In Vitro Evaluation of New 5-Nitroindazolin-3-one Derivatives as Promising Agents against Trypanosoma cruzi von Pozo-Martínez, Josué, Arán, Vicente J, Zúñiga-Bustos, Matías, Parra-Magna, Sebastián, Rocha-Valderrama, Esteban, Liempi, Ana, Castillo, Christian, Olea-Azar, Claudio, Moncada-Basualto, Mauricio

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Antimalarial Quinoline Drugs Inhibit β-Hematin and Increase Free Hemin Catalyzing Peroxidative Reactions and Inhibition of Cysteine Proteases von Herraiz, Tomás, Guillén, Hugo, González-Peña, Diana, Arán, Vicente J.

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Identification, occurrence and activity of quinazoline alkaloids in Peganum harmala von Herraiz, Tomás, Guillén, Hugo, Arán, Vicente J., Salgado, Antonio

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Experimental models in Chagas disease: a review of the methodologies applied for screening compounds against Trypanosoma cruzi von Fonseca-Berzal, Cristina, Arán, Vicente J., Escario, José A., Gómez-Barrio, Alicia

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Development of novel benznidazole formulations: Physicochemical characterization and in vivo evaluation on parasitemia reduction in Chagas disease von Palmeiro-Roldán, Ricardo, Fonseca-Berzal, Cristina, Gómez-Barrio, Alicia, Arán, Vicente J., Escario, José A., Torrado-Durán, Susana, Torrado-Santiago, Santiago

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5-Nitroindazole-based compounds: further studies for activity optimization as anti-Trypanosoma cruzi agents von Fonseca-Berzal, Cristina, Ibáñez-Escribano, Alexandra, de Castro, Sonia, Escario, José A., Gómez-Barrio, Alicia, Arán, Vicente J.

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5-Nitroindazole derivatives as potential therapeutic alternatives against Acanthamoeba castellanii von Martín-Escolano, Rubén, Pérez-Cordón, Gregorio, Arán, Vicente J., Marín, Clotilde, Sánchez-Moreno, Manuel, Rosales, María José

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Oxidative Metabolism of the Bioactive and Naturally Occurring β-Carboline Alkaloids, Norharman and Harman, by Human Cytochrome P450 Enzymes von Herraiz, Tomás, Guillén, Hugo, Arán, Vicente J

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Promising hit compounds against resistant trichomoniasis: Synthesis and antiparasitic activity of 3-(ω-aminoalkoxy)-1-benzyl-5-nitroindazoles von Ibáñez-Escribano, Alexandra, Reviriego, Felipe, Vela, Nerea, Fonseca-Berzal, Cristina, Nogal-Ruiz, Juan José, Arán, Vicente J., Escario, José Antonio, Gómez-Barrio, Alicia

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Discovery of nitroheterocycles active against African trypanosomes. In vitro screening and preliminary SAR studies von Arán, Vicente J., Kaiser, Marcel, Dardonville, Christophe

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Antichagasic and trichomonacidal activity of 1-substituted 2-benzyl-5-nitroindazolin-3-ones and 3-alkoxy-2-benzyl-5-nitro-2H-indazoles von Fonseca-Berzal, Cristina, Ibáñez-Escribano, Alexandra, Reviriego, Felipe, Cumella, José, Morales, Paula, Jagerovic, Nadine, Nogal-Ruiz, Juan José, Escario, José Antonio, da Silva, Patricia Bernardino, Soeiro, Maria de Nazaré C., Gómez-Barrio, Alicia, Arán, Vicente J.

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New perspectives on the synthesis and antichagasic activity of 3-alkoxy-1-alkyl-5-nitroindazoles von Muro, Beatriz, Reviriego, Felipe, Navarro, Pilar, Marín, Clotilde, Ramírez-Macías, Inmaculada, Rosales, María José, Sánchez-Moreno, Manuel, Arán, Vicente J.

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Novel solid dispersions of benznidazole: Preparation, dissolution profile and biological evaluation as alternative antichagasic drug delivery system von Fonseca-Berzal, Cristina, Palmeiro-Roldán, Ricardo, Escario, José A., Torrado, Susana, Arán, Vicente J., Torrado-Santiago, Santiago, Gómez-Barrio, Alicia

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Further insights into biological evaluation of new anti-Trypanosoma cruzi 5-nitroindazoles von Fonseca-Berzal, Cristina, Escario, José Antonio, Arán, Vicente J, Gómez-Barrio, Alicia

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In vitro leishmanicidal activity of 1,3-disubstituted 5-nitroindazoles von Marín, Clotilde, Ramírez-Macías, Inmaculada, Rosales, María José, Muro, Beatriz, Reviriego, Felipe, Navarro, Pilar, Arán, Vicente J., Sánchez-Moreno, Manuel

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In vitro assessment of 3-alkoxy-5-nitroindazole-derived ethylamines and related compounds as potential antileishmanial drugs von Martín-Montes, Álvaro, Aguilera-Venegas, Benjamín, Mª Morales-Martín, Rosa, Martín-Escolano, Rubén, Zamora-Ledesma, Salvador, Marín, Clotilde, Arán, Vicente J., Sánchez-Moreno, Manuel

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A sequential procedure for rapid and accurate identification of putative trichomonacidal agents von Ibáñez-Escribano, Alexandra, Meneses-Marcel, Alfredo, Marrero-Ponce, Yovani, Nogal-Ruiz, Juan José, Arán, Vicente J., Gómez-Barrio, Alicia, Escario, José Antonio

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Biological assay of a novel quinoxalinone with antimalarial efficacy on Plasmodium yoelii yoelii von Rivera, Norma, Ponce, Yovani Marrero, Arán, Vicente J., Martínez, Cecilia, Malagón, Filiberto

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Synthesis and in vitro and in vivo biological evaluation of substituted nitroquinoxalin-2-ones and 2,3-diones as novel trichomonacidal agents von Ibáñez-Escribano, Alexandra, Reviriego, Felipe, Nogal-Ruiz, Juan José, Meneses-Marcel, Alfredo, Gómez-Barrio, Alicia, Escario, José Antonio, Arán, Vicente J.

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Study of 5-nitroindazoles' anti- Trypanosoma cruzi mode of action: Electrochemical behaviour and ESR spectroscopic studies von Rodríguez, Jorge, Gerpe, Alejandra, Aguirre, Gabriela, Kemmerling, Ulrike, Piro, Oscar E., Arán, Vicente J., Maya, Juan Diego, Olea-Azar, Claudio, González, Mercedes, Cerecetto, Hugo

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