A High-Throughput BRET Cellular Target Engagement Assay Links Biochemical to Cellular Activity for Bruton’s Tyrosine Kinase von Ong, L.L., Vasta, J.D., Monereau, L., Locke, G., Ribeiro, H., Pattoli, M.A., Skala, S., Burke, J.R., Watterson, S.H., Tino, J.A., Meisenheimer, P.L., Arey, B., Lippy, J., Zhang, L., Robers, M.B., Tebben, A., Chaudhry, C.

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Cycloaddition reactions of unsaturated sulfones von Padwa, A., Ni, Z., Watterson, S. H.

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Cyclization Reactions of 2,3-Bis(phenylsulfonyl)-1,3-butadiene with Various Carbanions. A [4 + 1] Anionic Annulation Approach to Phenylsulfonyl-Substituted Cyclopentenes von Padwa, Albert, Filipkowski, Michelle A, Meske, Michael, Murphree, S. Shaun, Watterson, Scott H, Ni, Zhijie

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A New Cyclopentannulation Approach to Bicyclo[3.3.0]octenes Employing a Tandem Michael Addition-[3 + 2]-Anionic Cyclization Sequence von Padwa, Albert, Watterson, Scott H, Ni, Zhijie

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Phenylsulfonyl Ene−Allenes as Efficient Precursors to Bicyclic Systems via Intramolecular [2 + 2]-Cycloaddition Reactions von Padwa, Albert, Lipka, Helmut, Watterson, Scott H, Murphree, S. Shaun

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alto: a link-time optimizer for the Compaq Alpha von Muth, Robert, Debray, Saumya K., Watterson, Scott, De Bosschere, Koen

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Acridone-Based Inhibitors of Inosine 5‘-Monophosphate Dehydrogenase:  Discovery and SAR Leading to the Identification of N-(2-(6-(4-Ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2-... von Watterson, Scott H, Chen, Ping, Zhao, Yufen, Gu, Henry H, Dhar, T. G. Murali, Xiao, Zili, Ballentine, Shelley K, Shen, Zhongqi, Fleener, Catherine A, Rouleau, Katherine A, Obermeier, Mary, Yang, Zheng, McIntyre, Kim W, Shuster, David J, Witmer, Mark, Dambach, Donna, Chao, Sam, Mathur, Arvind, Chen, Bang-Chi, Barrish, Joel C, Robl, Jeffrey A, Townsend, Robert, Iwanowicz, Edwin J

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The Total Synthesis of (±)-Ginkgolide B von Crimmins, Michael T, Pace, Jennifer M, Nantermet, Philippe G, Kim-Meade, Agnes S, Thomas, James B, Watterson, Scott H, Wagman, Allan S

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3-Cyanoindole-based inhibitors of inosine monophosphate dehydrogenase: Synthesis and initial structure-activity relationships von MURALI DHAR, T. G, ZHONGQI SHEN, TOWNSEND, Robert, HOLLENBAUGH, Diane L, IWANOWICZ, Edwin J, GU, Henry H, PING CHEN, NORRIS, Derek, WATTERSON, Scott H, BALLENTINE, Shelley K, FLEENER, Catherine A, ROULEAU, Katherine A, BARRISH, Joel C

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Discovery of N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4- morpholineacetamide as a Novel and Potent Inhibitor of Inosine Monophosphate Dehydrogena... von Dhar, T. G. Murali, Shen, Zhongqi, Guo, Junqing, Liu, Chunjian, Watterson, Scott H, Gu, Henry H, Pitts, William J, Fleener, Catherine A, Rouleau, Katherine A, Sherbina, N. Z, McIntyre, Kim W, Witmer, Mark R, Tredup, Jeffrey A, Chen, Bang-Chi, Zhao, Rulin, Bednarz, Mark S, Cheney, Daniel L, MacMaster, John F, Miller, Laura M, Berry, Karen K, Harper, Timothy W, Barrish, Joel C, Hollenbaugh, Diane L, Iwanowicz, Edwin J

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Novel indole-based inhibitors of IMPDH: introduction of hydrogen bond acceptors at indole C-3 von Watterson, Scott H., Dhar, T.G.Murali, Ballentine, Shelley K., Shen, Zhongqi, Barrish, Joel C., Cheney, Daniel, Fleener, Catherine A., Rouleau, Katherine A., Townsend, Robert, Hollenbaugh, Diane L., Iwanowicz, Edwin J.

