A Scalable Synthesis of a 1,7-Naphthyridine Derivative, a PDE-4 Inhibitor von Jiang, Xinglong, Lee, George T, Villhauer, Edwin B, Prasad, Kapa, Prashad, Mahavir

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NVP-DPP728 (1-[[[2-[(5-Cyanopyridin-2-yl)amino]ethyl]amino]acetyl]-2-cyano-(S)-pyrrolidine), a Slow-Binding Inhibitor of Dipeptidyl Peptidase IV von Hughes, Thomas E, Mone, Manisha D, Russell, Mary E, Weldon, Stephen C, Villhauer, Edwin B

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1-[[(3-Hydroxy-1-adamantyl)amino]acetyl]-2-cyano-(S)-pyrrolidine:  A Potent, Selective, and Orally Bioavailable Dipeptidyl Peptidase IV Inhibitor with Antihyperglycemic Properties... von Villhauer, Edwin B, Brinkman, John A, Naderi, Goli B, Burkey, Bryan F, Dunning, Beth E, Prasad, Kapa, Mangold, Bonnie L, Russell, Mary E, Hughes, Thomas E

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Facile and practical synthesis of a cannabinoid-1 antagonist via regio- and stereoselective ring-opening of an aziridinium ion von Villhauer, Edwin B., Shieh, Wen-Chung, Du, Zhengming, Vargas, Kevin, Ciszewski, Lech, Lu, Yansong, Girgis, Michael, Lin, Melissa, Prashad, Mahavir

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Conformation of [1-13C,15N]Acetyl-L-carnitine. Rotational-Echo, Double-Resonance Nuclear Magnetic Resonance Spectroscopy von Anderson, Robert C, Gullion, Terry, Joers, Jim M, Shapiro, Michael, Villhauer, Edwin B, Weber, Hans Peter

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Kinetically Controlled Diastereoselective Synthesis of CPS124, a Carnitine Monothiophosphate von Prasad, Kapa, Xu, David D, Tempkin, Orin, Villhauer, Edwin B, Repič, Oljan

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Application of a transition-metal-mediated stereospecific Michael reaction equivalent to the synthesis of alloyohimbone von Godleski, Stephen A, Villhauer, Edwin B

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1-[2-[(5-Cyanopyridin-2-yl)amino]ethylamino]acetyl-2-(S)-pyrrolidinecarbonitrile:  A Potent, Selective, and Orally Bioavailable Dipeptidyl Peptidase IV Inhibitor with Antihyperglyc... von Villhauer, Edwin B, Brinkman, John A, Naderi, Goli B, Dunning, Beth E, Mangold, Bonnie L, Mone, Manisha D, Russell, Mary E, Weldon, Stephen C, Hughes, Thomas E

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Antidiabetic agents: a new class of reversible carnitine palmitoyltransferase I inhibitors von Anderson, Robert C, Balestra, Michael, Bell, Philip A, Deems, Rhonda O, Fillers, William S, Foley, James E, Fraser, James D, Mann, William R, Rudin, Markus, Villhauer, Edwin B

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Metal-catalyzed stereospecific Michael reaction equivalent von Godleski, Stephen A, Villhauer, Edwin B

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Synthesis of the CDE ring system of the ginkgolides von Villhauer, Edwin B, Anderson, Robert C

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1-[2-[(5-Cyanopyridin-2-yl)amino]-ethylamino]acetyl-2-(S)-pyrrolidine-carbonitri le: A potent, selective, and orally bioavailable Dipeptidyl peptidase IV inhibitor with antihypergl... von VILLHAUER, Edwin B, BRINKMAN, John A, NADERI, Goli B, DUNNING, Beth E, MANGOLD, Bonnie L, MONE, Manisha D, RUSSELL, Mary E, WELDON, Stephen C, HUGHES, Thomas E

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The individual enantiomers of cis-cromakalim possess K + channel opening activity von Quast, Ulrich, Villhauer, Edwin B.

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Use of DPP-IV inhibitor to reduce hypoglycemic events von VILLHAUER EDWIN B, BALKAN BOERK, HUGHES THOMAS E, HOLMES DAVID G

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Use of DPP-IV inhibitor to reduce hypoglycemic events von Balkan, Boerk, Holmes, David G, Hughes, Thomas E, Villhauer, Edwin B

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COMBINATIONS COMPRISING DEPEPTIDYPEPTIDASE-IV INHIBITORS AND ANTIDIABETIC AGENTS von VILLHAUER EDWIN B, HUGHES THOMAS E, BALKAN BORK, HOLMES DAVID G

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Process For The Preparation Of 6, 8-Subs Tituted '1, 7 Naphthpyridin Derivatives By Reacting The 8-Halo-'1, 7 Naphthpyrid In-Derivate With An Organic Boronic Acid Derivatives And I... von VILLHAUER EDWIN B, KAPA PRASAD K, JIANG XINGLONG, LEE GEORGE T

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Phosphinyloxy propanaminium inner salt derivatives von ANDERSON, ROBERT C, HUGHES, JEFFREY W, FRASER, JAMES D, VILLHAUER, EDWIN B, BEBERNITZ, GREGORY R, SMITH, HOWARD C

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Diaryl substituted cyclopentane and cyclopentene derivatives von ANDERSON, ROBERT C, HOULIHAN, WILLIAM J, VILLHAUER, EDWIN B, SMITH, HOWARD C

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PHOSPHINYLOXY PROPANAMINIUM INNER SALT DERIVATIVES von VILLHAUER EDWIN B, BEBERNITZ GREGORY R, KAPA PRASAD K, PRASHAD MAHAVIR, SMITH HOWARD C, ANDERSON ROBERT C, HUGHES JEFFREY W, FRASER JAMES

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