Benzodiazepine gastrin and brain cholecystokinin receptor ligands; L-365,260 von Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Anderson, Paul S, Freidinger, Roger M

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Development of 1,4-benzodiazepine cholecystokinin type B antagonists von Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Garsky, Victor M, Gilbert, Kevin F, Leighton, James L, Carson, Kenneth L

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Large-scale synthesis of a cyclic hexapeptide analog of somatostatin von Brady, Stephen F, Freidinger, Roger M, Paleveda, William J, Colton, Christiane D, Homnick, Carl F, Whitter, Willie L, Curley, Paul, Nutt, Ruth F, Veber, Daniel F

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Development of a novel class of cyclic hexapeptide oxytocin antagonists based on a natural product von Williams, Peter D, Bock, Mark G, Tung, Roger D, Garsky, Victor M, Perlow, Debra S, Erb, Jill M, Lundell, G. F, Gould, Norman P, Whitter, Willie L

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Renin inhibitors containing hydrophilic groups. Tetrapeptides with enhanced aqueous solubility and nanomolar potency von Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Freidinger, Roger M, Rittle, Kenneth E, Payne, Linda S, Boger, Joshua, Whitter, Willie L, LaMont, Bruce I

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Cholecystokinin-A receptor ligands based on the .kappa.-opioid agonist tifluadom von Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Freidinger, Roger M, Chang, Raymond S. L, Chen, T. B, Lotti, Victor J

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Design of Potent, Orally Effective, Nonpeptidal Antagonists of the Peptide Hormone Cholecystokinin von Evans, Ben E., Bock, Mark G., Rittle, Kenneth E., DiPardo, Robert M., Whitter, Willie L., Veber, Daniel F., Anderson, Paul S., Freidinger, Roger M.

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A new amine resolution method and its application to 3-aminobenzodiazepines von Rittle, Kenneth E, Evans, Ben E, Bock, Mark G, DiPardo, Robert M, Whitter, Willie L, Homnick, Carl F, Veber, Daniel F, Freidinger, Roger M

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Cholecystokinin-A receptor ligands based on the .kappa.-opioid agonist tifluadom [Erratum to document cited in CA112(5):30228d] von Bock, Mark G, DiPardo, Robert M, Evans, Ben E, Rittle, Kenneth E, Whitter, Willie L, Veber, Daniel F, Freidinger, Roger M, Chang, Raymond S. L, Chen, T. B, Lotti, Victor J

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Synthesis of 2H-isoindole-4,7-diones by 1,3-dipolar addition of oxazolium 5-oxides to 1,4-quinones von Myers, John A, Moore, Lloyd D, Whitter, Willie L, Council, Samuel L, Waldo, Rosalyn M, Lanier, Jerry L, Omoji, Bassey U

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Synthesis, antiviral activity, and bioavailability studies of γ-lactam derived HIV protease inhibitors von Hungate, Randall W., Chen, Jenny L., Starbuck, Ken E., Vacca, Joseph P., McDaniel, Stacey L., Levin, Rhonda B., Dorsey, Bruce D., Guare, James P., Holloway, M.Katharine, Whitter, Willie, Darke, Paul L., Zugay, Joan A., Schleif, William A., Emini, Emilio A., Quintero, Julio C., Lin, Juinn H., Chen, I-Wu, Anderson, Paul S., Huff, Joel R.

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Nanomolar-affinity, non-peptide oxytocin receptor antagonists von Evans, Ben E, Lundell, George F, Gilbert, Kevin F, Bock, Mark G, Rittle, Kenneth E, Carroll, Leigh Anne, Williams, Peter D, Pawluczyk, Joseph M, Leighton, James L

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Design of cholecystokinin peptidomimetics von Bock, Mark G., DiPardo, Robert M., Evans, Ben E., Rittle, Kenneth E., Veber, Daniel F., Whitter, Willie L., Chang, Raymond S.L., Lotti, Victor J., Anderson, Paul S., Freidinger, Roger M.

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4-CYCLOALKYLAMINOPYRAZOLOPYRIMIDIN ALS NMDA/NR2B-ANTAGONISTEN von SANDERSON, E, BUTCHER, JOHN, WHITTER, WILLIE, MCINTYRE, J, LIVERTON, NIGEL, YOUNG, D, DIECKHAUS, CHRISTINE, MUNSON, PETER, THOMPSON, WAYNE, LAYTON, E, MCCAULEY, A, PHILLIPS, T

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4-cycloakylaminopyrazolo pyrimidine NMDA/NR2B antagonists von Thompson, Wayne, Young, Steven D, Phillips, Brian T, Munson, Peter, Whitter, Willie, Liverton, Nigel, Dieckhaus, Christine, Butcher, John, McCauley, John A, McIntyre, Charles J, Layton, Mark E, Sanderson, Philip E

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4-cycloakylaminopyrazolo pyrimidine NMDA/NR2B antagonists von YOUNG STEVEN D, MUNSON PETER, WHITTER WILLIE, SANDERSON PHILIP E, PHILLIPS BRIAN T, MCCAULEY JOHN A, THOMPSON WAYNE, BUTCHER JOHN, DIECKHAUS CHRISTINE, MCINTYRE CHARLES J, LIVERTON NIGEL, LAYTON MARK E

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Radiation Sensitization and Chemical Studies on Isoindole-4,7-Diones von Infante, Gabriel A., Gonzalez, Pedro, Cruz, Daniel, Correa, Jose, Myers, John A., Ahmad, Mir F., Whitter, Willie L., Santos, Alfonso, Neta, P.

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1,4 SUBSTITUTED PIPERIDINYL NMDA/NR2B ANTAGONISTS von WHITTER, WILLIE, CLAREMON, DAVID, A, KULAGOWSKI, JANUSZ, HUSCROFT, IAN, THOMPSON, WAYNE, MUNSON, PETER, M

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1,4 substituted piperidinyl NMDA/NR2B antagonists von KULAGOWSKI JANUSZ, WHITTER WILLIE, HUSCROFT IAN, THOMPSON WAYNE, MUNSON PETER M, CLAREMON DAVID A

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1,4 substituted piperidinyl NMDA/NR2B antagonists von Thompson, Wayne, Claremon, David, Munson, Peter, Kulagowski, Janusz, Whitter, Willie, Huscroft, Ian

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