Search for new lead compounds: The example of the chemical and pharmacological dissection of aminopyridazines von Wermuth, Camille-Georges

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Palladium-Catalysed Cross-Coupling Reactions on Pyridazine Moieties von Nara, Susheel, Martinez, Jean, Wermuth, Camille-Georges, Parrot, Isabelle

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A Convenient 3-Step Synthesis of 3-Acetamido-6-arylpyridazines Directed to Novel Y5 Receptor Antagonist von Guéry, Sébastien, Rival, Yveline, Wermuth, Camille-Georges, Renard, Pierre, Boutin, Jean-Albert

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Diastereoselectivity in conjugate addition of alkylcuprates to vinylogous ester of N O-diprotected serinal von Jako, Isabelle, Uibera, Pierre, Mann, André, Taddei, Maurizio, Wermuth, Camille-Georges

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Synthesis of constrained arylpiperidines using intramolecular Heck or radical reactions von Morice, Christophe, Domostoj, Mathias, Briner, Karin, Mann, André, Suffert, Jean, Wermuth, Camille-Georges

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The synthesis of α-amino-γ-substituted adipic acids: stereoelectronic effects during the 1,4-addition of organocuprates to methyl N-tert-butoxy-6-oxo-1,2,3,6-tetrahydropyridine-2-c... von Muller, Mireille, Schoenfelder, Angèle, Didier, Bruno, Mann, André, Wermuth, Camille-Georges

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1,3-diastereocontrol with bromoallenes. Synthesis of enantiomerically pure β-branched α-amino acids von D'Aniello, Fabiana, Mann, André, Taddei, Maurizio, Wermuth, Camille-Georges

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From phenylaziridine to phenylkainoids. A formal synthesis of (±)-phenylkainic acid von Schneider, Marie-Reine, Klotz, Philippe, Ungureanu, Ioana, Mann, André, Wermuth, Camille-Georges

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Fragmentation of N-Boc arylpiperazines under basic conditions von Garrido, Fabrice, Mann, André, Wermuth, Camille-Georges

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Modelling of the binding site of the human m1 muscarinic receptor: experimental validation and refinement von Bourdon, H, Trumpp-Kallmeyer, S, Schreuder, H, Hoflack, J, Hibert, M, Wermuth, C G

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Inhibition of cyclic adenosine-3',5'-monophosphate phosphodiesterase from vascular smooth muscle by rolipram analogs von Marivet, Michel C, Bourguignon, Jean Jacques, Lugnier, Claire, Mann, Andre, Stoclet, Jean Claude, Wermuth, Camille Georges

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Stereoselective synthesis of 3-alkylated glutamic acids: application to the synthesis of secokainic acid von Jako, Isabelle, Uiber, Pierre, Mann, Andre, Wermuth, Camille Georges, Boulanger, Thierry, Norberg, Bernadette, Evrard, Guy, Durant, Francois

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Synthesis and structure-activity relationships of a series of aminopyridazine derivatives of .gamma.-aminobutyric acid acting as selective GABA-A antagonists von Wermuth, Camille Georges, Bourguignon, Jean Jacques, Schlewer, Gilbert, Gies, Jean Pierre, Schoenfelder, Angele, Melikian, Anita, Bouchet, Marie Jeanne, Chantreux, Dominique, Molimard, Jean Charles

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The active analog approach applied to the pharmacophore identification of benzodiazepine receptor ligands von Tebib, S, Bourguignon, J J, Wermuth, C G

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Synthesis of [3H]-labelled trans 4-hydroxycrotonic acid (T-HCA), an endogenous substance interfering with 4-hydroxybutyrate (GHB) von Schmitt, Martine, Bourguignon, Jean-Jacques, Wermuth, Camille-Georges, Schott, Dominique, Rousseau, Bernard, Beaucourt, Jean-Pierre

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Optically active benzamides as predictive tools for mapping the dopamine D2 receptor von ROGNAN, D, SOKOLOFF, P, MANN, A, MARTRES, M.-P, SCHWARTZ, J.-C, COSTENTIN, J, WERMUTH, C.-G

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SR 46559A : a novel and potent muscarinic compound with no cholinergic syndrome von KAN, J.-P, STEINBERG, R, WERMUTH, C.-G, WORMS, P, SOUBRIE, P, LE FUR, G, OURY-DONAT, F, MICHAUD, J.-C, THURNEYSSEN, O, TERRANOVA, J.-P, GUEUDET, C, SOUILHAC, J, BRODIN, R, BOIGEGRAIN, R

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Palladium-Catalyzed Cross-Coupling Reactions on Pyridazine Moieties von Nara, Susheel, Martinez, Jean, Wermuth, Camille-Georges, Parrot, Isabelle

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Synthesis of New Diazepinones von Wermuth, Camille-Georges, Koenig, Jean-Jacques

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ChemInform Abstract: Search for New Lead Compounds: The Example of the Chemical and Pharmacological Dissection of Aminopyridazines von Wermuth, Camille-Georges

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