Algorithmic Probability-Guided Machine Learning on Non-Differentiable Spaces von Hernández-Orozco, Santiago, Zenil, Hector, Riedel, Jürgen, Uccello, Adam, Kiani, Narsis A, Tegnér, Jesper

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Visual Representation Learning for Preference-Aware Path Planning von Sikand, Kavan Singh, Rabiee, Sadegh, Uccello, Adam, Xiao, Xuesu, Warnell, Garrett, Biswas, Joydeep

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Algorithmic Probability-guided Supervised Machine Learning on Non-differentiable Spaces von Hernández-Orozco, Santiago, Zenil, Hector, Riedel, Jürgen, Uccello, Adam, Kiani, Narsis A, Tegnér, Jesper

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Visual Representation Learning for Preference-Aware Path Planning von Kavan Singh Sikand, Rabiee, Sadegh, Uccello, Adam, Xiao, Xuesu, Warnell, Garrett, Biswas, Joydeep

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Algorithmic Probability-guided Supervised Machine Learning on Non-differentiable Spaces von Hernández-Orozco, Santiago, Zenil, Hector, Riedel, Jürgen, Uccello, Adam, Kiani, Narsis A, Tegnér, Jesper

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Chemical and Computational Methods for the Characterization of Covalent Reactive Groups for the Prospective Design of Irreversible Inhibitors von Flanagan, Mark E, Abramite, Joseph A, Anderson, Dennis P, Aulabaugh, Ann, Dahal, Upendra P, Gilbert, Adam M, Li, Chao, Montgomery, Justin, Oppenheimer, Stacey R, Ryder, Tim, Schuff, Brandon P, Uccello, Daniel P, Walker, Gregory S, Wu, Yan, Brown, Matthew F, Chen, Jinshan M, Hayward, Matthew M, Noe, Mark C, Obach, R. Scott, Philippe, Laurence, Shanmugasundaram, Veerabahu, Shapiro, Michael J, Starr, Jeremy, Stroh, Justin, Che, Ye

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Delineating the role of cooperativity in the design of potent PROTACs for BTK von Zorba, Adelajda, Nguyen, Chuong, Xu, Yingrong, Starr, Jeremy, Borzilleri, Kris, Smith, James, Zhu, Hongyao, Farley, Kathleen A., Ding, WeiDong, Schiemer, James, Feng, Xidong, Chang, Jeanne S., Uccello, Daniel P., Young, Jennifer A., Garcia-Irrizary, Carmen N., Czabaniuk, Lara, Schuff, Brandon, Oliver, Robert, Montgomery, Justin, Hayward, Matthew M., Coe, Jotham, Chen, Jinshan, Niosi, Mark, Luthra, Suman, Shah, Jaymin C., El-Kattan, Ayman, Qiu, Xiayang, West, Graham M., Noe, Mark C., Shanmugasundaram, Veerabahu, Gilbert, Adam M., Brown, Matthew F., Calabrese, Matthew F.

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Snapshots and ensembles of BTK and cIAP1 protein degrader ternary complexes von Schiemer, James, Horst, Reto, Meng, Yilin, Montgomery, Justin I., Xu, Yingrong, Feng, Xidong, Borzilleri, Kris, Uccello, Daniel P., Leverett, Carolyn, Brown, Stephen, Che, Ye, Brown, Matthew F., Hayward, Matthew M., Gilbert, Adam M., Noe, Mark C., Calabrese, Matthew F.

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Discovery of Trifluoromethyl Glycol Carbamates as Potent and Selective Covalent Monoacylglycerol Lipase (MAGL) Inhibitors for Treatment of Neuroinflammation von McAllister, Laura A, Butler, Christopher R, Mente, Scot, O’Neil, Steven V, Fonseca, Kari R, Piro, Justin R, Cianfrogna, Julie A, Foley, Timothy L, Gilbert, Adam M, Harris, Anthony R, Helal, Christopher J, Johnson, Douglas S, Montgomery, Justin I, Nason, Deane M, Noell, Stephen, Pandit, Jayvardhan, Rogers, Bruce N, Samad, Tarek A, Shaffer, Christopher L, da Silva, Rafael G, Uccello, Daniel P, Webb, Damien, Brodney, Michael A

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Snapshots and ensembles of BTK and cIAP1 protein degrader ternary complexes von Schiemer, James, Horst, Reto, Meng, Yilin, Montgomery, Justin I., Xu, Yingrong, Feng, Xidong, Borzilleri, Kris, Uccello, Daniel P., Leverett, Carolyn, Brown, Stephen, Che, Ye, Brown, Matthew F., Hayward, Matthew M., Gilbert, Adam M., Noe, Mark C., Calabrese, Matthew F.

