International Union of Basic and Clinical Pharmacology. CI. Structures and Small Molecule Modulators of Mammalian Adenylyl Cyclases von Dessauer, Carmen W, Watts, Val J, Ostrom, Rennolds S, Conti, Marco, Dove, Stefan, Seifert, Roland

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Discovery of a Potent and Selective human AC2 inhibitor based on 7-Deazapurine Analogues of Adefovir von Kraina, Pavel, Česnek, Michal, Tloušťová, Eva, Mertlíková-Kaiserová, Helena, J. Fulton, Camryn, K. Davidson, Emily, P. Smith, Brenton, J. Watts, Val, Janeba, Zlatko

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A molecular mechanism to diversify Ca2+ signaling downstream of Gs protein-coupled receptors von Brands, Julian, Bravo, Sergi, Jürgenliemke, Lars, Grätz, Lukas, Schihada, Hannes, Frechen, Fabian, Alenfelder, Judith, Pfeil, Cy, Ohse, Paul Georg, Hiratsuka, Suzune, Kawakami, Kouki, Schmacke, Luna C., Heycke, Nina, Inoue, Asuka, König, Gabriele, Pfeifer, Alexander, Wachten, Dagmar, Schulte, Gunnar, Steinmetzer, Torsten, Watts, Val J., Gomeza, Jesús, Simon, Katharina, Kostenis, Evi

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Editorial: Adenylyl cyclase isoforms as potential drug targets von Brust, Tarsis F, Ostrom, Rennolds S, Watts, Val J

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Dopamine receptor antagonists as new mode-of-action insecticide leads for control of Aedes and Culex mosquito vectors von Nuss, Andrew B, Ejendal, Karin F K, Doyle, Trevor B, Meyer, Jason M, Lang, Emma G, Watts, Val J, Hill, Catherine A

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Protein-protein interaction-based high throughput screening for adenylyl cyclase 1 inhibitors: Design, implementation, and discovery of a novel chemotype von Dwyer, Tiffany S, O'Brien, Joseph B, Ptak, Christopher P, LaVigne, Justin E, Flaherty, Daniel P, Watts, Val J, Roman, David L

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Reduced activity of adenylyl cyclase 1 attenuates morphine induced hyperalgesia and inflammatory pain in mice von Johnson, Kayla, Doucette, Alexis, Edwards, Alexis, Verdi, Aleeya, McFarland, Ryan, Hulke, Shelby, Fowler, Amanda, Watts, Val J, Klein, Amanda H

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Polydopamine-Based Simple and Versatile Surface Modification of Polymeric Nano Drug Carriers von Park, Joonyoung, Brust, Tarsis F, Lee, Hong Jae, Lee, Sang Cheon, Watts, Val J, Yeo, Yoon

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Fluorescent and Bioluminescent Protein-Fragment Complementation Assays in the Study of G Protein-Coupled Receptor Oligomerization and Signaling von Vidi, Pierre-Alexandre, Watts, Val J

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A “Genome-to-Lead” Approach for Insecticide Discovery: Pharmacological Characterization and Screening of Aedes aegypti D1-like Dopamine Receptors von Meyer, Jason M., Ejendal, Karin F. K., Avramova, Larisa V., Garland-Kuntz, Elisabeth E., Giraldo-Calderón, Gloria I., Brust, Tarsis F., Watts, Val J., Hill, Catherine A.

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Physiological roles of mammalian transmembrane adenylyl cyclase isoforms von Ostrom, Katrina F, LaVigne, Justin E, Brust, Tarsis F, Seifert, Roland, Dessauer, Carmen W, Watts, Val J, Ostrom, Rennolds S

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Selective Adenylyl Cyclase Type 1 Inhibitors as Potential Opioid Alternatives For Chronic Pain von Watts, Val J

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Pyrazolo-Pyrimidinones with Improved Solubility and Selective Inhibition of Adenylyl Cyclase Type 1 Activity for Treatment of Inflammatory Pain von Shrinidhi, Annadka, Dwyer, Tiffany S., Scott, Jason A., Watts, Val J., Flaherty, Daniel P.

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Biochemical pharmacology of adenylyl cyclases in cancer von Chandra Jena, Bikash, Flaherty, Daniel P., O'Brien, Valerie P., Watts, Val J.

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Identification of Novel Adenylyl Cyclase 5 (AC5) Signaling Networks in D1 and D2 Medium Spiny Neurons using Bimolecular Fluorescence Complementation Screening von Doyle, Trevor B., Muntean, Brian S., Ejendal, Karin F., Hayes, Michael P., Soto-Velasquez, Monica, Martemyanov, Kirill A., Dessauer, Carmen W., Hu, Chang-Deng, Watts, Val J.

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Comparative pharmacological characterization of D1-like dopamine receptors from Anopheles gambiae, Aedes aegypti and Culex quinquefasciatus suggests pleiotropic signaling in mosqui... von Hill, Catherine A, Doyle, Trevor, Nuss, Andrew B, Ejendal, Karin F K, Meyer, Jason M, Watts, Val J

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Insights into the Regulatory Properties of Human Adenylyl Cyclase Type 9 von Baldwin, Tanya A., Li, Yong, Brand, Cameron S., Watts, Val J., Dessauer, Carmen W.

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Structure of adenylyl cyclase 5 in complex with Gβγ offers insights into ADCY5-related dyskinesia von Yen, Yu-Chen, Li, Yong, Chen, Chun-Liang, Klose, Thomas, Watts, Val J., Dessauer, Carmen W., Tesmer, John J. G.

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The CUL3/neddylation inhibitor MLN4924 reduces ethanol-induced locomotor sensitization and inflammatory pain allodynia in mice von Ding, Zhong, Knipp, Gregory T., van Rijn, Richard M., Chester, Julia A., Watts, Val J.

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Molecular and pharmacological characterization of two D1-like dopamine receptors in the Lyme disease vector, Ixodes scapularis von Meyer, Jason M, Ejendal, Karin F.K, Watts, Val J, Hill, Catherine A

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