Chemoenzymatic Conjugation of Toxic Payloads to the Globally Conserved N‑Glycan of Native mAbs Provides Homogeneous and Highly Efficacious Antibody–Drug Conjugates von van Geel, Remon, Wijdeven, Marloes A, Heesbeen, Ryan, Verkade, Jorge M. M, Wasiel, Anna A, van Berkel, Sander S, van Delft, Floris L

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Organocatalysed asymmetric Mannich reactions von Verkade, Jorge M M, van Hemert, Lieke J C, Quaedflieg, Peter J L M, Rutjes, Floris P J T

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Genetic Encoding of a Bicyclo[6.1.0]nonyne-Charged Amino Acid Enables Fast Cellular Protein Imaging by Metal-Free Ligation von Borrmann, Annika, Milles, Sigrid, Plass, Tilman, Dommerholt, Jan, Verkade, Jorge M. M., Wießler, Manfred, Schultz, Carsten, van Hest, Jan C. M., van Delft, Floris L., Lemke, Edward A.

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Process Development for the Enzymatic Gram‐Scale Production of the Unnatural Nucleotide Sugar UDP‐6‐Azido‐GalNAc von Frohnmeyer, Hannes, Verkade, Jorge M. M., Spiertz, Markus, Rentsch, Andreas, Hoffmann, Niels, Sobota, Milan, Schwede, Frank, Tjeerdsma, Peter, Elling, Lothar

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Enzymatic glycan remodeling-metal free click (GlycoConnect™) provides homogenous antibody-drug conjugates with improved stability and therapeutic index without sequence engineering... von Wijdeven, Marloes A., van Geel, Remon, Hoogenboom, Jorin H., Verkade, Jorge M. M., Janssen, Brian M. G., Hurkmans, Inge, de Bever, Laureen, van Berkel, Sander S., van Delft, Floris L.

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Emergence of single-molecular chirality from achiral reactants von Steendam, René R. E., Verkade, Jorge M. M., van Benthem, Tim J. B., Meekes, Hugo, van Enckevort, Willem J. P., Raap, Jan, Rutjes, Floris P. J. T., Vlieg, Elias

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Oligonucleotide tagging for copper-free click conjugation von Jawalekar, Anup M, Malik, Sudip, Verkade, Jorge M M, Gibson, Brian, Barta, Nancy S, Hodges, John C, Rowan, Alan, van Delft, Floris L

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Enantio- and diastereoselective synthesis of γ-amino alcohols von Verkade, Jorge M M, Quaedflieg, Peter J L M, Verzijl, Gerard K M, Lefort, Laurent, van Delft, Floris L, de Vries, Johannes G, Rutjes, Floris P J T

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A Polar Sulfamide Spacer Significantly Enhances the Manufacturability, Stability, and Therapeutic Index of Antibody–Drug Conjugates von Verkade, Jorge, Wijdeven, Marloes, Van Geel, Remon, Janssen, Brian, Van Berkel, Sander, Van Delft, Floris

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An Enantioselective Organocatalytic Approach to Both Enantiomers of Lasubine II von Verkade, Jorge M. M, van der Pijl, Ferdi, Willems, Marian M. J. H. P, Quaedflieg, Peter J. L. M, van Delft, Floris L, Rutjes, Floris P. J. T

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Mild and efficient deprotection of the amine protecting p-methoxyphenyl (PMP) group von Verkade, Jorge M.M., van Hemert, Lieke J.C., Quaedflieg, Peter J.L.M., Alsters, Paul L., van Delft, Floris L., Rutjes, Floris P.J.T.

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Laccase-Mediated Deprotection of para-Methoxyphenyl (PMP)-Protected Amines von Verkade, Jorge M. M., van Hemert, Lieke J. C., Quaedflieg, Peter J. L. M., Schoemaker, Hans E., Schürmann, Martin, van Delft, Floris L., Rutjes, Floris P. J. T.

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Correction: Verkade, J.M.M.; et al. A Polar Sulfamide Spacer Significantly Enhances the Manufacturability, Stability, and Therapeutic Index of Antibody–Drug Conjugates. Antibodies... von Verkade, Jorge, Wijdeven, Marloes, van Geel, Remon, Janssen, Brian, van Berkel, Sander, van Delft, Floris

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Optimizing the Deprotection of the Amine Protecting p-Methoxyphenyl Group in an Automated Microreactor Platform von Koch, Kaspar, van Weerdenburg, Bram J. A, Verkade, Jorge M. M, Nieuwland, Pieter J, Rutjes, Floris P. J. T, van Hest, Jan C. M

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Abstract 3815: Decomposition of parameters contributing to the improved therapeutic index of ADCs obtained by GlycoConnect™ and HydraSpace™ Technologies von Delft, Floris van, Janssen, Brian, Geel, Remon van, Wijdeven, Marloes, Verkade, Jorge, Berkel, Sander van

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A Novel Purification Method in Organic Synthesis Using Hydrogen Bonding von Gruijters, Bas W. T., Verkade, Jorge M. M., van Delft, Floris L., Sijbesma, Rint P., Hermkens, Pedro H. H., Rutjes, Floris P. J. T.

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Enantio- and diastereoselective synthesis of γ-amino alcoholsElectronic supplementary information (ESI) available: Experimental data, characterization data and crystal data and str... von Verkade, Jorge M. M, Quaedflieg, Peter J. L. M, Verzijl, Gerard K. M, Lefort, Laurent, van Delft, Floris L, de Vries, Johannes G, Rutjes, Floris P. J. T

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SYNTHESIS OF ENDO-BICYCLONONENE von VERKADE, Jorge Merijn Mathieu, VAN DELFT, Floris Louis, VAN SCHAIK, Arnoldus Jacobus, VAN BERKEL, Sander Sebastiaan

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ENEDIYNE CONJUGATES von VERKADE, Jorge Merijn Mathieu, VAN DELFT, Floris Louis, HOOGENBOOM, Jorin, VAN BERKEL, Maria Antonia

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METHODS FOR THE PREPARATION OF LINKER PAYLOAD CONSTRUCTS von VERKADE, Jorge Merijn Mathieu, VAN DELFT, Floris Louis, VAN BERKEL, Sander Sebastiaan

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