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Optimization of a Dicarboxylic Series for in Vivo Inhibition of Citrate Transport by the Solute Carrier 13 (SLC13) Family von Huard, Kim, Gosset, James R, Montgomery, Justin I, Gilbert, Adam, Hayward, Matthew M, Magee, Thomas V, Cabral, Shawn, Uccello, Daniel P, Bahnck, Kevin, Brown, Janice, Purkal, Julie, Gorgoglione, Matthew, Lanba, Adhiraj, Futatsugi, Kentaro, Herr, Michael, Genung, Nathan E, Aspnes, Gary, Polivkova, Jana, Garcia-Irizarry, Carmen N, Li, Qifang, Canterbury, Daniel, Niosi, Mark, Vera, Nicholas B, Li, Zhenhong, Khunte, Bhagyashree, Siderewicz, Jaclyn, Rolph, Timothy, Erion, Derek M

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Design and Synthesis of Clinical Candidate PF-06852231 (CVL-231): A Brain Penetrant, Selective, Positive Allosteric Modulator of the M4 Muscarinic Acetylcholine Receptor von Butler, Christopher R., Popiolek, Michael, McAllister, Laura A., LaChapelle, Erik A., Kramer, Melissa, Beck, Elizabeth M., Mente, Scot, Brodney, Michael A., Brown, Matthew, Gilbert, Adam, Helal, Chris, Ogilvie, Kevin, Starr, Jeremy, Uccello, Daniel, Grimwood, Sarah, Edgerton, Jeremy, Garst-Orozco, Jonathan, Kozak, Rouba, Lotarski, Susan, Rossi, Amie, Smith, Deborah, O’Connor, Rebecca, Lazzaro, John, Steppan, Claire, Steyn, Stefanus J.

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Design and Synthesis of Clinical Candidate PF-06852231 (CVL-231): A Brain Penetrant, Selective, Positive Allosteric Modulator of the M 4 Muscarinic Acetylcholine Receptor von Butler, Christopher R, Popiolek, Michael, McAllister, Laura A, LaChapelle, Erik A, Kramer, Melissa, Beck, Elizabeth M, Mente, Scot, Brodney, Michael A, Brown, Matthew, Gilbert, Adam, Helal, Chris, Ogilvie, Kevin, Starr, Jeremy, Uccello, Daniel, Grimwood, Sarah, Edgerton, Jeremy, Garst-Orozco, Jonathan, Kozak, Rouba, Lotarski, Susan, Rossi, Amie, Smith, Deborah, O'Connor, Rebecca, Lazzaro, John, Steppan, Claire, Steyn, Stefanus J

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Intramolecular Ring-Opening Decomposition of Aryl Azetidines von Bai, Guoyun, O’Connell, Thomas N, Brodney, Michael A, Butler, Christopher R, Czabaniuk, Lara C, Gilbert, Adam M, LaChapelle, Erik A, Li, Chao, McAllister, Laura A, Ogilvie, Kevin, Philippe, Laurence, Salomon-Ferrer, Romelia, Shapiro, Michael J, Starr, Jeremy T, Uccello, Daniel P, Withka, Jane M, Yan, Jiangli, Brown, Matthew F

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Intrinsic reactivity profile of electrophilic moieties to guide covalent drug design: N-α-acetyl- l -lysine as an amine nucleophile von Dahal, Upendra P., Gilbert, Adam M., Obach, R. Scott, Flanagan, Mark E., Chen, Jinshan M., Garcia-Irizarry, Carmen, Starr, Jeremy T., Schuff, Brandon, Uccello, Daniel P., Young, Jennifer A.

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Intrinsic reactivity profile of electrophilic moieties to guide covalent drug design: -α-acetyl--lysine as an amine nucleophile von Dahal, Upendra P, Gilbert, Adam M, Obach, R. Scott, Flanagan, Mark E, Chen, Jinshan M, Garcia-Irizarry, Carmen, Starr, Jeremy T, Schuff, Brandon, Uccello, Daniel P, Young, Jennifer A

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DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES von BRODNEY, Michael Aaron, GILBERT, Adam Matthew, ZHANG, Lei, MCALLISTER, Laura Ann, LACHAPELLE, Erik Alphie, BUTLER, Christopher Ryan, UCCELLO, Daniel Paul, BECK, Elizabeth Mary, BROWN, Matthew Frank

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DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES von ZHANG, LEI, BROWN, MATTHEW FRANK, UCCELLO, DANIEL PAUL, BECK, ELIZABETH MARY, LACHAPELLE, ERIK ALPHIE, BUTLER, CHRISTOPHER RYAN, GILBERT, ADAM MATTHEW, BRODNEY, MICHAEL AARON, MCALLISTER, LAURA ANN

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DIHYDRO-PYRROLO-PYRIDINE DERIVATIVES von BRODNEY, Michael Aaron, GILBERT, Adam Matthew, ZHANG, Lei, MCALLISTER, Laura Ann, LACHAPELLE, Erik Alphie, BUTLER, Christopher Ryan, UCCELLO, Daniel Paul, BECK, Elizabeth Mary, BROWN, Matthew Frank

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Dihydro-pyrrolo-pyridin-derivater von BRODNEY, Michael Aaron, GILBERT, Adam Matthew, ZHANG, Lei, MCALLISTER, Laura Ann, LACHAPELLE, Erik Alphie, BUTLER, Christopher Ryan, UCCELLO, Daniel Paul, BROWN, Matthew Frank, BECK, Elizabeth Mary

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