3-Oxoisoxazole-2(3H)-carboxamides and isoxazol-3-yl carbamates: Resistance-breaking acetylcholinesterase inhibitors targeting the malaria mosquito, Anopheles gambiae von Verma, Astha, Wong, Dawn M., Islam, Rafique, Tong, Fan, Ghavami, Maryam, Mutunga, James M., Slebodnick, Carla, Li, Jianyong, Viayna, Elisabet, Lam, Polo C.-H., Totrov, Maxim M., Bloomquist, Jeffrey R., Carlier, Paul R.

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Select small core structure carbamates exhibit high contact toxicity to "carbamate-resistant" strain malaria mosquitoes, Anopheles gambiae (Akron) von Wong, Dawn M, Li, Jianyong, Chen, Qiao-Hong, Han, Qian, Mutunga, James M, Wysinski, Ania, Anderson, Troy D, Ding, Haizhen, Carpenetti, Tiffany L, Verma, Astha, Islam, Rafique, Paulson, Sally L, Lam, Polo C-H, Totrov, Maxim, Bloomquist, Jeffrey R, Carlier, Paul R

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Bivalent Carbamates as Novel Control Agents of the Malaria Mosquito, Anopheles gambiae von Mutunga, James M, Chen, Qiao-Hong, Wong, Dawn M, Lam, Polo C-H, Li, Jianyong, Totrov, Maxim M, Gross, Aaron D, Carlier, Paul R, Bloomquist, Jeffrey R

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Difluoromethyl ketones: Potent inhibitors of wild type and carbamate-insensitive G119S mutant Anopheles gambiae acetylcholinesterase von Camerino, Eugene, Wong, Dawn M., Tong, Fan, Körber, Florian, Gross, Aaron D., Islam, Rafique, Viayna, Elisabet, Mutunga, James M., Li, Jianyong, Totrov, Maxim M., Bloomquist, Jeffrey R., Carlier, Paul R.

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Complexes of Alkylene-Linked Tacrine Dimers with Torpedo californica Acetylcholinesterase:  Binding of Bis(5)-tacrine Produces a Dramatic Rearrangement in the Active-Site Gorge von RYDBERG, Edwin H., BRUMSHTEIN, Boris, GREENBLATT, Harry M., WONG, Dawn M., SHAYA, David, WILLIAMS, Larry D., CARLIER, Paul R., PANG, Yuan-Ping, SILMAN, Israel, SUSSMAN, Joel L.

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Crystal structure of acetylcholinesterase catalytic subunits of the malaria vector Anopheles gambiae von Han, Qian, Wong, Dawn M., Robinson, Howard, Ding, Haizhen, Lam, Polo C. H., Totrov, Maxim M., Carlier, Paul R., Li, Jianyong

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Mosquito Acetylcholinesterase as a Target for Novel Phenyl-Substituted Carbamates von Mutunga, James M, Ma, Ming, Chen, Qiao-Hong, Hartsel, Joshua A, Wong, Dawn M, Ding, Sha, Totrov, Max, Carlier, Paul R, Bloomquist, Jeffrey R

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Re-engineering aryl methylcarbamates to confer high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase von Hartsel, Joshua A., Wong, Dawn M., Mutunga, James M., Ma, Ming, Anderson, Troy D., Wysinski, Ania, Islam, Rafique, Wong, Eric A., Paulson, Sally L., Li, Jianyong, Lam, Polo C.H., Totrov, Maxim M., Bloomquist, Jeffrey R., Carlier, Paul R.

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Carbamate and pyrethroid resistance in the akron strain of Anopheles gambiae von Mutunga, James M, Anderson, Troy D, Craft, Derek T, Gross, Aaron D, Swale, Daniel R, Tong, Fan, Wong, Dawn M, Carlier, Paul R, Bloomquist, Jeffrey R

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Select β- and γ-branched 1-alkylpyrazol-4-yl methylcarbamates exhibit high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase von Carlier, Paul R., Chen, Qiao-Hong, Verma, Astha, Wong, Dawn M., Mutunga, James M., Müller, Jasmin, Islam, Rafique, Shimozono, Alex M., Tong, Fan, Li, Jianyong, Totrov, Max, Bloomquist, Jeffrey R.

