General Synthesis of N‑Alkylindoles from N,N‑Dialkylanilines via [4 + 1] Annulative Double C–H Functionalization von Zhang, Bowen, Erb, Frederik R., Vasilopoulos, Aristidis, Voight, Eric A., Alexanian, Erik J.

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Foslevodopa/Foscarbidopa: A New Subcutaneous Treatment for Parkinson's Disease von Rosebraugh, Matthew, Voight, Eric A., Moussa, Ehab M., Jameel, Feroz, Lou, Xiaochun, Zhang, Geoff G. Z., Mayer, Peter T., Stolarik, Deanne, Carr, Robert A., Enright, Brian P., Liu, Wei, Facheris, Maurizio F., Kym, Philip R.

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Diversifying chemical space of DNA-encoded libraries: synthesis of 2-oxa-1-azaspiro(bicyclo[3.2.0])heptanes on-DNA via visible light-mediated energy transfer catalysis von Matsuo, Bianca, Kim, Saegun, Shreiber, Scott T, Levitre, Guillaume, Li, Longbo, Crane, Erika A, McClain, Edward J, Voight, Eric A, Molander, Gary A

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Parkinson’s Disease: Advances in Treatment and the Syntheses of Various Classes of Pharmaceutical Drug Substances von Hill, David R., Huters, Alexander D., Towne, Timothy B., Reddy, Rajarathnam E., Fogle, Jace L., Voight, Eric A., Kym, Philip R.

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Synthesis of Substituted Cyclopropanecarboxylates via Room Temperature Palladium-Catalyzed α‑Arylation of Reformatsky Reagents von Greszler, Stephen N, Halvorsen, Geoff T, Voight, Eric A

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Dearomative intermolecular [2 + 2] photocycloaddition for construction of C(sp)-rich heterospirocycles on-DNA von Li, Longbo, Matsuo, Bianca, Levitre, Guillaume, McClain, Edward J, Voight, Eric A, Crane, Erika A, Molander, Gary A

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Asymmetric synthesis of pharmaceutically relevant 1-aryl-2-heteroaryl- and 1,2-diheteroarylcyclopropane-1-carboxylates von Sharland, Jack C, Wei, Bo, Hardee, David J, Hodges, Timothy R, Gong, Wei, Voight, Eric A, Davies, Huw M. L

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Lithioarene Cycliacylation and Pd-Catalyzed Aminoethylation/Cyclization to Access Electronically Diverse Saturated Isoquinoline Derivatives von Buchman, Marek, Farney, Elliot P, Greszler, Stephen N, Altenbach, Robert J, Gfesser, Gregory A, Voight, Eric A

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Scale-Up of a Continuous Extraction Process for Driving an Equilibrium-Limited Reaction to Completion von Tudesco, Michael T, Moschetta, Eric G, Voight, Eric A

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Scalable Asymmetric Syntheses of Foslevodopa and Foscarbidopa Drug Substances for the Treatment of Parkinson’s Disease von Huters, Alexander D, Stambuli, James, Klix, Russell C, Matulenko, Mark A, Chan, Vincent S, Simanis, Justin, Hill, David R, Reddy, Rajarathnam E, Towne, Timothy B, Bellettini, John R, Kotecki, Brian J, Cardinal-David, Benoit, Ji, Jianguo, Voight, Eric A, Shou, Minshan, Balaraman, Selvakumar, Ashok, Abhishek, Ghosh, Soma

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Synthesis of ABBV-168, a 2′-Bromouridine for the Treatment of Hepatitis C von Voight, Eric A, Brown, Brian S, Greszler, Stephen N, Halvorsen, Geoff T, Zhao, Gang, Kruger, Albert W, Hartung, John, Lukin, Kirill A, Martinez, Steven R, Moschetta, Eric G, Tudesco, Michael T, Ide, Nathan D

