Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer von Lücking, Ulrich, Scholz, Arne, Lienau, Philip, Siemeister, Gerhard, Kosemund, Dirk, Bohlmann, Rolf, Briem, Hans, Terebesi, Ildiko, Meyer, Kirstin, Prelle, Katja, Denner, Karsten, Bömer, Ulf, Schäfer, Martina, Eis, Knut, Valencia, Ray, Ince, Stuart, von Nussbaum, Franz, Mumberg, Dominik, Ziegelbauer, Karl, Klebl, Bert, Choidas, Axel, Nussbaumer, Peter, Baumann, Matthias, Schultz‐Fademrecht, Carsten, Rühter, Gerd, Eickhoff, Jan, Brands, Michael

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Multiple Attack on Bacteria by the New Antibiotic Teixobactin von von Nussbaum, Franz, Süssmuth, Roderich D

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Probing the catalytic functions of Bub1 kinase using the small molecule inhibitors BAY-320 and BAY-524 von Baron, Anna P, von Schubert, Conrad, Cubizolles, Fabien, Siemeister, Gerhard, Hitchcock, Marion, Mengel, Anne, Schröder, Jens, Fernández-Montalván, Amaury, von Nussbaum, Franz, Mumberg, Dominik, Nigg, Erich A

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Industrial Organic Synthesis in Life Sciences – Today and Tomorrow von Nising, Carl F., Nussbaum, Franz

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Platensimycin, a New Antibiotic and "Superbug Challenger" from Nature von Häbich, Dieter, von Nussbaum, Franz

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Antibacterial Natural Products in Medicinal Chemistry-Exodus or Revival? von von Nussbaum, Franz, Brands, Michael, Hinzen, Berthold, Weigand, Stefan, Häbich, Dieter

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BAY 1024767 blocks androgen receptor mutants found in castration-resistant prostate cancer patients von Sugawara, Tatsuo, Lejeune, Pascale, Köhr, Silke, Neuhaus, Roland, Faus, Hortensia, Gelato, Kathy A, Busemann, Matthias, Cleve, Arwed, Lücking, Ulrich, von Nussbaum, Franz, Brands, Michael, Mumberg, Dominik, Jung, Klaus, Stephan, Carsten, Haendler, Bernard

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Frontiers in Medicinal Chemistry 2022 Goes Virtual von Diamanti, Eleonora, Méndez, María, Ross, Tatjana, Kuttruff, Christian A., Lefranc, Julien, Klingler, Franca‐Maria, Nussbaum, Franz, Jung, Manfred, Gehringer, Matthias

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Aspergillomarasmine A, an Inhibitor of Bacterial Metallo-β-Lactamases Conferring blaNDM and blaVIM Resistance von von Nussbaum, Franz, Schiffer, Guido

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European Medicinal Chemistry Leaders in Industry (EMCL) – On the Status and Future of Medicinal Chemistry Research in Europe von Ali, Amjad, Bauser, Marcus, Bertrand, Sophie, Blackaby, Wesley, Boss, Christoph, Bossart, Martin, Hall, Adrian, Binch, Hayley, Czechtizky, Werngard, Gijsen, Harrie, Haning, Helmut, Hartung, Ingo V., Kilburn, Paul, Lassalle, Gilbert, Lücking, Ulrich, Mack, Jürgen, Missbach, Martin, Otsomaa, Leena, Torrens, Antoni, Wagner, Michael, Walter, Magnus, Weinstabl, Harald, Hijfte, Luc, Nussbaum, Franz

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Structure and Total Synthesis of Lysobactin (Katanosin B) von von Nussbaum, Franz, Anlauf, Sonja, Benet-Buchholz, Jordi, Häbich, Dieter, Köbberling, Johannes, Musza, László, Telser, Joachim, Rübsamen-Waigmann, Helga, Brunner, Nina A.

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Lost in Transcription--Inhibition of RNA Polymerase von Haebich, Dieter, von Nussbaum, Franz

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The potent AMPK inhibitor BAY-3827 shows strong efficacy in androgen-dependent prostate cancer models von Lemos, Clara, Schulze, Volker K., Baumgart, Simon J., Nevedomskaya, Ekaterina, Heinrich, Tobias, Lefranc, Julien, Bader, Benjamin, Christ, Clara D., Briem, Hans, Kuhnke, Lara P., Holton, Simon J., Bömer, Ulf, Lienau, Philip, von Nussbaum, Franz, Nising, Carl F., Bauser, Marcus, Hägebarth, Andrea, Mumberg, Dominik, Haendler, Bernard

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Potent and Selective Human Neutrophil Elastase Inhibitors with Novel Equatorial Ring Topology: in vivo Efficacy of the Polar Pyrimidopyridazine BAY-8040 in a Pulmonary Arterial Hyp... von von Nussbaum, Franz, Li, Volkhart M., Meibom, Daniel, Anlauf, Sonja, Bechem, Martin, Delbeck, Martina, Gerisch, Michael, Harrenga, Axel, Karthaus, Dagmar, Lang, Dieter, Lustig, Klemens, Mittendorf, Joachim, Schäfer, Martina, Schäfer, Stefan, Schamberger, Jens

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Total Synthesis and Initial Structure-Activity Relationships of Longicatenamycin A von von Nussbaum, Franz, Anlauf, Sonja, Freiberg, Christoph, Benet-Buchholz, Jordi, Schamberger, Jens, Henkel, Thomas, Schiffer, Guido, Häbich, Dieter

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Abstract 2718: Synthesis and characterization of novel benzylpyrazole-based BUB1 kinase inhibitors with anti-tumor activity von Hitchcock, Marion, Siemeister, Gerhard, Briem, Hans, Fernandez-Montalvan, Amaury Ernest, Holton, Simon, Mengel, Anne, Mönning, Ursula, Brands, Michael, Ziegelbauer, Karl, Mumberg, Dominik, Nussbaum, Franz von

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Abstract 3022: BAY 1143572, a first-in-class, highly selective, potent and orally available inhibitor of PTEFb/CDK9 currently in Phase I, shows convincing anti-tumor activity in pr... von Scholz, Arne, Oellerich, Thomas, Hussain, Akhtar, Lindner, Sarah, Luecking, Ulrich, Walter, Annette O., Ellinghaus, Peter, Valencia, Ray, von Nussbaum, Franz, Mumberg, Dominik, Brands, Michael, Ince, Stuart, Serve, Hubert, Ziegelbauer, Karl

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A Rapid Total Synthesis of Spirotryprostatin B: Proof of Its Relative and Absolute Stereochemistry von von Nussbaum, Franz, Danishefsky, Samuel J.

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Front Cover: Industrial Organic Synthesis in Life Sciences – Today and Tomorrow (Eur. J. Org. Chem. 17/2022) von Nising, Carl F., Nussbaum, Franz

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"Superbugs Bunny" Outsmarts Our Immune Defense von Haebich, Dieter, von Nussbaum, Franz

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