Toward Structurally Novel and Metabolically Stable HIV-1 Capsid-Targeting Small Molecules von Vernekar, Sanjeev Kumar V., Sahani, Rajkumar Lalji, Casey, Mary C., Kankanala, Jayakanth, Wang, Lei, Kirby, Karen A., Du, Haijuan, Zhang, Huanchun, Tedbury, Philip R., Xie, Jiashu, Sarafianos, Stefan G., Wang, Zhengqiang

Volltext

5‑Arylidenethioxothiazolidinones as Inhibitors of Tyrosyl–DNA Phosphodiesterase I von Sirivolu, Venkata Ramana, Vernekar, Sanjeev Kumar V, Marchand, Christophe, Naumova, Alena, Chergui, Adel, Renaud, Amelie, Stephen, Andrew G, Chen, Feng, Sham, Yuk Y, Pommier, Yves, Wang, Zhengqiang

Volltext

Novel PF74-like small molecules targeting the HIV-1 capsid protein: Balance of potency and metabolic stability von Wang, Lei, Casey, Mary C., Vernekar, Sanjeev Kumar V., Sahani, Rajkumar Lalji, Kirby, Karen A., Du, Haijuan, Zhang, Huanchun, Tedbury, Philip R., Xie, Jiashu, Sarafianos, Stefan G., Wang, Zhengqiang

Volltext

Design, Synthesis and Characterization of HIV-1 CA-Targeting Small Molecules: Conformational Restriction of PF74 von Sahani, Rajkumar Lalji, Diana-Rivero, Raquel, Vernekar, Sanjeev Kumar V., Wang, Lei, Du, Haijuan, Zhang, Huanchun, Castaner, Andres Emanuelli, Casey, Mary C., Kirby, Karen A., Tedbury, Philip R., Xie, Jiashu, Sarafianos, Stefan G., Wang, Zhengqiang

Volltext

Toward Biophysical Probes for the 5-HT3 Receptor: Structure−Activity Relationship Study of Granisetron Derivatives von Vernekar, Sanjeev Kumar V, Hallaq, Hasan Y, Clarkson, Guy, Thompson, Andrew J, Silvestri, Linda, Lummis, Sarah C. R, Lochner, Martin

Volltext

5′-Silylated 3′-1,2,3-triazolyl Thymidine Analogues as Inhibitors of West Nile Virus and Dengue Virus von Vernekar, Sanjeev Kumar V, Qiu, Li, Zhang, Jing, Kankanala, Jayakanth, Li, Hongmin, Geraghty, Robert J, Wang, Zhengqiang

Volltext

Clicking 3′-Azidothymidine into Novel Potent Inhibitors of Human Immunodeficiency Virus von Sirivolu, Venkata Ramana, Vernekar, Sanjeev Kumar V, Ilina, Tatiana, Myshakina, Nataliya S, Parniak, Michael A, Wang, Zhengqiang

Volltext

Design, Synthesis, Biochemical, and Antiviral Evaluations of C6 Benzyl and C6 Biarylmethyl Substituted 2‑Hydroxylisoquinoline-1,3-diones: Dual Inhibition against HIV Reverse Transc... von Vernekar, Sanjeev Kumar V, Liu, Zheng, Nagy, Eva, Miller, Lena, Kirby, Karen A, Wilson, Daniel J, Kankanala, Jayakanth, Sarafianos, Stefan G, Parniak, Michael A, Wang, Zhengqiang

Volltext

Chemical profiling of HIV-1 capsid-targeting antiviral PF74 von Wang, Lei, Casey, Mary C., Vernekar, Sanjeev Kumar V., Do, Ha T., Sahani, Rajkumar Lalji, Kirby, Karen A., Du, Haijuan, Hachiya, Atsuko, Zhang, Huanchun, Tedbury, Philip R., Xie, Jiashu, Sarafianos, Stefan G., Wang, Zhengqiang

