Organocatalytic Asymmetric Conjugate Additions to Cyclopent-1-enecarbaldehyde: A Critical Assessment of Organocatalytic Approaches towards the Telaprevir Bicyclic Core von Bernardi, Luca, Fochi, Mariafrancesca, Carbone, Riccardo, Martinelli, Ada, Fox, Martin E., Cobley, Christopher J., Kandagatla, Bhaskar, Oruganti, Srinivas, Dahanukar, Vilas H., Carlone, Armando

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Synthesis and Optimization of Canagliflozin by Employing Quality by Design (QbD) Principles von Metil, Dattatray S, Sonawane, Swapnil P, Pachore, Sharad S, Mohammad, Aaseef, Dahanukar, Vilas H, McCormack, Peter J, Reddy, Ch. Venkatramana, Bandichhor, Rakeshwar

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Investigation of a Kumada Cross Coupling Reaction for Large-Scale Production of (2S, 7R, E)‑2-Isopropyl-7-(4-methoxy-3-(3-methoxypropoxy)benzyl)‑N,N,8-trimethylnon-4-enamide von Gangula, Srinivas, Neelam, Uday Kumar, Baddam, Sudharkar Reddy, Dahanukar, Vilas H, Bandichhor, Rakeshwar

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A morpholine-free process amenable convergent synthesis of apixaban: a potent factor Xa inhibitor von Nevuluri, Narasimha Rao, Rapolu, Rajesh Kumar, Iqbal, Javed, Kandagatla, Bhaskar, Sen, Saikat, Dahanukar, Vilas H., Oruganti, Srinivas

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Practical, Asymmetric Route to Sitagliptin and Derivatives: Development and Origin of Diastereoselectivity von Gutierrez, Osvaldo, Metil, Dattatray, Dwivedi, Namrata, Gudimalla, Nagaraju, Chandrashekar, E. R. R, Dahanukar, Vilas H, Bhattacharya, Apurba, Bandichhor, Rakeshwar, Kozlowski, Marisa C

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Synthesis and Process Optimization of Boceprevir: A Protease Inhibitor Drug von Bhalerao, Dinesh S, Arkala, Anil Kumar Reddy, Madhavi, Y. V, Nagaraju, M, Gade, Srinivas Reddy, Kumar, U. K. Syam, Bandichhor, Rakeshwar, Dahanukar, Vilas H

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Correction to “Synthesis and Optimization of Canagliflozin by Employing Quality by Design (QbD) Principles” von Metil, Dattatray S, Murugan, Andiappan, Sonawane, Swapnil P, Pachore, Sharad S, Mohammad, Aaseef, Dahanukar, Vilas H, McCormack, Peter J, Reddy, Ch. Venkatramana, Bandichhor, Rakeshwar

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One pot oxidative dehydration - oxidation of polyhydroxyhexanal oxime to polyhydroxy oxohexanenitrile: A versatile methodology for the facile access of azasugar alkaloids von Khobare, Sandip R., Gajare, Vikas, Reddy, E. Vishnuvardhan, Datrika, Rajender, Banda, Malavika, Siddaiah, Vidavalur, Pachore, Sharad S., Timanna, Upadhya, Dahanukar, Vilas H., Syam Kumar, U.K.

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Successful utilization of β-ketonitrile in Biginelli reaction: synthesis of 5-cyanodihydropyrimidine von Pachore, Sharad S, Ambhaikar, Narendra B, Siddaiah, Vidavalur, Khobare, Sandip R, Kumar, Sarvesh, Dahanukar, Vilas H, Kumar, U K Syam

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A Practical and Enantiospecific Synthesis of (−)-(R)- and (+)-(S)-Piperidin-3-ols von Suresh Babu, Meruva, Raghunadh, Akula, Ramulu, Konda, Dahanukar, Vilas H., Syam Kumar, Unniaran K., Kumar Dubey, P.

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General Synthesis of α-Acetoxy Ethers from Esters by DIBALH Reduction and Acetylation von Dahanukar, Vilas H, Rychnovsky, Scott D

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New and Practical Method for Synthesis of 1- and 1,3-Substituted Xanthines von Zavialov, Ilia A, Dahanukar, Vilas H, Nguyen, Hoa, Orr, Cecilia, Andrews, David R

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Synthesis, Equilibration, and Coupling of 4-Lithio-1,3-dioxanes:  Synthons for syn- and anti-1,3-Diols von RYCHNOVSKY, Scott D., BUCKMELTER, Alexandre J., DAHANUKAR, Vilas H., SKALITZKY, Donald J.

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Discovery of redox system enabling C–N–C bonds formation: Unprecedented Aza-Cannizzaro reaction von Sud, Abhishek, Chaudhari, Pramod S., Agarwal, Ishu, Mohammad, Amjad Basha, Dahanukar, Vilas H., Bandichhor, Rakeshwar

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Effects of a 3-alkyl-, 4-hydroxy- and/or 8-aromatic-substituent on the phenylethanolamine N-methyltransferase inhibitor potency and α2-adrenoceptor affinity of 2,3,4,5-tetrahydro-1... von GRUNEWALD, Gary L, DAHANUKAR, Vilas H, CRISCIONE, Kevin R

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Development of an Efficient Process for the Preparation of Sch 39166:  Aziridinium Chemistry on Scale von Gala, Dinesh, Dahanukar, Vilas H, Eckert, Jeffery M, Lucas, Brian S, Schumacher, Doris P, Zavialov, Ilia A, Buholzer, Patrik, Kubisch, Peter, Mergelsberg, Ingrid, Scherer, Dominik

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Synthesis of (R)‐3‐(tert‐Butoxycarbonylamino)‐4‐(2,4,5‐trifluorophenyl)butanoic Acid, a Key Intermediate, and the Formal Synthesis of Sitagliptin Phosphate von Sreenivasulu, Kurella, Chaudhari, Pramod S., Achanta, Srinivas, Sud, Abhishek, Dahanukar, Vilas, Cobley, Christopher J., Llewellyn‐Beard, Fiona, Bandichhor, Rakeshwar

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Carbon−Carbon Bond Formation from Small- and Medium-Ring Lactol Acetates via Radical and Oxonium Ion Intermediates. Synthesis of (±)-Laurenan von Rychnovsky, Scott D., Dahanukar, Vilas H.

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Reaction of aziridinium ions with organometallic reagents: optimization of the key step of ecopipam synthesis von Andrews, David R, Dahanukar, Vilas H, Eckert, Jeffrey M, Gala, Dinesh, Lucas, Brian S, Schumacher, Doris P, Zavialov, Ilia A

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Enantiospecific Synthesis of 3-Fluoromethyl-, 3-Hydroxymethyl-, and 3-Chloromethyl-1,2,3,4-tetrahydroisoquinolines as Selective Inhibitors of Phenylethanolamine N-Methyltransferase... von Grunewald, Gary L, Caldwell, Timothy M, Li, Qifang, Dahanukar, Vilas H, McNeil, Brynn, Criscione, Kevin R

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