Imidazoles as Potential Anticancer Agents: An Update on Recent Studies von Sharma, Pankaj, LaRosa, Chris, Antwi, Janet, Govindarajan, Rajgopal, Werbovetz, Karl A.

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CYP5122A1 encodes an essential sterol C4-methyl oxidase in Leishmania donovani and determines the antileishmanial activity of antifungal azoles von Jin, Yiru, Basu, Somrita, Feng, Mei, Ning, Yu, Munasinghe, Indeewara, Joachim, Arline M., Li, Junan, Qin, Lingli, Madden, Robert, Burks, Hannah, Gao, Philip, Wu, Judy Qiju, Sheikh, Salma Waheed, Joice, April C., Perera, Chamani, Werbovetz, Karl A., Zhang, Kai, Wang, Michael Zhuo

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Synthesis and Antiprotozoal Activity of Cationic 1,4-Diphenyl-1H-1,2,3-triazoles von Bakunov, Stanislav A, Bakunova, Svetlana M, Wenzler, Tanja, Ghebru, Maedot, Werbovetz, Karl A, Brun, Reto, Tidwell, Richard R

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Synthesis and antileishmanial evaluation of thiazole orange analogs von Abdelhameed, Ahmed, Liao, Xiaoping, McElroy, Craig A., Joice, April C., Rakotondraibe, Liva, Li, Junan, Slebodnick, Carla, Guo, Pu, Wilson, W. David, Werbovetz, Karl A.

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Antileishmanial activity of a series of N²,N⁴-disubstituted quinazoline-2,4-diamines von Van Horn, Kurt S, Zhu, Xiaohua, Pandharkar, Trupti, Yang, Sihyung, Vesely, Brian, Vanaerschot, Manu, Dujardin, Jean-Claude, Rijal, Suman, Kyle, Dennis E, Wang, Michael Zhuo, Werbovetz, Karl A, Manetsch, Roman

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New antileishmanial candidates and lead compounds von Richard, Julian V, Werbovetz, Karl A

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Sterol profiling of Leishmania parasites using a new HPLC-tandem mass spectrometry-based method and antifungal azoles as chemical probes reveals a key intermediate sterol that supp... von Feng, Mei, Jin, Yiru, Yang, Sihyung, Joachim, Arline M., Ning, Yu, Mori-Quiroz, Luis M., Fromm, Jacob, Perera, Chamani, Zhang, Kai, Werbovetz, Karl A., Wang, Michael Zhuo

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Highly Effective Oral Amphotericin B Formulation against Murine Visceral Leishmaniasis von Wasan, Kishor M., Wasan, Ellen K., Gershkovich, Pavel, Zhu, Xiaohua, Tidwell, Richard R., Werbovetz, Karl A., Clement, John G., Thornton, Sheila J.

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Antileishmanial and Cytotoxic Activity of Some Highly Oxidized Abietane Diterpenoids from the Bald Cypress, Taxodium distichum von Naman, C. Benjamin, Gromovsky, Anthony D, Vela, Cory M, Fletcher, Joshua N, Gupta, Gaurav, Varikuti, Sanjay, Zhu, Xiaohua, Zywot, Emilia M, Chai, Heebyung, Werbovetz, Karl A, Satoskar, Abhay R, Kinghorn, A. Douglas

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Synthesis and Antiprotozoal Activity of Dicationic m‑Terphenyl and 1,3-Dipyridylbenzene Derivatives von Patrick, Donald A, Ismail, Mohamed A, Arafa, Reem K, Wenzler, Tanja, Zhu, Xiaohua, Pandharkar, Trupti, Jones, Susan Kilgore, Werbovetz, Karl A, Brun, Reto, Boykin, David W, Tidwell, Richard R

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Novel Arylimidamides for Treatment of Visceral Leishmaniasis von ZHUO WANG, Michael, XIAOHUA ZHU, MANDAL, Swati, MADHUBALA, Rentala, TIDWELL, Richard R, WILSON, W. David, BOYKIN, David W, HALL, James Edwin, KYLE, Dennis E, WERBOVETZ, Karl A, SRIVASTAVA, Anuradha, QIANG LIU, SWEAT, J. Mark, PANDHARKAR, Trupti, STEPHENS, Chad E, RICCIO, Ed, PARMAN, Toufan, MUNDE, Manoj

