Phthalazinone Pyrazoles as Potent, Selective, and Orally Bioavailable Inhibitors of Aurora-A Kinase von Prime, Michael E, Courtney, Stephen M, Brookfield, Frederick A, Marston, Richard W, Walker, Victoria, Warne, Justin, Boyd, Andrew E, Kairies, Norman A, von der Saal, Wolfgang, Limberg, Anja, Georges, Guy, Engh, Richard A, Goller, Bernhard, Rueger, Petra, Rueth, Matthias

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Candidate Biomarkers of Response to an Experimental Cancer Drug Identified through a Large-scale RNA Interference Genetic Screen von MULLENDERS, Jasper, VON DER SAAL, Wolfgang, VAN DONGEN, Miranda M. W, REIFF, Ulrike, VAN WILLIGEN, Rogier, BEIJERSBERGEN, Roderick L, TIEFENTHALER, Georg, KLEIN, Christian, BERNARDS, René

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Non-nucleoside inhibitors of HIV-1 reverse transcriptase: molecular modeling and x-ray structure investigations von Schaefer, Wolfgang, Friebe, Walter Gunar, Leinert, Herbert, Mertens, Alfred, Poll, Thomas, Von der Saal, Wolfgang, Zilch, Harald, Nuber, Bernhard, Ziegler, Manfred L

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Development of a Virtual Screening Method for Identification of “Frequent Hitters” in Compound Libraries von Roche, Olivier, Schneider, Petra, Zuegge, Jochen, Guba, Wolfgang, Kansy, Manfred, Alanine, Alexander, Bleicher, Konrad, Danel, Franck, Gutknecht, Eva-Maria, Rogers-Evans, Mark, Neidhart, Werner, Stalder, Henri, Dillon, Michael, Sjögren, Eric, Fotouhi, Nader, Gillespie, Paul, Goodnow, Robert, Harris, William, Jones, Phil, Taniguchi, Mikio, Tsujii, Shinji, von der Saal, Wolfgang, Zimmermann, Gerd, Schneider, Gisbert

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X-ray structure of active site-inhibited clotting factor Xa. Implications for drug design and substrate recognition von Brandstetter, H, Kühne, A, Bode, W, Huber, R, von der Saal, W, Wirthensohn, K, Engh, R A

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Improved Procedures For Large Scale Preparation Of 6- and 7-Oxy-Substituted Isoquinolines and A Convenient Work-Up Protocol For Titanium Supported Reactions von Kucznierz, Ralf, Dickhaut, Joachim, Leinert, Herbert, Saal, Wolfgang von der

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Cytidine-5'-triphosphate synthetase catalyzes the phosphorylation of uridine 5'-triphosphate by adenosine 5'-triphosphate von Von der Saal, Wolfgang, Villafranca, Joseph J, Anderson, Paul M

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X-ray Structure of Active Site-inhibited Clotting Factor Xa von Brandstetter, Hans, Kühne, Anja, Bode, Wolfram, Huber, Robert, von der Saal, Wolfgang, Wirthensohn, Klaus, Engh, Richard A.

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A Short Synthesis of the Factor-Xa Inhibitor DX-9065a using palladium-catalyzed key steps von Kehr, Christiane, Neidlein, Richard, Engh, Richard A., Brandsretter, Hans, Kucznierz, Ralf, Leinert, Herbert, Marzenell, Klaus, Strein, Klaus, Saal, Wolfgang Von Der

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Enzyme flexibility, solvent and ‘weak’ interactions characterize thrombin–ligand interactions: implications for drug design von Engh, Richard A, Brandstetter, Hans, Sucher, Gudrun, Eichinger, Andreas, Baumann, Ulrich, Bode, Wolfram, Huber, Robert, Poll, Thomas, Rudolph, Rainer, von der Saal, Wolfgang

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Tetrahydro-isoquinoline-Based Factor Xa Inhibitors von Kucznierz, Ralf, Grams, Frank, Leinert, Herbert, Marzenell, Klaus, Engh, Richard A, von der Saal, Wolfgang

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Pyrroles from 1,2-Cyclopropanediamines and Aldehydes von von der Saal, Wolfgang, Reinhardt, Robert, Stawitz, Josef, Quast, Helmut

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DERIVATIVES OF 4-AMINO-PYRIDINE AS SELECTIVE THROMBIN INHIBITORS von von der Saal, Wolfgang, Kucznierz, Ralf, Leinert, Herbert, Engh, Richard A.

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Proton and carbon-13 nuclear magnetic resonance spectra of methylenecyclopropane and proton nuclear magnetic resonance spectra of some methyl-substituted methylenecyclopropanes. A... von Von der Saal, Wolfgang, Risler, Wolfgang, Stawitz, Josef, Quast, Helmut

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Cyclopropanediamines. 6. 1 Autocatalytic Conversion of 1-Methyl- r -1, t -2-cyclopropanediamine into 4-Aminobutan-2-one in Aqueous Buffer Solutions of pH 6.5−10. Azomethine Ylides... von von der Saal, Wolfgang, Quast, Helmut

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Comparison of two implementations of the incremental construction algorithm in flexible docking of thrombin inhibitors von Knegtel, R M, Bayada, D M, Engh, R A, von der Saal, W, van Geerestein, V J, Grootenhuis, P D

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Cyclopropanediamines. 6. Autocatalytic Conversion of 1-Methyl-r-1,t-2-cyclopropanediamine into 4-Aminobutan-2-one in Aqueous Buffer Solutions of pH 6.5−10. Azomethine Ylides as Int... von von der Saal, Wolfgang, Quast, Helmut

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DESAMINOANTHRACYCLINES FROM THE ANTIBIOTIC COMPLEX CICLAMYCIN von BIEBER, LOTHAR W., ÁLVARO A. DA SILVA FILHO, MÉLLO, JOSÉ F. DE, LIMA, OSWALDO G. DE, NASCIMENTO, MARCIA S. DO, VEITH, HANS J., SAAL, WOLFGANG VON DER

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Diarylsulfonamides as selective, non-peptidic thrombin inhibitors von Weber, Ingo R., Neidlein, Richard, von der Saal, Wolfgang, Grams, Frank, Leinert, Herbert, Strein, Klaus, Engh, Richard A., Kucznierz, Ralf

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Desaminoanthracyclines from the antibotic complex ciclamycin von BIEBER, LOTHAR W., FILHO, ÁLVARO A. DA SILVA, MÉLLO, JOSÉ F. DE, LIMA, OSWALDO G. DE, NASCIMENTO, MARCIA S. DO, VEITH, HANS J., SAAL, WOLFGANG VON DER

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