The discovery of carboline analogs as potent MAPKAP-K2 inhibitors von Wu, Jiang-Ping, Wang, Ji, Abeywardane, Asitha, Andersen, Denise, Emmanuel, Michel, Gautschi, Elda, Goldberg, Daniel R., Kashem, Mohammed A., Lukas, Susan, Mao, Wang, Martin, Leslie, Morwick, Tina, Moss, Neil, Pargellis, Christopher, Patel, Usha R., Patnaude, Lori, Peet, Gregory W., Skow, Donna, Snow, Roger J., Ward, Yancey, Werneburg, Brian, White, Andre

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Discovery and characterization of the N-phenyl- N′-naphthylurea class of p38 kinase inhibitors von Cirillo, Pier F., Hickey, Eugene R., Moss, Neil, Breitfelder, Steffen, Betageri, Raj, Fadra, Tazmeen, Gaenzler, Faith, Gilmore, Thomas, Goldberg, Daniel R., Kamhi, Victor, Kirrane, Thomas, Kroe, Rachel R., Madwed, Jeffrey, Moriak, Monica, Netherton, Matthew, Pargellis, Christopher A., Patel, Usha R., Qian, Kevin C., Sharma, Rajiv, Sun, Sanxing, Swinamer, Alan, Torcellini, Carol, Takahashi, Hidenori, Tsang, Michele, Xiong, Zhaoming

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Directed Lithiation of 3-[(tert-Butoxycarbonyl)amino]-2-methoxypyridines: Synthetic Route to Nevirapine and Its 4-Substituted Derivatives von Kelly, Terence A, Patel, Usha R

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Novel non-nucleoside inhibitors of HIV-1 reverse transcriptase. 1. Tricyclic pyridobenzo- and dipyridodiazepinones von Hargrave, Karl D, Proudfoot, John R, Grozinger, Karl G, Cullen, Ernest, Kapadia, Suresh R, Patel, Usha R, Fuchs, Victor U, Mauldin, Scott C, Vitous, Jana

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Antipsychotic activity of substituted .gamma.-carbolines von Abou-Gharbia, Magid, Patel, Usha R, Webb, Michael B, Moyer, John A, Andree, Terrance H, Muth, Eric A

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Nonpeptidic, Monocharged, Cell Permeable Ligands for the p56lck SH2 Domain von Proudfoot, John R, Betageri, Rajashehar, Cardozo, Mario, Gilmore, Thomas A, Glynn, Susan, Hickey, Eugene R, Jakes, Scott, Kabcenell, Alisa, Kirrane, Thomas M, Tibolla, Annette K, Lukas, Susan, Patel, Usha R, Sharma, Rajiv, Yazdanian, Mehran, Moss, Neil, Beaulieu, Pierre L, Cameron, Dale R, Ferland, Jean-Marie, Gauthier, Jean, Gillard, James, Gorys, Vida, Poirier, Martin, Rancourt, Jean, Wernic, Dominik, Llinas-Brunet, Montse

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Novel Non-nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Reverse Transcriptase. 4. 2-Substituted Dipyridodiazepinones as Potent Inhibitors of Both Wild-Type a... von Proudfoot, John R, Hargrave, Karl D, Kapadia, Suresh R, Patel, Usha R, Grozinger, Karl G, McNeil, Daniel W, Cullen, Ernest, Cardozo, Mario, Tong, Liang

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Synthesis of 7-Substituted Saccharins and 8-Substituted Oxicams, and a Novel Saccharin to Oxicam Transformation von Proudfoot, John R, Patel, Usha R, Dyatkin, Alexey B

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Novel Non-nucleoside Inhibitors of Human Immunodeficiency Virus Type 1 Reverse Transcriptase. 5. 4-Substituted and 2,4-Disubstituted Analogs of Nevirapine von Kelly, Terence A, Proudfoot, John R, McNeil, Daniel W, Patel, Usha R, David, Eva, Hargrave, Karl D, Grob, Peter M, Cardozo, Mario, Agarwal, Atul, Adams, Julian

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A novel Smiles rearrangement gives access to the A-ring pyridine isomers of the nevirapine ring system von Proudfoot, John R, Patel, Usha R, Campbell, Scot J

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The synthesis of 11-cyclopropyl-5,11-dihydro-4-(hydroxymethyl)-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepin-6-one, a putative metabolite of the HIV-1 reverse transcriptase inhibitor nev... von Patel, Usha R, Proudfoot, John R

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Novel Non-nucleoside Inhibitors of HIV-1 Reverse Transcriptase. 3. Dipyrido[2,3-b:2',3'-e]diazepinones von Proudfoot, John R, Patel, Usha R, Kapadia, Suresh R, Hargrave, Karl D

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Polycyclic aryl- and heteroarylpiperazinyl imides as 5-HT1A receptor ligands and potential anxiolytic agents: synthesis and structure-activity relationship studies von Abou-Gharbia, Magid, Patel, Usha R, Webb, Michael B, Moyer, John A, Andree, Terrance H, Muth, Eric A

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Psychotropic agents: synthesis and antipsychotic activity of substituted .beta.-carbolines von Abou-Gharbia, Magid, Patel, Usha R, Moyer, John A, Muth, Eric A

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Nonpeptidic, monocharged, cell permeable ligands for the p561ck SH2 domain von PROUDFOOT, John R, BETAGERI, Rajashehar, LUKAS, Susan, PATEL, Usha R, SHARMA, Rajiv, YAZDANIAN, Mehran, MOSS, Neil, BEAULIEU, Pierre L, CAMERON, Dale R, FERLAND, Jean-Marie, GAUTHIER, Jean, GILLARD, James, CARDOZO, Mario, GORYS, Vida, POIRIER, Martin, RANCOURT, Jean, WERNIC, Dominik, LLINAS-BRUNET, Montse, GILMORE, Thomas A, GLYNN, Susan, HICKEY, Eugene R, JAKES, Scott, KABCENELL, Alisa, KIRRANE, Thomas M, TIBOLLA, Annette K

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SPIROHETEROCYCLIC NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES von PATEL, USHA, R

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Bioavailability of Hydrochlorothiazide from Tablets and Suspensions von Patel, Rajni B., Patel, Usha R., Rogge, Mark C., Shah, Vinod P., Prasad, Vadlamani K., Selen, Arzu, Welling, Peter G.

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NOVEL NITRILES USEFUL AS REVERSIBLE INHIBITORS OF CYSTEINE PROTEASES von HICKEY, EUGENE R, SPERO, DENICE M, YOUNG, ERICK R. R, BEKKALI, YOUNES, THOMSON, DAVID S, PATEL, USHA R

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Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof von ZINDELL RENEE, LIU PINGRONG, RIETHER DORIS, HAMMACH ABDELHAKIM, TAKAHASHI HIDENORI, PATEL USHA R, WANG JI, RAZAVI HOSSEIN, LEE THOMAS WAI-HO, HARCKEN CHRISTIAN HANKE JUSTUS JOACHIM, KUZMICH DANIEL, PROUDFOOT JOHN ROBERT, BEKKALI YOUNES, THOMSON DAVID S, KIRRANE, JR. THOMAS MARTIN, BETAGERI RAJASHEKHAR, EMMANUEL MICHEL J

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NITRILE VERWENDBAR ALS REVERSIBLE CYSTEIN- PROTEASE INHIBITOREN von HICKEY, EUGENE R, SPERO, DENICE M, YOUNG, ERICK R. R, BEKKALI, YOUNES, THOMSON, DAVID S, PATEL, USHA R

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