Copper-Catalyzed Trifluoromethylation of Alkoxypyridine Derivatives von Gyorfi, Nandor, Farkas, Emese, Nemet, Norbert, Weber, Csaba, Novak, Zoltan, Kotschy, Andras

Volltext

New Electrophilic Difluoromethylating Reagent von Prakash, G. K. Surya, Weber, Csaba, Chacko, Sujith, Olah, George A

Volltext

Selective disruption of NRF2-KEAP1 interaction leads to NASH resolution and reduction of liver fibrosis in mice von Seedorf, Klaus, Weber, Csaba, Vinson, Cedric, Berger, Sylvie, Vuillard, Laurent-Michel, Kiss, Arpad, Creusot, Stephanie, Broux, Olivier, Geant, Anne, Ilic, Catherine, Lemaitre, Karine, Richard, Johann, Hammoutene, Adel, Mahieux, Julien, Martiny, Virginie, Durand, Didier, Melchiore, Fabien, Nyerges, Miklos, Paradis, Valerie, Provost, Nicolas, Duvivier, Valérie, Delerive, Philippe

Volltext

Efficient Copper-Catalyzed Trifluoromethylation of Aromatic and Heteroaromatic Iodides: The Beneficial Anchoring Effect of Borates von Gonda, Zsombor, Kovács, Szabolcs, Wéber, Csaba, Gáti, Tamás, Mészáros, Attila, Kotschy, András, Novák, Zoltán

Volltext

Structure‐Based Design and Synthesis of Harmine Derivatives with Different Selectivity Profiles in Kinase versus Monoamine Oxidase Inhibition von Bálint, Balázs, Wéber, Csaba, Cruzalegui, Francisco, Burbridge, Mike, Kotschy, Andras

Volltext

Structure–Activity Relationship of Azaindole-Based Glucokinase Activators von Paczal, Attila, Bálint, Balázs, Wéber, Csaba, Szabó, Zoltán B, Ondi, Levente, Theret, Isabelle, De Ceuninck, Frédéric, Bernard, Catherine, Ktorza, Alain, Perron-Sierra, Francoise, Kotschy, András

Volltext

Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs von Wágner, Gábor, Wéber, Csaba, Nyéki, Olga, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György

Volltext

Structure-Guided Discovery of Potent and Selective DYRK1A Inhibitors von Weber, Csaba, Sipos, Melinda, Paczal, Attila, Balint, Balazs, Kun, Vilibald, Foloppe, Nicolas, Dokurno, Pawel, Massey, Andrew J, Walmsley, David Lee, Hubbard, Roderick E, Murray, James, Benwell, Karen, Edmonds, Thomas, Demarles, Didier, Bruno, Alain, Burbridge, Mike, Cruzalegui, Francisco, Kotschy, Andras

Volltext

Carbon Protonation of 2,4,6-Triaminopyrimidines:  Synthesis, NMR Studies, and Theoretical Calculations von NMETH, Balazs, WEBER, Csaba, VESZPREMI, Tamas, GATI, Tamas, DEMETER, Adam

Volltext

Structure-Guided Discovery of Selective USP7 Inhibitors with In Vivo Activity von Vasas, Attila, Ivanschitz, Lisa, Molnár, Balázs, Kiss, Árpád, Baker, Lisa, Fiumana, Andrea, Macias, Alba, Murray, James B., Sanders, Emma, Whitehead, Neil, Hubbard, Roderick E., Saunier, Carine, Monceau, Elodie, Girard, Anne Marie, Rousseau, Marion, Chanrion, Maia, Demarles, Didier, Geneste, Olivier, Weber, Csaba, Lewkowicz, Elodie, Kotschy, Andras

Volltext

Covalent Inhibitors of KEAP1 with Exquisite Selectivity von Fejes, Imre, Markacz, Piroska, Tatai, Janos, Rudas, Monika, Dunkel, Petra, Gyuris, Mario, Nyerges, Miklos, Provost, Nicolas, Duvivier, Valérie, Delerive, Philippe, Martiny, Virginie, Bristiel, Alexandra, Vidal, Brice, Richardson, William, Rothweiler, Elisabeth M, Tranberg-Jensen, Jeppe, Manning, Charlotte E, Sweeney, Melissa N, Chalk, Rod, Huber, Kilian V M, Bullock, Alex N, Herner, Andras, Seedorf, Klaus, Vinson, Cedric, Weber, Csaba, Kotschy, Andras

Volltext

Protonation of the Pyrimidine Ring at the C(5) Position:  Formation of a Stable Cationic σ-Complex von Demeter, Ádám, Wéber, Csaba, Brlik, János

Volltext

Novel solid-phase synthesis of 2,6-disubstituted 4(3 H)-quinazolinones for combinatorial library generation von Wéber, Csaba, Bielik, Attila, Szendrei, Györgyi I, Greiner, István

Volltext

Solid-phase synthesis of an N-(phenylalkyl)cinnamide library via Horner-Wadsworth-Emmons reaction von WEBER, Csaba, BIELIK, Attila, SZENDREI, Györgyi I, KESERU, György M, GREINER, Istvan

Volltext

Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluRS NAMs von WAGNER, Gábor, WEBER, Csaba, NAGY, József, KURKO, Dalma, GAL, Krisztina, GREINER, István, SZOMBATHELYI, Zsolt, KESERU, György M, DOMANY, György, NYEKI, Olga, NOGRADI, Katalin, BIELIK, Attila, MOLNAR, László, BOBOK, Amrita, HORVATH, Attila, KISS, Béla, KOLOK, Sándor

Volltext

NEW PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHANRION, Maia, VASAS, Attila, KISS, Arpad, MURRAY, James Brooke, GENESTE OLIVIER, LEWKOWICZ, Elodie, KOTSCHY, Andras, DEMARLES, Didier, WEBER, Csaba, MOLNAR, Balazs, MACIAS, Alba

Volltext bestellen

NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM von CHANRION, Maia, VASAS, Attila, KISS, Arpad, MURRAY, James Brooke, IVANSCHITZ, Lisa, GENESTE OLIVIER, LEWKOWICZ, Elodie, KOTSCHY, Andras, DEMARLES, Didier, WEBER, Csaba, MOLNAR, Balazs, MACIAS, Alba

Volltext bestellen

An efficient solid-phase synthesis of 2-alkyl-4,6-diaminopyrimidines and 2,4,6-triaminopyrimidines von Wéber, Csaba, Demeter, Ádám, Greiner, István

Volltext

PIPERIDINYL DERIVATIVES AS INHIBITORS OF UBIQUITIN SPECIFIC PROTEASE 7 von MURRAY, JAMES BROOKE, MOLNAR, BALAZS, VASAS, ATTILA, MACIAS, ALBA, KISS, ARPAD, GENESTE, OLIVIER, STROFEK, AGNES, LEWKOWICZ, ELODIE, CHANRION, MAIA, IVANSCHITZ, LISA, KUN, VILIBALD, WEBER, CSABA, KOTSCHY, ANDRAS

Volltext bestellen

Corrigendum to “Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs” [Bioorg. Med. Chem. Lett. 20 (2010) 3737–3741] von Wágner, Gábor, Wéber, Csaba, Nyéki, Olga, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György

Volltext