Nonpeptide oxytocin antagonists: Analogs of L-371,257 with improved potency von Williams, Peter D., Bock, Mark G., Evans, Ben E., Freidinger, Roger M., Gallicchio, Steven N., Guidotti, Maribeth T., Jacobson, Marlene A., Kuo, Michelle S., Levy, Michelle R., Lis, Edward V., Michelson, Stuart R., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Salvatore, Christopher, Stauffer, Kenneth J., Woyden, Carla J.

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Nonpeptide oxytocin antagonists: Potent, orally bioavailable analogs of L-371,257 containing A 1- R-(pyridyl)ethyl ether terminus von Kuo, Michelle S., Bock, Mark G., Freidinger, Roger M., Guidotti, Maribeth T., Lis, Edward V., Pawluczyk, Joseph M., Perlow, Debra S., Pettibone, Douglas J., Quigley, Amy G., Reiss, Duane R., Williams, Peter D., Woyden, Carla J.

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Development of Orally Active Oxytocin Antagonists:  Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d... von Bell, Ian M, Erb, Jill M, Freidinger, Roger M, Gallicchio, Steven N, Guare, James P, Guidotti, Maribeth T, Halpin, Rita A, Hobbs, Doug W, Homnick, Carl F, Kuo, Michelle S, Lis, Edward V, Mathre, David J, Michelson, Stuart R, Pawluczyk, Joseph M, Pettibone, Douglas J, Reiss, Duane R, Vickers, Stanley, Williams, Peter D, Woyden, Carla J

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L-368,899, a potent orally active oxytocin antagonist for potential use in preterm labor von Pettibone, D. J., Clineschmidt, B. V., Guidotti, M. T., Lis, E. V., Reiss, D. R., Woyden, C. J., Bock, M. G., Evans, B. E., Freidinger, R. M., Hobbs, D. W., Veber, D. F., Williams, P. D., Chiu, S.-H. L., Thompson, K. L., Schorn, T. W., Siegl, P. K. S., Kaufman, M. J., Cukierski, M. A., Haluska, G. J., Cook, M. J., Novy, M. J.

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Cloning and Expression of the Rhesus Monkey Oxytocin Receptor von Salvatore, Christopher A., Woyden, Carla J., Guidotti, Maribeth T., Pettibone, Douglas J., Jacobson, Marlene A.

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Identification of functional oxytocin receptors in lactating rat mammary gland in vitro von PETTIBONE, D. J, WOYDEN, C. J, TOTARO, J. A

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1-{1-[4-[(N-acetyl-4-piperidinyl)oxy]-2-methoxybenzoyl]piperidin-4-yl}-4H-3,1-benzoxazin-2(1H)-one (L-371,257) : a new, orally bioavailable, non-peptide oxytocin antagonist von WILLIAMS, P. D, CLINESCHMIDT, B. V, WOYDEN, C. J, ERB, J. M, FREIDINGER, R. M, GUIDOTTI, M. T, LIS, E. V, PAWLUCZYK, J. M, PETTIBONE, D. J, REISS, D. R, VEBER, D. F

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Radioligand binding studies reveal marked species differences in the vasopressin V1 receptor of rat, rhesus and human tissues von Pettibone, D J, Kishel, M T, Woyden, C J, Clineschmidt, B V, Bock, M G, Freidinger, R M, Veber, D F, Williams, P D

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Development of orally active oxytocin antagonists : Studies on 1-(1-{4-[1-(2-methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2-methoxybenzo yl}piperidin-4-yl)-1,4-dihydrobenz[d... von BELL, I. M, ERB, J. M, LIS, E. V, MATHRE, D. J, MICHELSON, S. R, PAWLUCZYK, J. M, PETTIBONE, D. J, REISS, D. R, VICKERS, S, WILLIAMS, P. D, WOYDEN, C. J, FREIDINGER, R. M, GALLICCHIO, S. N, GUARE, J. P, GUIDOTTI, M. T, HALPIN, R. A, HOBBS, D. W, HOMNICK, C. F, KUO, M. S

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RADIOLIGAND BINDING-STUDIES REVEAL MARKED SPECIES-DIFFERENCES IN THE VASOPRESSIN-V(1) RECEPTOR OF RAT, RHESUS AND HUMAN TISSUES von PETTIBONE, DJ, KISHEL, MT, WOYDEN, CJ, CLINESCHMIDT, BV, BOCK, MG, FREIDINGER, RM, VEBER, DF, WILLIAMS, PD

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Radioligand binding studies reveal marked species differences in the vasopressin V sub(1) receptor of rat, rhesus and human tissues von Pettibone, D J, Kishel, M T, Woyden, C J, Clineschmidt, B V, Bock, M G, Freidinger, R M, Veber, D F, Williams, P D

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Radioligand binding studies reveal marked species differences in the vasoprressin V1 receptor of rat, rhesus and human tissues von PETTIBONE, D. J, KISHEL, M. T, WOYDEN, C. J, CLINESCHMIDT, B. V, BOCK, M. G, FREINDINGER, R. M, VEBER, D. F, WILLIAMS, P. D

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Preparation and evaluation of 1,3-diaminocyclopentane-linked dihydropyrimidinone derivatives as selective α1a-Receptor antagonists von BARROW, J. C, GLASS, K. L, SELNICK, H. G, FREIDINGER, R. M, CHANG, R. S. L, O'MALLEY, S. S, WOYDEN, C

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Preparation and evaluation of 1,3-diaminocyclopentane-linked dihydropyrimidinone derivatives as selective alpha1a-receptor antagonists von Barrow, J C, Glass, K L, Selnick, H G, Freidinger, R M, Chang, R S, O'Malley, S S, Woyden, C

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