Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps von Plé, Coline, Tam, Heng-Keat, Vieira Da Cruz, Anais, Compagne, Nina, Jiménez-Castellanos, Juan-Carlos, Müller, Reinke T., Pradel, Elizabeth, Foong, Wuen Ee, Malloci, Giuliano, Ballée, Alexia, Kirchner, Moritz A., Moshfegh, Parisa, Herledan, Adrien, Herrmann, Andrea, Deprez, Benoit, Willand, Nicolas, Vargiu, Attilio Vittorio, Pos, Klaas M., Flipo, Marion, Hartkoorn, Ruben C.

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Combination therapy for tuberculosis treatment: pulmonary administration of ethionamide and booster co-loaded nanoparticles von Costa-Gouveia, Joana, Pancani, Elisabetta, Jouny, Samuel, Machelart, Arnaud, Delorme, Vincent, Salzano, Giuseppina, Iantomasi, Raffaella, Piveteau, Catherine, Queval, Christophe J., Song, Ok-Ryul, Flipo, Marion, Deprez, Benoit, Saint-André, Jean-Paul, Hureaux, José, Majlessi, Laleh, Willand, Nicolas, Baulard, Alain, Brodin, Priscille, Gref, Ruxandra

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Regioselective and Stereoselective Synthesis of Parthenolide Analogs by Acyl Nitroso-Ene Reaction and Their Biological Evaluation against Mycobacterium tuberculosis von Gioia, Bruna, Ruggieri, Francesca, Biela, Alexandre, Landry, Valérie, Roussel, Pascal, Piveteau, Catherine, Leroux, Florence, Hartkoorn, Ruben C, Willand, Nicolas

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Rubrolone production by Dactylosporangium vinaceum: biosynthesis, modulation and possible biological function von Moureu, Sophie, Caradec, Thibault, Trivelli, Xavier, Drobecq, Hervé, Beury, Delphine, Bouquet, Peggy, Caboche, Segolene, Desmecht, Eva, Maurier, Florence, Muharram, Ghaffar, Villemagne, Baptiste, Herledan, Adrien, Hot, David, Willand, Nicolas, Hartkoorn, Ruben Christiaan

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Molecular Design in Practice: A Review of Selected Projects in a French Research Institute That Illustrates the Link between Chemical Biology and Medicinal Chemistry von Deprez, Benoit, Bosc, Damien, Charton, Julie, Couturier, Cyril, Deprez-Poulain, Rebecca, Flipo, Marion, Leroux, Florence, Villemagne, Baptiste, Willand, Nicolas

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A Three-Step Process to Isolate Large Quantities of Bioactive Sesquiterpene Lactones from Cichorium intybus L. Roots and Semisynthesis of Chicory STLs Standards von Ruggieri, Francesca, Hance, Philippe, Gioia, Bruna, Biela, Alexandre, Roussel, Pascal, Hilbert, Jean-Louis, Willand, Nicolas

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Rapid and Efficient Access to Novel Bio-Inspired 3-Dimensional Tricyclic SpiroLactams as Privileged Structures via Meyers' Lactamization von Tangara, Salia, Faïon, Léo, Piveteau, Catherine, Capet, Frédéric, Godelier, Romain, Michel, Marion, Flipo, Marion, Deprez, Benoit, Willand, Nicolas, Villemagne, Baptiste

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Exploring the Antitubercular Activity of Anthranilic Acid Derivatives: From MabA (FabG1) Inhibition to Intrabacterial Acidification von Faïon, Léo, Djaout, Kamel, Pintiala, Catalin, Piveteau, Catherine, Leroux, Florence, Biela, Alexandre, Slupek, Stéphanie, Antoine, Rudy, Záhorszká, Monika, Cantrelle, Francois-Xavier, Hanoulle, Xavier, Korduláková, Jana, Deprez, Benoit, Willand, Nicolas, Baulard, Alain R, Flipo, Marion

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On the Hunt for Next-Generation Antimicrobial Agents: An Online Symposium Organized Jointly by the French Society for Medicinal Chemistry (Société de Chimie Thérapeutique) and the... von Antraygues, Kevin, Compagne, Nina, Ruggieri, Francesca, Djaout, Kamel, Edoo, Zainab, Eveque, Maxime, Faïon, Léo, Gioia, Bruna, Tangara, Salia, Vieira Da Cruz, Anais, Villemagne, Baptiste, Flipo, Marion, Baulard, Alain, Willand, Nicolas

