V

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Phosphinyl acid-based bisubstrate analog inhibitors of ras farnesyl protein transferase von PATEL, D. V, GORDON, E. M, RICCA, C, ROBINSON, S, SEIZINGER, B. R, TUOMARI, A. V, MANNE, V, SCHMIDT, R. J, WELLER, H. N, YOUNG, M. G, ZAHLER, R, BARBACID, M, CARBONI, J. M, GULLO-BROWN, J. L, HUNIHAN, L

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A high-throughput bioanalytical platform using automated infusion for tandem mass spectrometric method optimization and its application in a metabolic stability screen von Kieltyka, Kasia, Zhang, Jun, Li, Shu, Vath, Marianne, Baglieri, Chris, Ferraro, Cheryl, Zvyaga, Tatyana A., Drexler, Dieter M., Weller, Harold N., Shou, Wilson Z.

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Purification of combinatorial libraries von Weller, H N

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High throughput analysis and purification in support of automated parallel synthesis von Weller, H N, Young, M G, Michalczyk, S J, Reitnauer, G H, Cooley, R S, Rahn, P C, Loyd, D J, Fiore, D, Fischman, S J

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Ketomethyldipeptides I. A new class of angiotensin converting enzyme inhibitors von Natarajan, S., Gordon, E.M., Sabo, E.F., Godfrey, J.D., Weller, H.N., Pluščec, Jelka, Rom, M.B., Cushman, D.W.

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Ketomethyldipeptides II. Effect of modifications of the α-aminoketone portion on inhibition of angiotensin converting enzyme von Gordon, E.M., Natarajan, S., Pluščec, Jelka, Weller, H.N., Godfrey, J.D., Rom, M.B., Sabo, E.F., Engebrecht, J., Cushman, D.W.

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Design of conformationally constrained angiotensin-converting enzyme inhibitors von Weller, Harold N., Gordon, Eric M., Rom, Mary Beth, Pluščec, Jelka

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Rapid vinyl shifts in spiro[4.4]polyenes: verification of the rate-determining step and the identity of the migrating group von Semmelhack, M. F, Weller, H. N, Clardy, Jon

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Dihydropyrimidine angiotensin II receptor antagonists von Atwal, Karnail S, Ahmed, Syed Z, Bird, J. Eileen, Delaney, Carol L, Dickinson, Kenneth E. J, Ferrara, Francis N, Hedberg, Anders, Miller, Arthur V, Moreland, Suzanne

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Diol sulfonamides: A potent and novel class of inhibitors of human renin von Poss, Michael A., Reid, Joyce A., Free, Charles A., Rogers, W.Lynn, Weber, Helen, Ryono, Denis E., Dejneka, Tamara, DeForrest, Jack M., Waldron, Thomas L., Brittain, Russell J., Weller, Harold N., Cimarusti, Maria P., Petrillo, Edward W.

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Pharmacology of novel imidazole alcohol inhibitors of primate renin von DeForrest, Jack M, Waldron, Thomas L, Oehl, Robert S, Scalese, Robert J, Free, Charles A, Weller, Harold N, Ryono, Denis E

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Ketomethylureas. A New Class of Angiotensin Converting Enzyme Inhibitors von Natarajan, S., Gordon, E. M., Sabo, E. F., Godfrey, J. D., Weller, H. N., Pluscec, Jelka, Rom, M. B., Engebrecht, J., Cushman, D. W., Deforrest, J. M., Powell, J.

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Thermal rearrangements of spiro[4.4]nonapolyenes. Unusually rapid 1,5-vinyl migration von Semmelhack, M. F., Weller, H. N., Foos, J. S.

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Peptidomimetic Synthesis: A Novel, Highly Stereoselective Route to Substituted Freidinger Lactams von Robl, Jeffrey A, Cimarusti, Maria P, Simpkins, Ligaya M, Weller, Harold N, Pan, Yolanda Y, Malley, Mary, DiMarco, John D

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Design of tripeptide modeled inhibitors of angiotensin-converting enzyme: Studies on the role of the N-terminal acylamino group von Gordon, E.M., Godfrey, J.D., Weller, H.N., Natarajan, S., Pluščec, Jelka, Rom, M.B., Niemela, K., Sabo, E.F., Cushman, D.W.

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Cyclic (Hydroxyphosphinyl)Acyl Dipeptides: A New Class of Angiotensin Converting Enzyme Inhibitors von Weller, Harold N., Rom, Mary Beth

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PRESTRESSED CONCRETE PILES von Weller, N. H. E.

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Benzothiadiazine dioxides: A new class of potent angiotensin-II (AT 1) receptor antagonists von Weller, Harold N., Miller, Arthur V., Moquin, Robert V., Dickinson, Kenneth E.J., Hedberg, S.Anders, Moreland, Suzanne, Cohen, Robert B., Delaney, Carol L., Skwish, Stephen, Williams, Sharon

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