Volltext

Double-Winged 3‑Hydroxypyrimidine-2,4-diones: Potent and Selective Inhibition against HIV‑1 RNase H with Significant Antiviral Activity von Vernekar, Sanjeev Kumar V, Tang, Jing, Wu, Bulan, Huber, Andrew D, Casey, Mary C, Myshakina, Nataliya, Wilson, Daniel J, Kankanala, Jayakanth, Kirby, Karen A, Parniak, Michael A, Sarafianos, Stefan G, Wang, Zhengqiang

Volltext

Novel HIV-1 capsid-targeting small molecules of the PF74 binding site von Wang, Lei, Casey, Mary C., Vernekar, Sanjeev Kumar V., Sahani, Rajkumar Lalji, Kankanala, Jayakanth, Kirby, Karen A., Du, Haijuan, Hachiya, Atsuko, Zhang, Huanchun, Tedbury, Philip R., Xie, Jiashu, Sarafianos, Stefan G., Wang, Zhengqiang

Volltext

Synthesis, biological evaluation and molecular modeling of 2-Hydroxyisoquinoline-1,3-dione analogues as inhibitors of HIV reverse transcriptase associated ribonuclease H and polyme... von Tang, Jing, Vernekar, Sanjeev Kumar V., Chen, Yue-Lei, Miller, Lena, Huber, Andrew D., Myshakina, Nataliya, Sarafianos, Stefan G., Parniak, Michael A., Wang, Zhengqiang

Volltext

Mapping the Orthosteric Binding Site of the Human 5‑HT3 Receptor Using Photo-cross-linking Antagonists von Jack, Thomas, Leuenberger, Michele, Ruepp, Marc-David, Vernekar, Sanjeev Kumar V, Thompson, Andrew J, Braga-Lagache, Sophie, Heller, Manfred, Lochner, Martin

Volltext

Mapping the Orthosteric Binding Site of the Human 5-HT 3 Receptor Using Photo-cross-linking Antagonists von Jack, Thomas, Leuenberger, Michele, Ruepp, Marc-David, Vernekar, Sanjeev Kumar V, Thompson, Andrew J, Braga-Lagache, Sophie, Heller, Manfred, Lochner, Martin

Volltext

Synthesis and antiviral evaluation of 4′-(1,2,3-triazol-1-yl)thymidines von Vernekar, Sanjeev Kumar V., Qiu, Li, Zacharias, Jeana, Geraghty, Robert J., Wang, Zhengqiang

Volltext

High-affinity fluorescent ligands for the 5-HT3 receptor von Simonin, Jonathan, Vernekar, Sanjeev Kumar V., Thompson, Andrew J., Hothersall, J. Daniel, Connolly, Christopher N., Lummis, Sarah C.R., Lochner, Martin

Volltext

Synthesis and antiviral evaluation of 4′-(1,2,3-triazol-1-yl)thymidinesElectronic supplementary information (ESI) available: Chemistry, experimental details, and full characterizat... von Vernekar, Sanjeev Kumar V, Qiu, Li, Zacharias, Jeana, Geraghty, Robert J, Wang, Zhengqiang

Volltext

Toward Biophysical Probes for the 5-HT 3 Receptor: Structure−Activity Relationship Study of Granisetron Derivatives von Vernekar, Sanjeev Kumar V., Hallaq, Hasan Y., Clarkson, Guy, Thompson, Andrew J., Silvestri, Linda, Lummis, Sarah C. R., Lochner, Martin

Volltext

High-affinity fluorescent ligands for the 5-HT(3) receptor von Simonin, Jonathan, Vernekar, Sanjeev Kumar V, Thompson, Andrew J, Hothersall, J Daniel, Connolly, Christopher N, Lummis, Sarah C R, Lochner, Martin

Volltext

ChemInform Abstract: Syntheses of Branched Non-1-ynitols by Chemoselective Addition of (Trimethylsilyl)propargylmagnesium Bromide at the Anomeric Center of Side Chain Halogeno Func... von Vernekar, Sanjeev Kumar V., Kipke, Paul, Redlich, Hartmut

Volltext