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Induction of Oxidative Stress in Trypanosoma brucei by the Antitrypanosomal Dihydroquinoline OSU-40 von SHANSHAN HE, DAYTON, Alex, KUPPUSAMY, Periannan, WERBOVETZ, Karl A, DREW, Mark E

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Synthesis and in Vitro Antiprotozoal Activity of Bisbenzofuran Cations von Bakunova, Svetlana M, Bakunov, Stanislav A, Wenzler, Tanja, Barszcz, Todd, Werbovetz, Karl A, Brun, Reto, Hall, James Edwin, Tidwell, Richard R

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α-Tubulin Mutations Alter Oryzalin Affinity and Microtubule Assembly Properties To Confer Dinitroaniline Resistance von Lyons-Abbott, Sally, Sackett, Dan L, Wloga, Dorota, Gaertig, Jacek, Morgan, Rachel E, Werbovetz, Karl A, Morrissette, Naomi S

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Evaluation of Arylimidamides DB1955 and DB1960 as Candidates against Visceral Leishmaniasis and Chagas' Disease: In Vivo Efficacy, Acute Toxicity, Pharmacokinetics, and Toxicology... von XIAOHUA ZHU, QIANG LIU, STEPHENS, Chad E, BANERJEE, Moloy, FARAHAT, Abdelbasset A, MUNDE, Manoj, DAVID WILSON, W, BOYKIN, David W, ZHUO WANG, Michael, WERBOVETZ, Karl A, SIHYUNG YANG, PARMAN, Toufan, GREEN, Carol E, MIRSALIS, Jon C, DE NAZARE CORREIA SOEIRO, Maria, DE SOUZA, Elen Mello, DA SILVA, Cristiane França, DA GAMA JAEN BATISTA, Denise

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Synthesis and Antiprotozoal Activity of Cationic 2-Phenylbenzofurans von Bakunov, Stanislav A, Bakunova, Svetlana M, Wenzler, Tanja, Barszcz, Todd, Werbovetz, Karl A, Brun, Reto, Tidwell, Richard R

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Antikinetoplastid activity of 3-aryl-5-thiocyanatomethyl-1,2,4-oxadiazoles von Cottrell, Denise M, Capers, Jeffrey, Salem, Manar M, DeLuca-Fradley, Kate, Croft, Simon L, Werbovetz, Karl A

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Synthesis and antitrypanosomal evaluation of derivatives of N-benzyl-1,2-dihydroquinolin-6-ols: Effect of core substitutions and salt formation von Reid, Carolyn S., Patrick, Donald A., He, Shanshan, Fotie, Jean, Premalatha, Kokku, Tidwell, Richard R., Wang, Michael Zhuo, Liu, Qiang, Gershkovich, Pavel, Wasan, Kishor M., Wenzler, Tanja, Brun, Reto, Werbovetz, Karl A.

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N-substituted-4-(pyridin-4-ylalkyl)piperazine-1-carboxamides and related compounds as Leishmania CYP51 and CYP5122A1 inhibitors von La Rosa, Chris, Sharma, Pankaj, Junaid Dar, M., Jin, Yiru, Qin, Lingli, Roy, Anuradha, Kendall, Allie, Wu, Meng, Lin, Zhihong, Uchenik, Dmitriy, Li, Junan, Basu, Somrita, Moitra, Samrat, Zhang, Kai, Zhuo Wang, Michael, Werbovetz, Karl A.

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Selective Antimicrotubule Activity of N1-Phenyl-3,5-dinitro-N4,N4-di-n-propylsulfanilamide (GB-II-5) against Kinetoplastid Parasites von Werbovetz, Karl A, Sackett, Dan L, Delfín, Dawn, Bhattacharya, Gautam, Salem, Manar, Obrzut, Tomasz, Rattendi, Donna, Bacchi, Cyrus

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