Novel Nanomolar Allosteric Modulators of AMPA Receptor of Bis(pyrimidine) Series: Synthesis, Biotesting and SAR Analysis von Sedenkova, Kseniya N, Zverev, Denis V, Nazarova, Anna A, Lavrov, Mstislav I, Radchenko, Eugene V, Grishin, Yuri K, Gabrel'yan, Alexey V, Zamoyski, Vladimir L, Grigoriev, Vladimir V, Averina, Elena B, Palyulin, Vladimir A

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New Adamantane-Containing Edaravone Conjugates as Potential Neuroprotective Agents for ALS Treatments von Lapshina, Maria A, Shevtsova, Elena F, Grigoriev, Vladimir V, Aksinenko, Aleksey Yu, Ustyugov, Aleksey A, Steinberg, Daniil A, Maleev, Grigoriy V, Dubrovskaya, Elena S, Goreva, Tatiana V, Epishina, Tatiana A, Zamoyski, Vladimir L, Makhaeva, Galina F, Fisenko, Vladimir P, Veselov, Ivan M, Vinogradova, Daria V, Bachurin, Sergey O

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A Facile Approach to Bis(isoxazoles), Promising Ligands of the AMPA Receptor von Vasilenko, Dmitry A., Sadovnikov, Kirill S., Sedenkova, Kseniya N., Karlov, Dmitry S., Radchenko, Eugene V., Grishin, Yuri K., Rybakov, Victor B., Kuznetsova, Tamara S., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Palyulin, Vladimir A., Averina, Elena B.

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Conjugation of Aminoadamantane and γ-Carboline Pharmacophores Gives Rise to Unexpected Properties of Multifunctional Ligands von Bachurin, Sergey O., Makhaeva, Galina F., Shevtsova, Elena F., Aksinenko, Alexey Yu, Grigoriev, Vladimir V., Shevtsov, Pavel N., Goreva, Tatiana V., Epishina, Tatiana A., Kovaleva, Nadezhda V., Pushkareva, Elena A., Boltneva, Natalia P., Lushchekina, Sofya V., Gabrelyan, Alexey V., Zamoyski, Vladimir L., Dubova, Lyudmila G., Rudakova, Elena V., Fisenko, Vladimir P., Bovina, Elena V., Richardson, Rudy J.

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5-Nitroisoxazoles in SNAr Reactions: A Novel Chemo- and Regioselective Approach to Isoxazole-Based Bivalent Ligands of AMPA Receptors von Vasilenko, Dmitry A., Temnyakova, Nadezhda S., Dronov, Sevastian E., Radchenko, Eugene V., Grishin, Yuri K., Gabrel’yan, Alexey V., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Averina, Elena B., Palyulin, Vladimir A.

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Conjugates of γ-Carbolines and Phenothiazine as new selective inhibitors of butyrylcholinesterase and blockers of NMDA receptors for Alzheimer Disease von Makhaeva, Galina F., Lushchekina, Sofya V., Boltneva, Natalia P., Sokolov, Vladimir B., Grigoriev, Vladimir V., Serebryakova, Olga G., Vikhareva, Ekaterina A., Aksinenko, Alexey Yu, Barreto, George E., Aliev, Gjumrakch, Bachurin, Sergey O.

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Novel conjugates of aminoadamantanes with carbazole derivatives as potential multitarget agents for AD treatment von Bachurin, Sergey O., Shevtsova, Elena F., Makhaeva, Galina F., Grigoriev, Vladimir V., Boltneva, Natalia P., Kovaleva, Nadezhda V., Lushchekina, Sofya V., Shevtsov, Pavel N., Neganova, Margarita E., Redkozubova, Olga M., Bovina, Elena V., Gabrelyan, Alexey V., Fisenko, Vladimir P., Sokolov, Vladimir B., Aksinenko, Alexey Yu, Echeverria, Valentina, Barreto, George E., Aliev, Gjumrakch

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Positive and negative AMPA receptor modulators based on tricyclic bispidine derivative: Minor structural change inverts the type of activity von Lavrov, Mstislav I., Veremeeva, Polina N., Golubeva, Elena A., Radchenko, Eugene V., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Palyulin, Vladimir A.

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Novel Positive Allosteric Modulators of AMPA Receptors Based on 3,7-Diazabicyclo[3.3.1]nonane Scaffold von Lavrov, Mstislav I., Karlov, Dmitry S., Voronina, Tatiana A., Grigoriev, Vladimir V., Ustyugov, Aleksey A., Bachurin, Sergey O., Palyulin, Vladimir A.

