Identification, substrate specificity, and inhibition of the Streptococcus pneumoniae beta-ketoacyl-acyl carrier protein synthase III (FabH) von Khandekar, S S, Gentry, D R, Van Aller, G S, Warren, P, Xiang, H, Silverman, C, Doyle, M L, Chambers, P A, Konstantinidis, A K, Brandt, M, Daines, R A, Lonsdale, J T

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Expression, Purification, and Crystallization of the Escherichia coli Selenomethionyl β-Ketoacyl–Acyl Carrier Protein Synthase III von Khandekar, Sanjay S., Konstantinidis, Alex K., Silverman, Carol, Janson, Cheryl A., McNulty, Dean E., Nwagwu, Silas, Van Aller, Glenn S., Doyle, Michael L., Kane, James F., Qiu, Xiayang, Lonsdale, John

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First X-ray Cocrystal Structure of a Bacterial FabH Condensing Enzyme and a Small Molecule Inhibitor Achieved Using Rational Design and Homology Modeling von Daines, Robert A, Pendrak, Israil, Sham, Kelvin, Van Aller, Glenn S, Konstantinidis, Alex K, Lonsdale, John T, Janson, Cheryl A, Qiu, Xiayang, Brandt, Martin, Khandekar, Sanjay S, Silverman, Carol, Head, Martha S

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Mechanism of Time-Dependent Inhibition of Polypeptide Deformylase by Actinonin von Van Aller, Glenn S, Nandigama, Ravi, Petit, Chantal M, DeWolf, Walt E, Quinn, Chad J, Aubart, Kelly M, Zalacain, Magdalena, Christensen, Siegfried B, Copeland, Robert A, Lai, Zhihong

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Reversal or nitroglycerin tolerance by the cGMP phosphodiesterase inhibitor zaprinast von Silver, Paul J., Pagani, Edward D., de Garavilla, Lawrence, VanAller, Glenn S., Volberg, Marlo L., Pratt, Phillip F., Buchholz, R.Allan

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Weight loss maintenance in overweight subjects on ad libitum diets with high or low protein content and glycemic index: the DIOGENES trial 12-month results von Aller, E E J G, Larsen, T M, Claus, H, Lindroos, A K, Kafatos, A, Pfeiffer, A, Martinez, J A, Handjieva-Darlenska, T, Kunesova, M, Stender, S, Saris, W H M, Astrup, A, van Baak, M A

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Structural and functional diversity calls for a new classification of ABC transporters von Thomas, Christoph, Aller, Stephen G., Beis, Konstantinos, Carpenter, Elisabeth P., Chang, Geoffrey, Chen, Lei, Dassa, Elie, Dean, Michael, Duong Van Hoa, Franck, Ekiert, Damian, Ford, Robert, Gaudet, Rachelle, Gong, Xin, Holland, I. Barry, Huang, Yihua, Kahne, Daniel K., Kato, Hiroaki, Koronakis, Vassilis, Koth, Christopher M., Lee, Youngsook, Lewinson, Oded, Lill, Roland, Martinoia, Enrico, Murakami, Satoshi, Pinkett, Heather W., Poolman, Bert, Rosenbaum, Daniel, Sarkadi, Balazs, Schmitt, Lutz, Schneider, Erwin, Shi, Yigong, Shyng, Show‐Ling, Slotboom, Dirk J., Tajkhorshid, Emad, Tieleman, D. Peter, Ueda, Kazumitsu, Váradi, András, Wen, Po‐Chao, Yan, Nieng, Zhang, Peng, Zheng, Hongjin, Zimmer, Jochen, Tampé, Robert

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SMYD3 links lysine methylation of MAP3K2 to Ras-driven cancer von Mazur, Pawel K., Reynoird, Nicolas, Khatri, Purvesh, Jansen, Pascal W. T. C., Wilkinson, Alex W., Liu, Shichong, Barbash, Olena, Van Aller, Glenn S., Huddleston, Michael, Dhanak, Dashyant, Tummino, Peter J., Kruger, Ryan G., Garcia, Benjamin A., Butte, Atul J., Vermeulen, Michiel, Sage, Julien, Gozani, Or

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Starches, sugars and obesity von Aller, Erik E J G, Abete, Itziar, Astrup, Arne, Martinez, J Alfredo, van Baak, Marleen A

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EZH2 inhibition as a therapeutic strategy for lymphoma with EZH2-activating mutations von McCabe, Michael T., Ott, Heidi M., Ganji, Gopinath, Korenchuk, Susan, Thompson, Christine, Van Aller, Glenn S., Liu, Yan, Graves, Alan P., III, Anthony Della Pietra, Diaz, Elsie, LaFrance, Louis V., Mellinger, Mark, Duquenne, Celine, Tian, Xinrong, Kruger, Ryan G., McHugh, Charles F., Brandt, Martin, Miller, William H., Dhanak, Dashyant, Verma, Sharad K., Tummino, Peter J., Creasy, Caretha L.

