Enantioselective Organocatalytic Michael/Aldol Sequence: Anticancer Natural Product (+)-trans-Dihydrolycoricidine von McNulty, James, Zepeda-Velázquez, Carlos

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Targeting of the FOXM1 Oncoprotein by E3 Ligase-Assisted Degradation von Luo, Guoshun, Lin, Xin, Vega-Medina, Antonio, Xiao, Maoxu, Li, Guolong, Wei, Hanlin, Velázquez-Martínez, Carlos A, Xiang, Hua

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Editorial: The use of Baveno VI and VII criteria in patients with hepatocellular carcinoma von Moctezuma‐Velazquez, Carlos, Abraldes, Juan G.

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Discovery of Conformationally Constrained ALK2 Inhibitors von González-Álvarez, Héctor, Ensan, Deeba, Xin, Tao, Wong, Jong Fu, Zepeda-Velázquez, Carlos A., Cros, Julien, Sweeney, Melissa N., Hoffer, Laurent, Kiyota, Taira, Wilson, Brian J., Aman, Ahmed, Roberts, Owen, Isaac, Methvin B., Bullock, Alex N., Smil, David, Al-awar, Rima

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Structure–Activity Relationship of USP5 Inhibitors von Mann, Mandeep K, Zepeda-Velázquez, Carlos A, González-Álvarez, Héctor, Dong, Aiping, Kiyota, Taira, Aman, Ahmed M, Loppnau, Peter, Li, Yanjun, Wilson, Brian, Arrowsmith, Cheryl H, Al-Awar, Rima, Harding, Rachel J, Schapira, Matthieu

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NOSH-aspirin (NBS-1120), a novel nitric oxide- and hydrogen sulfide-releasing hybrid has enhanced chemo-preventive properties compared to aspirin, is gastrointestinal safe with all... von Kodela, Ravinder, Chattopadhyay, Mitali, Velázquez-Martínez, Carlos A., Kashfi, Khosrow

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Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma von Ensan, Deeba, Smil, David, Zepeda-Velázquez, Carlos A, Panagopoulos, Dimitrios, Wong, Jong Fu, Williams, Eleanor P, Adamson, Roslin, Bullock, Alex N, Kiyota, Taira, Aman, Ahmed, Roberts, Owen G, Edwards, Aled M, O’Meara, Jeff A, Isaac, Methvin B, Al-awar, Rima

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Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2 von Ferreira de Freitas, Renato, Liu, Yanli, Szewczyk, Magdalena M, Mehta, Naimee, Li, Fengling, McLeod, David, Zepeda-Velázquez, Carlos, Dilworth, David, Hanley, Ronan P, Gibson, Elisa, Brown, Peter J, Al-Awar, Rima, James, Lindsey I, Arrowsmith, Cheryl H, Barsyte-Lovejoy, Dalia, Min, Jinrong, Vedadi, Masoud, Schapira, Matthieu, Allali-Hassani, Abdellah

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PROTACs in Ovarian Cancer: Current Advancements and Future Perspectives von Vorderbruggen, Makenzie, Velázquez-Martínez, Carlos A, Natarajan, Amarnath, Karpf, Adam R

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Report from a Survey of Parents Regarding the Use of Cannabidiol (Medicinal cannabis) in Mexican Children with Refractory Epilepsy von Aguirre-Velázquez, Carlos G.

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A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6 von Shen, Yudao, Li, Fengling, Szewczyk, Magdalena M, Halabelian, Levon, Chau, Irene, Eram, Mohammad S, Dela Seña, Carlo, Park, Kwang-Su, Meng, Fanye, Chen, He, Zeng, Hong, McLeod, David, Zepeda-Velázquez, Carlos A, Campbell, Robert M, Mader, Mary M, Watson, Brian M, Schapira, Matthieu, Arrowsmith, Cheryl H, Al-Awar, Rima, Barsyte-Lovejoy, Dalia, Kaniskan, H. Ümit, Brown, Peter J, Vedadi, Masoud, Jin, Jian

