Optimized Inhibitors of MDM2 via an Attempted Protein‐Templated Reductive Amination von Vlag, Ramon, Yagiz Unver, M., Felicetti, Tommaso, Twarda‐Clapa, Aleksandra, Kassim, Fatima, Ermis, Cagdas, Neochoritis, Constantinos G., Musielak, Bogdan, Labuzek, Beata, Dömling, Alexander, Holak, Tad A., Hirsch, Anna K. H.

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Designed Spiroketal Protein Modulation von Scheepstra, Marcel, Andrei, Sebastian A., Unver, M. Yagiz, Hirsch, Anna K. H., Leysen, Seppe, Ottmann, Christian, Brunsveld, Luc, Milroy, Lech‐Gustav

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Modularly Evolved 2‑AminoDMAP/Squaramides as Highly Active Bifunctional Organocatalysts in Michael Addition von Işık, Murat, Unver, M. Yagiz, Tanyeli, Cihangir

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Druggability Assessment of Targets Used in Kinetic Target-Guided Synthesis von Unver, M Yagiz, Gierse, Robin M, Ritchie, Harry, Hirsch, Anna K H

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Stereoselective synthesis of optically active cyclopenta[c]pyridines and tetrahydropyridines von Sezer, Serdar, Gümrükçü, Yasemin, Bakırcı, İrem, Yağız Ünver, M., Tanyeli, Cihangir

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Compounds Interfering with Embryonic Lethal Abnormal Vision (ELAV) Protein-RNA Complexes: An Avenue for Discovering New Drugs von Nasti, Rita, Rossi, Daniela, Amadio, Marialaura, Pascale, Alessia, Unver, M Yagiz, Hirsch, Anna K H, Collina, Simona

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Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction von Mancini, Federica, Unver, M. Yagiz, Elgaher, Walid A. M., Jumde, Varsha R., Alhayek, Alaa, Lukat, Peer, Herrmann, Jennifer, Witte, Martin D., Köck, Matthias, Blankenfeldt, Wulf, Müller, Rolf, Hirsch, Anna K. H.

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Fragment-Based Drug Design Facilitated by Protein-Templated Click Chemistry: Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin von Mondal, Milon, Unver, M. Yagiz, Pal, Asish, Bakker, Matthijs, Berrier, Stephan P., Hirsch, Anna K. H.

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Frontispiece: Protein‐Templated Hit Identification through an Ugi Four‐Component Reaction von Mancini, Federica, Unver, M. Yagiz, Elgaher, Walid A. M., Jumde, Varsha R., Alhayek, Alaa, Lukat, Peer, Herrmann, Jennifer, Witte, Martin D., Köck, Matthias, Blankenfeldt, Wulf, Müller, Rolf, Hirsch, Anna K. H.

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Exploration of ligand binding modes towards the identification of compounds targeting HuR: a combined STD-NMR and Molecular Modelling approach von Vasile, Francesca, Della Volpe, Serena, Ambrosio, Francesca Alessandra, Costa, Giosuè, Unver, M. Yagiz, Zucal, Chiara, Rossi, Daniela, Martino, Emanuela, Provenzani, Alessandro, Hirsch, Anna K. H., Alcaro, Stefano, Potenza, Donatella, Collina, Simona

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Rapid Discovery of Aspartyl Protease Inhibitors Using an Anchoring Approach von Konstantinidou, Markella, Magari, Francesca, Sutanto, Fandi, Haupenthal, Jörg, Jumde, Varsha R., Ünver, M. Yagiz, Heine, Andreas, Camacho, Carlos Jamie, Hirsch, Anna K. H., Klebe, Gerhard, Dömling, Alexander

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Novel Compounds Targeting the RNA-Binding Protein HuR. Structure-Based Design, Synthesis, and Interaction Studies von Della Volpe, Serena, Nasti, Rita, Queirolo, Michele, Unver, M. Yagiz, Jumde, Varsha K, Dömling, Alexander, Vasile, Francesca, Potenza, Donatella, Ambrosio, Francesca Alessandra, Costa, Giosué, Alcaro, Stefano, Zucal, Chiara, Provenzani, Alessandro, Di Giacomo, Marcello, Rossi, Daniela, Hirsch, Anna K. H, Collina, Simona

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Design and Synthesis of Bioisosteres of Acylhydrazones as Stable Inhibitors of the Aspartic Protease Endothiapepsin von Jumde, Varsha R., Mondal, Milon, Gierse, Robin M., Unver, M. Yagiz, Magari, Francesca, van Lier, Roos C. W., Heine, Andreas, Klebe, Gerhard, Hirsch, Anna K. H.

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Designed Spiroketal Protein Modulation von Scheepstra, Marcel, Andrei, Sebastian A., Unver, M. Yagiz, Hirsch, Anna K. H., Leysen, Seppe, Ottmann, Christian, Brunsveld, Luc, Milroy, Lech‐Gustav

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Druggability Assessment of Targets Used in Kinetic Target-Guided Synthesis: Miniperspective von Unver, M. Yagiz, Gierse, Robin M, Ritchie, Harry, Hirsch, Anna K. H

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Compounds Interfering with Embryonic Lethal Abnormal Vision (ELAV) Protein–RNA Complexes: An Avenue for Discovering New Drugs: Miniperspective von Nasti, Rita, Rossi, Daniela, Amadio, Marialaura, Pascale, Alessia, Unver, M. Yagiz, Hirsch, Anna K. H, Collina, Simona

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ChemInform Abstract: Modularly Evolved 2-AminoDMAP/Squaramides as Highly Active Bifunctional Organocatalysts in Michael Addition von Isik, Murat, Unver, M. Yagiz, Tanyeli, Cihangir

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Towards the Modulation of RNA-Binding Proteins: New Compounds Targeting Protein HuR von Serena Della Volpe, Rita Nasti, Michele Queirolo, Yagiz M. Unver, Varsha R. Jumde, Alexander Dömling, Francesca Vasile, Donatella Potenza, Francesca Alessandra Ambrosio, Giosué Costa, Stefano Alcaro, Chiara Zucal, Alessandro Provenzani, Marcello Di Giacomo, Daniela Rossi, Anna K. H. Hirsch, Simona Collina

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