Selective Optimization of Side Activities:  Another Way for Drug Discovery von Wermuth, Camille G

Volltext

Are pyridazines privileged structures? von Wermuth, Camille G.

Volltext

Design, Synthesis, and Structure−Activity Relationships of a Series of 3-[2-(1-Benzylpiperidin-4-yl)ethylamino]pyridazine Derivatives as Acetylcholinesterase Inhibitors von Contreras, Jean-Marie, Parrot, Isabelle, Sippl, Wolfgang, Rival, Yveline M, Wermuth, Camille G

Volltext

Development of Novel 1,2,3,4-Tetrahydroisoquinoline Derivatives and Closely Related Compounds as Potent and Selective Dopamine D₃ Receptor Ligands von Mach, Ulrich R, Hackling, Anneke E, Perachon, Sylvie, Ferry, Sandrine, Wermuth, Camille G, Schwartz, Jean-Charles, Sokoloff, Pierre, Stark, Holger

Volltext

Selective optimization of side activities: the SOSA approach von Wermuth, Camille G.

Volltext

Multitargeted drugs: the end of the ‘one-target-one-disease’ philosophy? von Wermuth, Camille G.

Volltext

Similarity in drugs: reflections on analogue design von Wermuth, Camille G.

Volltext

N-(ω-(4-(2-Methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as Dopamine D2 and D3 Receptor Ligands von Hackling, Anneke, Ghosh, Robin, Perachon, Sylvie, Mann, André, Höltje, Hans-Dieter, Wermuth, Camille G, Schwartz, Jean-Charles, Sippl, Wolfgang, Sokoloff, Pierre, Stark, Holger

Volltext

Aminopyridazines as Acetylcholinesterase Inhibitors von Contreras, Jean-Marie, Rival, Yveline M, Chayer, Said, Bourguignon, Jean-Jacques, Wermuth, Camille G

Volltext

Prednisone reduces muscle degeneration in dystrophin-deficient Caenorhabditis elegans von Gaud, Aurélie, Simon, Jean-Marc, Witzel, Thomas, Carre-Pierrat, Maité, Wermuth, Camille G, Ségalat, Laurent

Volltext

Use of a fluorescent polarization based high throughput assay to identify new Calmodulin ligands von Dagher, Rania, Pigault, Claire, Bonnet, Dominique, Boeglin, Damien, Pourbaix, Christelle, Kilhoffer, Marie-Claude, Villa, Pascal, Wermuth, Camille G., Hibert, Marcel, Haiech, Jacques

Volltext

Efficient one-step synthesis of 3-amino-6-arylpyridazines von Guery, Sébastien, Parrot, Isabelle, Rival, Yveline, Wermuth, Camille G

Volltext

5-HT3 Antagonists Derived from Aminopyridazine-type Muscarinic M1 Agonists von Rival, Yveline, Hoffmann, Rémy, Didier, Bruno, Rybaltchenko, Volodymyr, Bourguignon, Jean-Jacques, Wermuth, Camille G

Volltext

Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist von Pilla, Maria, Perachon, Sylvie, Sautel, FranÇois, Garrido, Fabrice, Mann, André, Wermuth, Camille G., Schwartz, Jean-Charles, Everitt, Barry J., Sokoloff, Pierre

Volltext

(2S,4S)-2-Amino-4-(4,4-diphenylbut-1-yl)- pentane-1,5-dioic Acid:  A Potent and Selective Antagonist for Metabotropic Glutamate Receptors Negatively Linked to Adenylate Cyclase von Wermuth, Camille G, Mann, André, Schoenfelder, Angèle, Wright, Rebecca A, Johnson, Bryan G, Burnett, J. Paul, Mayne, Nancy G, Schoepp, Darryle D

Volltext

N -(ω-(4-(2-Methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as Dopamine D 2 and D 3 Receptor Ligands von Hackling, Anneke, Ghosh, Robin, Perachon, Sylvie, Mann, André, Höltje, Hans-Dieter, Wermuth, Camille G., Schwartz, Jean-Charles, Sippl, Wolfgang, Sokoloff, Pierre, Stark, Holger

Volltext

errata Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist von Pilla, Maria, Perachon, Sylvie, Sautel, François, Garrido, Fabrice, Mann, André, Wermuth, Camille G., Schwartz, Jean-Charles, Everitt, Barry J., Sokoloff, Pierre

Volltext

Characterization of the Binding of [3H]SR 95531, a GABAA Antagonist, to Rat Brain Membranes von Heaulme, Michel, Chambon, Jean‐Pierre, Leyris, Roger, Wermuth, Camille G., Biziere, Kathleen

Volltext

Structure-based 3D QSAR and design of novel acetylcholinesterase inhibitors von Sippl, W, Contreras, J M, Parrot, I, Rival, Y M, Wermuth, C G

Volltext

Efficient Palladium-catalyzed Amination and Alkylation of 3-Iodo-6-arylpyridazines von Parrot, Isabelle, Ritter, Guillaume, Wermuth, Camille G., Hibert, Marcel

Volltext