Syntheses of novel high affinity ligands for opioid receptors von Wentland, Mark P., Lou, Rongliang, Lu, Qun, Bu, Yigong, Denhardt, Christoph, Jin, Jin, Ganorkar, Rakesh, VanAlstine, Melissa A., Guo, Chengyun, Cohen, Dana J., Bidlack, Jean M.

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Structure‐activity relationships for several series of fragment‐based inhibitors that target Trichomonas vaginalis nucleoside ribohydrolase enzymes von Saljanin, Edina, Ajmal, Erum, Vanegas, Davi, VanAlstine‐Parris, Melissa, Stockman, Brian

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Opioids activate brain analgesic circuits through cytochrome P450/epoxygenase signaling von Ding, Xinxin, Hough, Lindsay B, Conroy, Jennie L, Fang, Cheng, Gu, Jun, Zeitlin, Scott O, Yang, Weizhu, Yang, Jun, VanAlstine, Melissa A, Nalwalk, Julia W, Albrecht, Phillip J, Mazurkiewicz, Joseph E, Snyder-Keller, Abigail, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P, Behr, Melissa, Knapp, Brian I, Bidlack, Jean M, Zuiderveld, Obbe P, Leurs, Rob

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Effects of Acetylenic Epoxygenase Inhibitors on Recombinant Cytochrome P450s von VANALSTINE, Melissa A, HOUGH, Lindsay B

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Insight into the Mechanism of the Pechmann Condensation Reaction Using NMR von Tyndall, Stephen, Wong, Koon Fai, VanAlstine-Parris, Melissa A

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Syntheses and opioid receptor binding properties of carboxamido-substituted opioids von Wentland, Mark P., Lou, Rongliang, Lu, Qun, Bu, Yigong, VanAlstine, Melissa A., Cohen, Dana J., Bidlack, Jean M.

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Redefining the structure–activity relationships of 2,6-methano-3-benzazocines. Part 8. High affinity ligands for opioid receptors in the picomolar Ki range: Oxygenated N-(2-[1,1′-b... von Wentland, Mark P., Jo, Sunjin, Gargano, Joseph M., VanAlstine, Melissa A., Cohen, Dana J., Bidlack, Jean M.

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Redefining the structure–activity relationships of 2,6-methano-3-benzazocines. Part 9: Synthesis, characterization and molecular modeling of pyridinyl isosteres of N-BPE-8-CAC (1),... von VanAlstine, Melissa A., Wentland, Mark P., Alvarez, Juan, Cao, Qing, Cohen, Dana J., Knapp, Brian I., Bidlack, Jean M.

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Brain P450 epoxygenase activity is required for the antinociceptive effects of improgan, a nonopioid analgesic von Hough, Lindsay B., Nalwalk, Julia W., Yang, Jun, Conroy, Jennie L., VanAlstine, Melissa A., Yang, Weizhu, Gargano, Joseph, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P., Phillips, James G., Knapp, Brian I., Bidlack, Jean M., Zuiderveld, Obbe P., Leurs, Rob, Ding, Xinxin

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Redefining the structure–activity relationships of 2,6-methano-3-benzazocines. 5. Opioid receptor binding properties of N-((4′-phenyl)-phenethyl) analogues of 8-CAC von VanAlstine, Melissa A., Wentland, Mark P., Cohen, Dana J., Bidlack, Jean M.

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Cytochrome P450 2C24: Expression, Tissue Distribution, High-Throughput Assay, and Pharmacological Inhibition von Yang, Jun, VanAlstine, Melissa A, Phillips, James G, Wentland, Mark P, Hough, Lindsay B

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Determining the IC50 Values for Vorozole and Letrozole, on a Series of Human Liver Cytochrome P450s, to Help Determine the Binding Site of Vorozole in the Liver von Raymond, Lendelle, Rayani, Nikita, Polson, Grace, Sikorski, Kylie, Lian, Ailin, VanAlstine-Parris, Melissa A.

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Determining the IC 50 Values for Vorozole and Letrozole, on a Series of Human Liver Cytochrome P450s, to Help Determine the Binding Site of Vorozole in the Liver von Raymond, Lendelle, Rayani, Nikita, Polson, Grace, Sikorski, Kylie, Lian, Ailin, VanAlstine-Parris, Melissa A

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Synthesis of 7-alkoxy-4-trifluoromethylcoumarins via the von Pechmann reaction catalyzed by molecular iodine von DeGrote, Jami, Tyndall, Stephen, Wong, Koon Fai, VanAlstine-Parris, Melissa

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Structure‐activity relationships of fragment‐based inhibitors of Trichomonas vaginalis adenosine/guanosine preferring nucleoside ribohydrolase von Emilcar, Melissa, Leonardo, Angelica, Li, Tian, Dulloo, Zaafir, Kabir, Nafeesathul Hanan, Gil, Ari, VanAlstine‐Parris, Melissa A., Stockman, Brian J.

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Redefining the Structure−Activity Relationships of 2,6-Methano-3-benzazocines. 4. Opioid Receptor Binding Properties of 8-[N-(4‘-phenyl)-phenethyl)carboxamido] Analogues of Cyclazo... von Wentland, Mark P, VanAlstine, Melissa, Kucejko, Robert, Lou, Rongliang, Cohen, Dana J, Parkhill, Amy L, Bidlack, Jean M

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Brain P450 Epoxygenase Activity is Required for the Antinociceptive Effects of Improgan, a Non-Opioid Analgesic von Hough, Lindsay B., Nalwalk, Julia W., Yang, Jun, Conroy, Jennie L., VanAlstine, Melissa A., Yang, Weizhu, Gargano, Joseph, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P, Phillips, James G., Knapp, Brian I., Bidlack, Jean M., Zuiderveld, Obbe P., Leurs, Rob, Ding, Xinxin

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Preparation of N-hydroxysuccinimido esters via palladium-catalyzed carbonylation of aryl triflates and halides von Lou, Rongliang, VanAlstine, Melissa, Sun, Xufeng, Wentland, Mark P.

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Determining the IC_(50) Values for Vorozole and Letrozole, on a Series of Human Liver Cytochrome P450s, to Help Determine the Binding Site of Vorozole in the Liver von Lendelle Raymond, Nikita Rayani, Grace Polson, Kylie Sikorski, Ailin Lian, Melissa A. VanAlstine-Parris

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Determining the [IC.sub.50] values for vorozole and letrozole, on a series of human liver cytochrome P450s, to help determine the binding site of vorozole in the liver von Raymond, Lendelle, Rayani, Nikita, Polson, Grace, Sikorski, Kylie, Lian, Ailin, VanAlstine-Parris, Melissa A

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