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Catalytic Asymmetric Synthesis of Protected Tryptophan Regioisomers von Carlier, Paul R, Lam, Polo C.-H, Wong, Dawn M

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Towards a species-selective acetylcholinesterase inhibitor to control the mosquito vector of malaria, Anopheles gambiae von Carlier, Paul R., Anderson, Troy D., Wong, Dawn M., Hsu, Danny C., Hartsel, Joshua, Ma, Ming, Wong, Eric A., Choudhury, Ranginee, Lam, Polo C.-H., Totrov, Maxim M., Bloomquist, Jeffrey R.

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Aryl methylcarbamates: Potency and selectivity towards wild-type and carbamate-insensitive (G119S) Anopheles gambiae acetylcholinesterase, and toxicity to G3 strain An. gambiae von Wong, Dawn M., Li, Jianyong, Lam, Polo C.H., Hartsel, Joshua A., Mutunga, James M., Totrov, Maxim, Bloomquist, Jeffrey R., Carlier, Paul R.

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Acetylcholinesterase Complexed with Bivalent Ligands Related to Huperzine A:  Experimental Evidence for Species-Dependent Protein−Ligand Complementarity von Wong, Dawn M, Greenblatt, Harry M, Dvir, Hay, Carlier, Paul R, Han, Yi-Fan, Pang, Yuan-Ping, Silman, Israel, Sussman, Joel L

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Crystal Packing Mediates Enantioselective Ligand Recognition at the Peripheral Site of Acetylcholinesterase von Haviv, Haim, Wong, Dawn M, Greenblatt, Harry M, Carlier, Paul R, Pang, Yuan-Ping, Silman, Israel, Sussman, Joel L

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NEUROTOXICOLOGY OF bis(n)-TACRINES ON Blattella germanica AND Drosophila melanogaster ACETYLCHOLINESTERASE von Mutunga, James M., Boina, Dhana Raj, Anderson, Troy D., Bloomquist, Jeffrey R., Carlier, Paul R., Wong, Dawn M., Lam, Polo C.-H., Totrov, Maxim. M.

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Complexes of Alkylene-Linked Tacrine Dimers with Torpedo c alifornica Acetylcholinesterase:  Binding of Bis(5)-tacrine Produces a Dramatic Rearrangement in the Active-Site Gorge von Rydberg, Edwin H, Brumshtein, Boris, Greenblatt, Harry M, Wong, Dawn M, Shaya, David, Williams, Larry D, Carlier, Paul R, Pang, Yuan-Ping, Silman, Israel, Sussman, Joel L

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Corrigendum to “Re-engineering aryl methylcarbamates to confer high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase” [Bioorg. Med. Chem. Lett. 22... von Hartsel, Joshua A., Wong, Dawn M., Mutunga, James M., Ma, Ming, Anderson, Troy D., Wysinski, Ania, Islam, Rafique, Wong, Eric A., Paulson, Sally L., Li, Jianyong, Lam, Polo C.H., Totrov, Maxim, Bloomquist, Jeffrey R., Carlier, Paul R.

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Re-engineering aryl methylcarbamates to confer high selectivity for inhibition of Anopheles gambiae vs human acetylcholinesterase von Hartsel, Joshua A., Wong, Dawn M., Mutunga, James M., Ma, Ming, Anderson, Troy D., Wysinski, Ania, Islam, Rafique, Wong, Eric A., Paulson, Sally L., Li, Jianyong, Lam, Polo C. H., Totrov, Maxim, Bloomquist, Jeffrey R., Carlier, Paul R.

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Preparation of the chiral amine salts [(η5-C5H5)Ru(PPh3)(CNtBu)(NH2R)]PF6, RNH2=α-methylbenzylamine, 1-cyclohexylethylamine, and 1-(1-naphthyl)ethylamine: X-ray single crystal stru... von Wong, Dawn M., Simpson, Stephen J.

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