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The role of training variability for model-based and model-free learning of an arbitrary visuomotor mapping von Velázquez-Vargas, Carlos A, Daw, Nathaniel D, Taylor, Jordan A

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Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1) von Getlik, Matthäus, Smil, David, Zepeda-Velázquez, Carlos, Bolshan, Yuri, Poda, Gennady, Wu, Hong, Dong, Aiping, Kuznetsova, Ekaterina, Marcellus, Richard, Senisterra, Guillermo, Dombrovski, Ludmila, Hajian, Taraneh, Kiyota, Taira, Schapira, Matthieu, Arrowsmith, Cheryl H, Brown, Peter J, Vedadi, Masoud, Al-awar, Rima

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FOXM1 Inhibitors as Potential Diagnostic Agents: First Generation of a PET Probe Targeting FOXM1 To Detect Triple‐Negative Breast Cancer in vitro and in vivo von Pérez, David J., Amirhossein Tabatabaei Dakhili, Seyed, Bergman, Cody, Dufour, Jennifer, Wuest, Melinda, Juengling, Freimut D., Wuest, Frank, Velázquez‐Martínez, Carlos A.

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Autistic traits foster effective curiosity-driven exploration von Poli, Francesco, Koolen, Maran, Velázquez-Vargas, Carlos A, Ramos-Sanchez, Jessica, Meyer, Marlene, Mars, Rogier B, Rommelse, Nanda, Hunnius, Sabine

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Ethanesulfohydroxamic Acid Ester Prodrugs of Nonsteroidal Anti-inflammatory Drugs (NSAIDs): Synthesis, Nitric oxide and Nitroxyl Release, Cyclooxygenase Inhibition, Anti-inflammato... von Huang, Zhangjian, Velázquez, Carlos A, Abdellatif, Khaled R. A, Chowdhury, Morshed A, Reisz, Julie A, DuMond, Jenna F, King, S. Bruce, Knaus, Edward E

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Hydrogen sulfide-releasing NSAIDs inhibit the growth of human cancer cells: A general property and evidence of a tissue type-independent effect von Chattopadhyay, Mitali, Kodela, Ravinder, Nath, Niharika, Dastagirzada, Yosef M., Velázquez-Martínez, Carlos A., Boring, Daniel, Kashfi, Khosrow

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A chemical biology toolbox to study protein methyltransferases and epigenetic signaling von Scheer, Sebastian, Ackloo, Suzanne, Medina, Tiago S., Schapira, Matthieu, Li, Fengling, Ward, Jennifer A., Lewis, Andrew M., Northrop, Jeffrey P., Richardson, Paul L., Kaniskan, H. Ümit, Shen, Yudao, Liu, Jing, Smil, David, McLeod, David, Zepeda-Velazquez, Carlos A., Luo, Minkui, Jin, Jian, Barsyte-Lovejoy, Dalia, Huber, Kilian V. M., De Carvalho, Daniel D., Vedadi, Masoud, Zaph, Colby, Brown, Peter J., Arrowsmith, Cheryl H.

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Synthesis and Chemical and Biological Comparison of Nitroxyl- and Nitric Oxide-Releasing Diazeniumdiolate-Based Aspirin Derivatives von Basudhar, Debashree, Bharadwaj, Gaurav, Cheng, Robert Y, Jain, Sarthak, Shi, Sa, Heinecke, Julie L, Holland, Ryan J, Ridnour, Lisa A, Caceres, Viviane M, Spadari-Bratfisch, Regina C, Paolocci, Nazareno, Velázquez-Martínez, Carlos A, Wink, David A, Miranda, Katrina M

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Patient stress due to surgery postponement in a tertiary referral centre transformed to a COVID-19 hospital von Moctezuma-Velázquez, Paulina, González-Martínez, Carlos A, Buerba, Gabriela A, Serment, Miriam, Moctezuma-Velázquez, Carlos

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