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Rapid synthesis of triazine inhibitors of inosine monophosphate dehydrogenase von Pitts, William J., Guo, Junqing, Dhar, T.G.Murali, Shen, Zhongqi, Gu, Henry H., Watterson, Scott H., Bednarz, Mark S., Chen, Bang-Chi, Barrish, Joel C., Bassolino, Donna, Cheney, Daniel, Fleener, Catherine A., Rouleau, Katherine A., Hollenbaugh, Diane L., Iwanowicz, Edwin J.

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Inhibitors of inosine monophosphate dehydrogenase: SARs about the N-[3-Methoxy-4-(5-oxazolyl)phenyl moiety von Iwanowicz, Edwin J., Watterson, Scott H., Guo, Junqing, Pitts, William J., Murali Dhar, T.G., Shen, Zhongqi, Chen, Ping, Gu, Henry H., Fleener, Catherine A., Rouleau, Katherine A., Cheney, Daniel L., Townsend, Robert M., Hollenbaugh, Diane L.

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Novel guanidine-based inhibitors of inosine monophosphate dehydrogenase von IWANOWICZ, Edwin J, WATTERSON, Scott H, HOLLENBAUGH, Diane L, CHUNJIAN LIU, GU, Henry H, MITT, Toomas, LEFTHERIS, Katerina, BARRISH, Joel C, FLEENER, Catherine A, ROULEAU, Katherine, SHERBINA, N. Z

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Identification of novel and potent isoquinoline aminooxazole-Based IMPDH inhibitors von Chen, Ping, Norris, Derek, Haslow, Kristin D., Murali Dhar, T.G., Pitts, William J., Watterson, Scott H., Cheney, Daniel L., Bassolino, Donna A., Fleener, Catherine A., Rouleau, Katherine A., Hollenbaugh, Diane L., Townsend, Robert M., Barrish, Joel C., Iwanowicz, Edwin J.

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Total Synthesis of (±)-Ginkgolide B von Crimmins, Michael T, Pace, Jennifer M, Nantermet, Philippe G, Kim-Meade, Agnes S, Thomas, James B, Watterson, Scott H, Wagman, Allan S

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Peri- and stereoselectivity effects in the intramolecular 2 + 2-cycloaddition reaction of phenylsulfonyl-substituted allenes von PADWA, A, FILIPKOWSKI, M. A, MESKE, M, WATTERSON, S. H, ZHIJIE NI

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Novel inhibitors of IMPDH: a highly potent and selective quinolone-based series von Watterson, Scott H., Carlsen, Marianne, Murali Dhar, T.G., Shen, Zhongqi, Pitts, William J., Guo, Junqing, Gu, Henry H., Norris, Derek, Chorba, John, Chen, Ping, Cheney, Daniel, Witmer, Mark, Fleener, Catherine A., Rouleau, Katherine, Townsend, Robert, Hollenbaugh, Diane L., Iwanowicz, Edwin J.

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Novel diamide-Based inhibitors of IMPDH von Gu, Henry H., Iwanowicz, Edwin J., Guo, Junqing, Watterson, Scott H., Shen, Zhongqi, Pitts, William J., Dhar, T.G.Murali, Fleener, Catherine A., Rouleau, Katherine, Sherbina, N.Z., Witmer, Mark, Tredup, Jeffrey, Hollenbaugh, Diane

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Novel amide-based inhibitors of inosine 5'-monophosphate dehydrogenase von WATTERSON, Scott H, CHUNJIAN LIU, IWANOWICZ, Edwin J, MURALI DHAR, T. G, GU, Henry H, PITTS, William J, BARRISH, Joel C, FLEENER, Catherine A, ROULEAU, Katherine, SHERBINA, N. Z, HOLLENBAUGH, Diane L

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