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Molecular mechanism of a triazole-containing inhibitor of Mycobacterium tuberculosis DNA gyrase von Gedeon, Antoine, Yab, Emilie, Dinut, Aurelia, Sadowski, Elodie, Capton, Estelle, Dreneau, Aurore, Petit, Julienne, Gioia, Bruna, Piveteau, Catherine, Djaout, Kamel, Lecat, Estelle, Wehenkel, Anne Marie, Gubellini, Francesca, Mechaly, Ariel, Alzari, Pedro M., Deprez, Benoît, Baulard, Alain, Aubry, Alexandra, Willand, Nicolas, Petrella, Stéphanie

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Natural Compounds: Leads or Ideas? Bioinspired Molecules for Drug Discovery von Beghyn, Terence, Deprez-Poulain, Rebecca, Willand, Nicolas, Folleas, Benoit, Deprez, Benoit

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Exploring Drug Target Flexibility Using in Situ Click Chemistry: Application to a Mycobacterial Transcriptional Regulator von Willand, Nicolas, Desroses, Matthieu, Toto, Patrick, Dirié, Bertrand, Lens, Zoé, Villeret, Vincent, Rucktooa, Prakash, Locht, Camille, Baulard, Alain, Deprez, Benoit

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Publisher Correction: Combination therapy for tuberculosis treatment: pulmonary administration of ethionamide and booster co-loaded nanoparticles von Costa-Gouveia, Joana, Pancani, Elisabetta, Jouny, Samuel, Machelart, Arnaud, Delorme, Vincent, Salzano, Giuseppina, Iantomasi, Raffaella, Piveteau, Catherine, Queval, Christophe J., Song, Ok-Ryul, Flipo, Marion, Deprez, Benoit, Saint-André, Jean-Paul, Hureaux, José, Majlessi, Laleh, Willand, Nicolas, Baulard, Alain, Brodin, Priscille, Gref, Ruxandra

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Water-based conditions for the microscale parallel synthesis of bicyclic lactams von Malaquin, Sandra, Jida, Mouhamad, Courtin, Justin, Laconde, Guillaume, Willand, Nicolas, Deprez, Benoit, Deprez-Poulain, Rebecca

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Sustainability in drug discovery von Wynendaele, Evelien, Furman, Christophe, Wielgomas, Bartosz, Larsson, Per, Hak, Eelko, Block, Thomas, Van Calenbergh, Serge, Willand, Nicolas, Markuszewski, Michal, Odell, Luke R., Poelarends, Gerrit J., De Spiegeleer, Bart

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Recent advances in Fragment-based strategies against tuberculosis von Villemagne, Baptiste, Faïon, Léo, Tangara, Salia, Willand, Nicolas

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Antibiotics with novel mode of action as new weapons to fight antimicrobial resistance von Ruggieri, Francesca, Compagne, Nina, Antraygues, Kevin, Eveque, Maxime, Flipo, Marion, Willand, Nicolas

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Desirable drug–drug interactions or when a matter of concern becomes a renewed therapeutic strategy von Guieu, Benjamin, Jourdan, Jean-Pierre, Dreneau, Aurore, Willand, Nicolas, Rochais, Christophe, Dallemagne, Patrick

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Reversion of antibiotic resistance in Mycobacterium tuberculosis by spiroisoxazoline SMARt-420 von Blondiaux, Nicolas, Moune, Martin, Desroses, Matthieu, Frita, Rosangela, Flipo, Marion, Mathys, Vanessa, Soetaert, Karine, Kiass, Mehdi, Delorme, Vincent, Djaout, Kamel, Trebosc, Vincent, Kemmer, Christian, Wintjens, René, Wohlkönig, Alexandre, Antoine, Rudy, Huot, Ludovic, Hot, David, Coscolla, Mireia, Feldmann, Julia, Gagneux, Sebastien, Locht, Camille, Brodin, Priscille, Gitzinger, Marc, Déprez, Benoit, Willand, Nicolas, Baulard, Alain R.

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Crystal structure of the Mycobacterium tuberculosis VirS regulator reveals its interaction with the lead compound SMARt751 von Grosse, Camille, Sigoillot, Maud, Megalizzi, Véronique, Tanina, Abdalkarim, Willand, Nicolas, Baulard, Alain R., Wintjens, René

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