Identification and Preclinical Development of a 2,5,6-Trisubstituted Fluorinated Pyridine Derivative as a Radioligand for the Positron Emission Tomography Imaging of Cannabinoid Ty... von Haider, Ahmed, Gobbi, Luca, Kretz, Julian, Ullmer, Christoph, Brink, Andreas, Honer, Michael, Woltering, Thomas J, Muri, Dieter, Iding, Hans, Bürkler, Markus, Binder, Martin, Bartelmus, Christian, Knuesel, Irene, Pacher, Pal, Herde, Adrienne Müller, Spinelli, Francesco, Ahmed, Hazem, Atz, Kenneth, Keller, Claudia, Weber, Markus, Schibli, Roger, Mu, Linjing, Grether, Uwe, Ametamey, Simon M

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BACE1 inhibitors: A head group scan on a series of amides von Woltering, Thomas J., Wostl, Wolfgang, Hilpert, Hans, Rogers-Evans, Mark, Pinard, Emmanuel, Mayweg, Alexander, Göbel, Martin, Banner, David W., Benz, Jörg, Travagli, Massimiliano, Pollastrini, Martina, Marconi, Guido, Gabellieri, Emanuele, Guba, Wolfgang, Mauser, Harald, Andreini, Matteo, Jacobsen, Helmut, Power, Eoin, Narquizian, Robert

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Conformationally restricted pyrrolidines by intramolecular [2+2] photocycloaddition reactions von Fort, Diego A, Woltering, Thomas J, Nettekoven, Matthias, Knust, Henner, Bach, Thorsten

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Synthesis and characterization of 1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: Part 4. In vivo active potent and selective non-competitive metabotropic glutamate receptor... von Woltering, Thomas J., Wichmann, Jürgen, Goetschi, Erwin, Knoflach, Frédéric, Ballard, Theresa M., Huwyler, Jörg, Gatti, Silvia

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Pharmacological manipulation of mGlu2 receptors influences cognitive performance in the rodent von Higgins, Guy A., Ballard, Theresa M., Kew, James N.C., Grayson Richards, J., Kemp, John A., Adam, Geo, Woltering, Thomas, Nakanishi, Shigetada, Mutel, Vincent

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Effects of the mGluR2/3 agonist LY354740 on computerized tasks of attention and working memory in marmoset monkeys von Spinelli, Simona, Ballard, Theresa, Gatti-McArthur, Silvia, Richards, Grayson J, Kapps, Martin, Woltering, Thomas, Wichmann, Jurgen, Stadler, Heinz, Feldon, Joram, Pryce, Christopher R

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Synthesis and characterization of 8-ethynyl-1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: New potent non-competitive metabotropic glutamate receptor 2/3 antagonists. Part 1 von Woltering, Thomas J., Adam, Geo, Alanine, Alexander, Wichmann, Jürgen, Knoflach, Frédéric, Mutel, Vincent, Gatti, Silvia

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Synthesis and characterization of 1,3-dihydro-benzo[ b][1,4]diazepin-2-one derivatives: Part 3. New potent non-competitive metabotropic glutamate receptor 2/3 antagonists von Woltering, Thomas J., Wichmann, Jürgen, Goetschi, Erwin, Adam, Geo, Kew, James N.C., Knoflach, Frédéric, Ballard, Theresa M., Huwyler, Jörg, Mutel, Vincent, Gatti, Silvia

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Asymmetric Synthesis and Receptor Pharmacology of the Group II mGlu Receptor Ligand (1S,2R,3R,5R,6S)-2-Amino-3-hydroxy-bicyclo[3.1.0]hexane-2,6-dicarboxylic Acid-HYDIA von Woltering, Thomas J., Adam, Geo, Huguenin, Philipp, Wichmann, Jürgen, Kolczewski, Sabine, Gatti, Silvia, Bourson, Anne, Kew, James N. C., Richards, Grayson, Kemp, John A., Mutel, Vincent, Knoflach, Frédéric

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Mutagenesis and Molecular Modeling of the Orthosteric Binding Site of the mGlu2 Receptor Determining Interactions of the Group II Receptor Antagonist 3H-HYDIA von Lundström, Linda, Kuhn, Bernd, Beck, Jennifer, Borroni, Edilio, Wettstein, Joseph G., Woltering, Thomas J., Gatti, Silvia

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In Vitro Binding Characteristics of a New Selective Group II Metabotropic Glutamate Receptor Radioligand, [3H]LY354740, in Rat Brain von Schaffhauser, H, Richards, J G, Cartmell, J, Chaboz, S, Kemp, J A, Klingelschmidt, A, Messer, J, Stadler, H, Woltering, T, Mutel, V

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Design, synthesis and biological evaluation of aryl-substituted sialyl Lewis X mimetics prepared via cross-metathesis of C-fucopeptides von Huwe, Christoph M, Woltering, Thomas J, Jiricek, Jan, Weitz-Schmidt, Gabriele, Wong, Chi-Huey

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Synthesis of Fluorinated Tricyclic Scaffolds by Intramolecular [2+2] Photocycloaddition Reactions von Fort, Diego A., Woltering, Thomas J., Nettekoven, Matthias, Knust, Henner, Bach, Thorsten

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Synthesis of Fluorinated Tricyclic Scaffolds by Intramolecular [2+2] Photocycloaddition Reactions von Fort, Diego A., Woltering, Thomas J., Nettekoven, Matthias, Knust, Henner, Bach, Thorsten

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Characterization of (2S,2′R,3′R)‐2‐(2′,3′‐[3H]‐Dicarboxycyclopropyl)glycine Binding in Rat Brain von Mutel, Vincent, Adam, Geo, Chaboz, Sylvie, Kemp, John A., Klingelschmidt, Agnés, Messer, Jürg, Wichmann, Jürgen, Woltering, Thomas, Richards, John Grayson

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A Real-World Perspective on Molecular Design: Miniperspective von Kuhn, Bernd, Guba, Wolfgang, Hert, Jérôme, Banner, David, Bissantz, Caterina, Ceccarelli, Simona, Haap, Wolfgang, Körner, Matthias, Kuglstatter, Andreas, Lerner, Christian, Mattei, Patrizio, Neidhart, Werner, Pinard, Emmanuel, Rudolph, Markus G, Schulz-Gasch, Tanja, Woltering, Thomas, Stahl, Martin

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BACE1 INHIBITORS von HAAP, Wolfgang, WOLTERING, Thomas

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Design and synthesis of C-linked fucosides as inhibitors of E-selectin von Uchiyama, Taketo, Woltering, Thomas J., Wong, Weichyun, Lin, Chun-Cheng, Kajimoto, Tetsuya, Takebayashi, Maki, Wéitz-Schmidt, Gabriel, Asakura, Tetsuo, Noda, Masatoshi, Wong, Chi-Huey

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Structure-activity relationships of substituted 5H-thiazolo[3,2-a]pyrimidines as group 2 metabotropic glutamate receptor antagonists von Wichmann, Jürgen, Adam, Geo, Kolczewski, Sabine, Mutel, Vincent, Woltering, Thomas

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Mutagenesis and Molecular Modeling of the Orthosteric Binding Site of the mGlu2 Receptor Determining Interactions of the Group II Receptor Antagonist 3 H‐HYDIA von Lundström, Linda, Kuhn, Bernd, Beck, Jennifer, Borroni, Edilio, Wettstein, Joseph G., Woltering, Thomas J., Gatti, Silvia

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