Optimized Opioid-Neurotensin Multitarget Peptides: From Design to Structure–Activity Relationship Studies von Gonzalez, Simon, Dumitrascuta, Maria, Eiselt, Emilie, Louis, Stevany, Kunze, Linda, Blasiol, Annalisa, Vivancos, Mélanie, Previti, Santo, Dewolf, Elke, Martin, Charlotte, Tourwé, Dirk, Cavelier, Florine, Gendron, Louis, Sarret, Philippe, Spetea, Mariana, Ballet, Steven

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Insightful Backbone Modifications Preventing Proteolytic Degradation of Neurotensin Analogs Improve NTS1-Induced Protective Hypothermia von Previti, Santo, Vivancoe, Melanie, Remand, Emmanuelle, Beaulieu, Sabrina, Longpre, Jean-Michel, Ballet, Steven, Sarret, Philippe, Cavelier, Florine

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Structural Optimization and Characterization of Potent Analgesic Macrocyclic Analogues of Neurotensin (8–13) von Sousbie, Marc, Vivancos, Mélanie, Brouillette, Rebecca L., Besserer-Offroy, Élie, Longpré, Jean-Michel, Leduc, Richard, Sarret, Philippe, Marsault, Éric

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Freely Behaving Mice Can Brake and Turn During Optogenetic Stimulation of the Mesencephalic Locomotor Region von van der Zouwen, Cornelis Immanuel, Boutin, Joel, Fougere, Maxime, Flaive, Aurelie, Vivancos, Melanie, Santuz, Alessandro, Akay, Turgay, Sarret, Philippe, Ryczko, Dimitri

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Use of Molecular Modeling to Design Selective NTS2 Neurotensin Analogues von Fanelli, Roberto, Floquet, Nicolas, Besserer-Offroy, Élie, Delort, Bartholomé, Vivancos, Mélanie, Longpré, Jean-Michel, Renault, Pedro, Martinez, Jean, Sarret, Philippe, Cavelier, Florine

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Metabolically stable neurotensin analogs exert potent and long-acting analgesia without hypothermia von Vivancos, Mélanie, Fanelli, Roberto, Besserer-Offroy, Élie, Beaulieu, Sabrina, Chartier, Magali, Resua-Rojas, Martin, Mona, Christine E., Previti, Santo, Rémond, Emmanuelle, Longpré, Jean-Michel, Cavelier, Florine, Sarret, Philippe

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Stereoselective Synthesis of [beta]-(5-Arylthiazolyl) [alpha]-Amino Acids and Use in Neurotensin Analogues von HapAu, Denisa, Remond, Emmanuelle, Fanelli, Roberto, Vivancos, Mélanie, Rene, Adeline, Cote, Jérôme, Besserer-Offroy, Élie, Longpre, Jean-Michel, Martinez, Jean, Zaharia, Valentin, Sarret, Philippe, Cavelier, Florine

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Pharmacological targeting of valosin containing protein (VCP) induces DNA damage and selectively kills canine lymphoma cells von Nadeau, Marie-Ève, Rico, Charlène, Tsoi, Mayra, Vivancos, Mélanie, Filimon, Sabin, Paquet, Marilène, Boerboom, Derek

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Identification of 2-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)tricyclo[3.3.1.13,7]decane-2-carboxylic Acid (NTRC-844) as a Selective Antagonist for t... von Thomas, James B, Vivancos, Mélanie, Giddings, Angela M, Wiethe, Robert W, Warner, Keith R, Murza, Alexandre, Besserer-Offroy, Élie, Longpré, Jean-Michel, Runyon, Scott P, Decker, Ann M, Gilmour, Brian P, Sarret, Philippe

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Stereoselective Synthesis of β-(5-Arylthiazolyl) α-Amino Acids and Use in Neurotensin Analogues von Hapău, Denisa, Rémond, Emmanuelle, Fanelli, Roberto, Vivancos, Mélanie, René, Adeline, Côté, Jérôme, Besserer-Offroy, Élie, Longpré, Jean-Michel, Martinez, Jean, Zaharia, Valentin, Sarret, Philippe, Cavelier, Florine