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Conjugates of Methylene Blue with Cycloalkaneindoles as New Multifunctional Agents for Potential Treatment of Neurodegenerative Disease von Bachurin, Sergey O, Shevtsova, Elena F, Makhaeva, Galina F, Aksinenko, Alexey Yu, Grigoriev, Vladimir V, Goreva, Tatiana V, Epishina, Tatiana A, Kovaleva, Nadezhda V, Boltneva, Natalia P, Lushchekina, Sofya V, Rudakova, Elena V, Vinogradova, Darya V, Shevtsov, Pavel N, Pushkareva, Elena A, Dubova, Ludmila G, Serkova, Tatiana P, Veselov, Ivan M, Fisenko, Vladimir P, Richardson, Rudy J

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Bivalent AMPA receptor positive allosteric modulators of the bis(pyrimidine) series von Nazarova, Anna A, Sedenkova, Kseniya N, Karlov, Dmitry S, Lavrov, Mstislav I, Grishin, Yuri K, Kuznetsova, Tamara S, Zamoyski, Vladimir L, Grigoriev, Vladimir V, Averina, Elena B, Palyulin, Vladimir A

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Biphenyl scaffold for the design of NMDA-receptor negative modulators: molecular modeling, synthesis, and biological activity von Karlov, Dmitry S, Temnyakova, Nadezhda S, Vasilenko, Dmitry A, Barygin, Oleg I, Dron, Mikhail Y, Zhigulin, Arseniy S, Averina, Elena B, Grishin, Yuri K, Grigoriev, Vladimir V, Gabrel'yan, Alexey V, Aniol, Viktor A, Gulyaeva, Natalia V, Osipenko, Sergey V, Kostyukevich, Yury I, Palyulin, Vladimir A, Popov, Petr A, Fedorov, Maxim V

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5-Nitroisoxazoles in ISNAr/I Reactions: A Novel Chemo- and Regioselective Approach to Isoxazole-Based Bivalent Ligands of AMPA Receptors von Vasilenko, Dmitry A, Temnyakova, Nadezhda S, Dronov, Sevastian E, Radchenko, Eugene V, Grishin, Yuri K, Gabrel’yan, Alexey V, Zamoyski, Vladimir L, Grigoriev, Vladimir V, Averina, Elena B, Palyulin, Vladimir A

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Synthesis and modulatory activity of 3-acetyl-7-(benzofuran-5-carbonyl)-1,5-dimethyl-3,7-diazabicyclo[3.3.1]nonan-9-one on AMPA receptors von Matthews, James, Veremeeva, Polina N., Golubeva, Elena A., Lavrov, Mstislav I., Radchenko, Eugene V., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Palyulin, Vladimir A.

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Tricyclic derivatives of bispidine as AMPA receptor allosteric modulators von Lavrov, Mstislav I., Veremeeva, Polina N., Karlov, Dmitry S., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Palyulin, Vladimir A.

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CHANGES IN THE PROPERTIES OF PERMANENT JOINTS DEPENDING ON THE MANUFACTURING PROCESSES OF LARGE-SIZE POWER TITANIUM STRUCTURES OF AIRCRAFT MADE BY ELECTRON BEAM WELDING von Grigoriev, Vladimir V., Muravyev, Vasily I., Bakhmatov, Pavel V.

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CERAMIC COATINGS ON A CARBIDE TOOL FOR TURNING STAINLESS HARD-TO-WORK STEELS von Mokritskii, Boris Ya, Sablin, Pavel A., Grigoriev, Vladimir V., Shelkovnikov, Vadim Yu

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Synthesis of an allosteric modulator of ionotropic glutamate receptors von Lavrov, Mstislav I., Stroganov, Oleg V., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Zapolskiy, Maxim E., Sysolyatin, Sergey V., Malykhin, Valeriy V., Surmachev, Vladimir N., Palyulin, Vladimir A.

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Novel positive allosteric modulator of AMPA-receptors based on tricyclic scaffold von Lavrov, Mstislav I., Karlov, Dmitry S., Palyulin, Vladimir A., Grigoriev, Vladimir V., Zamoyski, Vladimir L., Brkich, Galina E., Pyatigorskaya, Natalia V., Zapolskiy, Maxim E.

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Novel bivalent positive allosteric AMPA receptor modulator of bis-amide series von Temnyakova, Nadezhda S., Vasilenko, Dmitry A., Lavrov, Mstislav I., Karlov, Dmitry S., Grishin, Yuri K., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Averina, Elena B., Palyulin, Vladimir A.

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