Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models von Teuscher, Kevin B, Chowdhury, Somenath, Meyers, Kenneth M, Tian, Jianhua, Sai, Jiqing, Van Meveren, Mayme, South, Taylor M, Sensintaffar, John L, Rietz, Tyson A, Goswami, Soumita, Wang, Jing, Grieb, Brian C, Lorey, Shelly L, Howard, Gregory C, Liu, Qi, Moore, William J, Stott, Gordon M, Tansey, William P, Lee, Taekyu, Fesik, Stephen W

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Discovery of Potent Orally Bioavailable WD Repeat Domain 5 (WDR5) Inhibitors Using a Pharmacophore-Based Optimization von Teuscher, Kevin B, Meyers, Kenneth M, Wei, Qiangqiang, Mills, Jonathan J, Tian, Jianhua, Alvarado, Joseph, Sai, Jiqing, Van Meveren, Mayme, South, Taylor M, Rietz, Tyson A, Zhao, Bin, Moore, William J, Stott, Gordon M, Tansey, William P, Lee, Taekyu, Fesik, Stephen W

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Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors von Teuscher, Kevin B., Mills, Jonathan J., Tian, Jianhua, Han, Changho, Meyers, Kenneth M., Sai, Jiqing, South, Taylor M., Crow, Mackenzie M., Van Meveren, Mayme, Sensintaffar, John L., Zhao, Bin, Amporndanai, Kangsa, Moore, William J., Stott, Gordon M., Tansey, William P., Lee, Taekyu, Fesik, Stephen W.

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