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Identification of 2-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1 H -pyrazol-3-yl]carbonyl}amino)tricyclo[3.3.1.13,7]decane-2-carboxylic Acid (NTRC-844) as a Selective Antagonist for... von Thomas, James B., Vivancos, Mélanie, Giddings, Angela M., Wiethe, Robert W., Warner, Keith R., Murza, Alexandre, Besserer-Offroy, Élie, Longpré, Jean-Michel, Runyon, Scott P., Decker, Ann M., Gilmour, Brian P., Sarret, Philippe

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Pharmacokinetics and bioequivalence of 2 meloxicam oral dosage formulations in healthy adult horses von Vivancos, Melanie, Barker, Jessica, Engbers, Sarah, Fischer, Carrie, Frederick, Jami, Friedt, Heather, Rybicka, Joanna M, Stastny, Tereza, Banse, Heidi, Cribb, Alastair E

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Metabolically Stable Neurotensin Analogs Exert Potent and Long-Acting Analgesia Without Hypothermia von Vivancos, Mélanie, Fanelli, Roberto, Élie Besserer-Offroy, Beaulieu, Sabrina, Chartier, Magali, Resua-Rojas, Martin, Mona, Christine E, Previti, Santo, Rémond, Emmanuelle, Longpré, Jean-Michel, Cavelier, Florine, Sarret, Philippe

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Identification of 2‑({[1-(4-Fluorophenyl)-5-(2-meth­oxy­phen­yl)‑1H‑pyr­azol-3-yl]­carb­onyl}ami­no)tri­cyclo[3.3.1.13,7]­dec­ane-2-carb­oxy­lic Acid (NTRC-844) as a Selective Anta... von Thomas, James B, Vivancos, Mélanie, Giddings, Angela M, Wiethe, Robert W, Warner, Keith R, Murza, Alexandre, Besserer-Offroy, Élie, Longpré, Jean-Michel, Runyon, Scott P, Decker, Ann M, Gilmour, Brian P, Sarret, Philippe

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Prospective observational study of SARS-CoV-2 infection, transmission and immunity in a cohort of households in Liverpool City Region, UK (COVID-LIV): a study protocol von Setiabudi, Wega, Hungerford, Daniel, Subramaniam, Krishanthi, Vaselli, Natasha Marcella, Shaw, Victoria E, Wilton, Moon, Vivancos, Roberto, Aston, Stephen, Platt, Gareth, Moitt, Tracy, Jones, Ashley P, Gabbay, Mark, Buchan, Iain, Carrol, Enitan D, Iturriza-Gomara, Miren, Solomon, Tom, Greenhalf, William, Naisbitt, Dean J, Adams, Emily R, Cunliffe, Nigel A, Turtle, Lance, French, Neil

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RT-PCR genotyping assays to identify SARS-CoV-2 variants in England in 2021: a design and retrospective evaluation study von Bray, Neil, Sopwith, Will, Edmunds, Matt, Vansteenhouse, Harper, Feenstra, Jelena D M, Jacobs, Peter, Rajput, Kamal, O’Connell, Anne Marie, Smith, Melanie L, Blomquist, Paula, Hatziioanou, Diane, Elson, Richard, Vivancos, Roberto, Gallagher, Eileen, Wigglesworth, Mark J, Dominiczak, Anna, Hopkins, Susan, Lake, Iain R

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Investigation of SARS-CoV-2 faecal shedding in the community: a prospective household cohort study (COVID-LIV) in the UK von Vaselli, Natasha Marcella, Setiabudi, Wega, Subramaniam, Krishanthi, Adams, Emily R., Turtle, Lance, Iturriza-Gomara, Miren, Solomon, Tom, Cunliffe, Nigel A., French, Neil, Hungerford, Daniel

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