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A DNA Hypomethylation Signature Predicts Antitumor Activity of LSD1 Inhibitors in SCLC von Mohammad, Helai P., Smitheman, Kimberly N., Kamat, Chandrashekhar D., Soong, David, Federowicz, Kelly E., Van Aller, Glenn S., Schneck, Jess L., Carson, Jeffrey D., Liu, Yan, Butticello, Michael, Bonnette, William G., Gorman, Shelby A., Degenhardt, Yan, Bai, Yuchen, McCabe, Michael T., Pappalardi, Melissa B., Kasparec, Jiri, Tian, Xinrong, McNulty, Kenneth C., Rouse, Meagan, McDevitt, Patrick, Ho, Thau, Crouthamel, Michelle, Hart, Timothy K., Concha, Nestor O., McHugh, Charles F., Miller, William H., Dhanak, Dashyant, Tummino, Peter J., Carpenter, Christopher L., Johnson, Neil W., Hann, Christine L., Kruger, Ryan G.

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Smyd3 regulates cancer cell phenotypes and catalyzes histone H4 lysine 5 methylation von Van Aller, Glenn S, Reynoird, Nicolas, Barbash, Olena, Huddleston, Michael, Liu, Shichong, Zmoos, Anne-Flore, McDevitt, Patrick, Sinnamon, Robert, Le, BaoChau, Mas, Gloria, Annan, Roland, Sage, Julien, Garcia, Benjamin A, Tummino, Peter J, Gozani, Or, Kruger, Ryan G

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The cilium: a cellular antenna with an influence on obesity risk von Mariman, Edwin C. M., Vink, Roel G., Roumans, Nadia J. T., Bouwman, Freek G., Stumpel, Constance T. R. M., Aller, Erik E. J. G., van Baak, Marleen A., Wang, Ping

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N-terminal domain of tyrosyl-DNA phosphodiesterase I regulates topoisomerase I-induced toxicity in cells von Brettrager, Evan J., Cuya, Selma M., Tibbs, Zachary E., Zhang, Jun, Falany, Charles N., Aller, Stephen G., van Waardenburg, Robert C. A. M.

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Structure-Based Design of a Novel SMYD3 Inhibitor that Bridges the SAM-and MEKK2-Binding Pockets von Van Aller, Glenn S., Graves, Alan P., Elkins, Patricia A., Bonnette, William G., McDevitt, Patrick J., Zappacosta, Francesca, Annan, Roland S., Dean, Tony W., Su, Dai-Shi, Carpenter, Christopher L., Mohammad, Helai P., Kruger, Ryan G.

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EZH2 Is Required for Germinal Center Formation and Somatic EZH2 Mutations Promote Lymphoid Transformation von Béguelin, Wendy, Popovic, Relja, Teater, Matt, Jiang, Yanwen, Bunting, Karen L., Rosen, Monica, Shen, Hao, Yang, Shao Ning, Wang, Ling, Ezponda, Teresa, Martinez-Garcia, Eva, Zhang, Haikuo, Zheng, Yupeng, Verma, Sharad K., McCabe, Michael T., Ott, Heidi M., Van Aller, Glenn S., Kruger, Ryan G., Liu, Yan, McHugh, Charles F., Scott, David W., Chung, Young Rock, Kelleher, Neil, Shaknovich, Rita, Creasy, Caretha L., Gascoyne, Randy D., Wong, Kwok-Kin, Cerchietti, Leandro, Levine, Ross L., Abdel-Wahab, Omar, Licht, Jonathan D., Elemento, Olivier, Melnick, Ari M.

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ICAM-2 confers a non-metastatic phenotype in neuroblastoma cells by interaction with α-actinin von Feduska, J M, Aller, S G, Garcia, P L, Cramer, S L, Council, L N, van Waardenburg, R C A M, Yoon, K J

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Extreme obesity is associated with variation in genes related to the circadian rhythm of food intake and hypothalamic signaling von Mariman, Edwin C M, Bouwman, Freek G, Aller, Erik E J G, van Baak, Marleen A, Wang, Ping

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Long Residence Time Inhibition of EZH2 in Activated Polycomb Repressive Complex 2 von Van Aller, Glenn S, Pappalardi, Melissa Baker, Ott, Heidi M, Diaz, Elsie, Brandt, Martin, Schwartz, Benjamin J, Miller, William H, Dhanak, Dashyant, McCabe, Michael T, Verma, Sharad K, Creasy, Caretha L, Tummino, Peter J, Kruger, Ryan G

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Identification of Potent, Selective, Cell-Active Inhibitors of the Histone Lysine Methyltransferase EZH2 von Verma, Sharad K, Tian, Xinrong, LaFrance, Louis V, Duquenne, Céline, Suarez, Dominic P, Newlander, Kenneth A, Romeril, Stuart P, Burgess, Joelle L, Grant, Seth W, Brackley, James A, Graves, Alan P, Scherzer, Daryl A, Shu, Art, Thompson, Christine, Ott, Heidi M, Aller, Glenn S. Van, Machutta, Carl A, Diaz, Elsie, Jiang, Yong, Johnson, Neil W, Knight, Steven D, Kruger, Ryan G, McCabe, Michael T, Dhanak, Dashyant, Tummino, Peter J, Creasy, Caretha L, Miller, William H

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