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Structure−Activity Relationship Studies on a Series of Novel, Substituted 1-Benzyl-5-phenyltetrazole P2X7 Antagonists von Nelson, Derek W, Gregg, Robert J, Kort, Michael E, Perez-Medrano, Arturo, Voight, Eric A, Wang, Ying, Grayson, George, Namovic, Marian T, Donnelly-Roberts, Diana L, Niforatos, Wende, Honore, Prisca, Jarvis, Michael F, Faltynek, Connie R, Carroll, William A

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Pharmacology of modality-specific transient receptor potential vanilloid-1 antagonists that do not alter body temperature von Reilly, Regina M, McDonald, Heath A, Puttfarcken, Pamela S, Joshi, Shailen K, Lewis, LaGeisha, Pai, Madhavi, Franklin, Pamela H, Segreti, Jason A, Neelands, Torben R, Han, Ping, Chen, Jun, Mantyh, Patrick W, Ghilardi, Joseph R, Turner, Teresa M, Voight, Eric A, Daanen, Jerome F, Schmidt, Robert G, Gomtsyan, Arthur, Kort, Michael E, Faltynek, Connie R, Kym, Philip R

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Synthesis of A‑9758, an Inverse Agonist of Retinoic Acid-Related Orphan Receptor γt von Marvin, Christopher C., Greszler, Stephen N., Shelat, Bhadra H., Voight, Eric A.

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Discovery of (R)‑1-(7-Chloro-2,2-bis(fluoromethyl)chroman-4-yl)-3-(3-methylisoquinolin-5-yl)urea (A-1165442): A Temperature-Neutral Transient Receptor Potential Vanilloid‑1 (TRPV1)... von Voight, Eric A, Gomtsyan, Arthur R, Daanen, Jerome F, Perner, Richard J, Schmidt, Robert G, Bayburt, Erol K, DiDomenico, Stanley, McDonald, Heath A, Puttfarcken, Pamela S, Chen, Jun, Neelands, Torben R, Bianchi, Bruce R, Han, Ping, Reilly, Regina M, Franklin, Pamela H, Segreti, Jason A, Nelson, Richard A, Su, Zhi, King, Andrew J, Polakowski, James S, Baker, Scott J, Gauvin, Donna M, Lewis, LaGeisha R, Mikusa, Joseph P, Joshi, Shailen K, Faltynek, Connie R, Kym, Philip R, Kort, Michael E

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TRENCHING & EXCAVATION SAFETY: Q&A With Eric Voight von Voight, Eric

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Synthesis of (+)-Didemniserinolipid B via Ketalization/Ring-Closing Metathesis von Marvin, Christopher C, Voight, Eric A, Burke, Steven D

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Synthesis of (+)-Didemniserinolipid B: Application of a 2-Allyl-4-fluorophenyl Auxiliary for Relay Ring-Closing Metathesis von Marvin, Christopher C, Voight, Eric A, Suh, Judy M, Paradise, Christopher L, Burke, Steven D

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Target-Directed Synthesis of Antibacterial Drug Candidate GSK966587 von Voight, Eric A, Yin, Hao, Downing, Susan V, Calad, Stacie A, Matsuhashi, Hayao, Giordano, Ilaria, Hennessy, Alan J, Goodman, Richard M, Wood, Jeffery L

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Synthesis and Pharmacology of (Pyridin-2-yl)methanol Derivatives as Novel and Selective Transient Receptor Potential Vanilloid 3 Antagonists von Gomtsyan, Arthur, Schmidt, Robert G, Bayburt, Erol K, Gfesser, Gregory A, Voight, Eric A, Daanen, Jerome F, Schmidt, Diana L, Cowart, Marlon D, Liu, Huaqing, Altenbach, Robert J, Kort, Michael E, Clapham, Bruce, Cox, Phil B, Shrestha, Anurupa, Henry, Rodger, Whittern, David N, Reilly, Regina M, Puttfarcken, Pamela S, Brederson, Jill-Desiree, Song, Ping, Li, Bin, Huang, Susan M, McDonald, Heath A, Neelands, Torben R, McGaraughty, Steve P, Gauvin, Donna M, Joshi, Shailen K, Banfor, Patricia N, Segreti, Jason A, Shebley, Mohamad, Faltynek, Connie R, Dart, Michael J, Kym, Philip R

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