C–H activation reactions as useful tools for medicinal chemists von Caro-Diaz, Eduardo J.E., Urbano, Mariangela, Buzard, Daniel J., Jones, Robert M.

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Microwave-assisted extraction of coumarin and related compounds from Melilotus officinalis (L.) Pallas as an alternative to Soxhlet and ultrasound-assisted extraction von Martino, Emanuela, Ramaiola, Ilaria, Urbano, Mariangela, Bracco, Francesco, Collina, Simona

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Discovery, design and synthesis of the first reported potent and selective sphingosine-1-phosphate 4 (S1P 4) receptor antagonists von Guerrero, Miguel, Urbano, Mariangela, Velaparthi, Subash, Zhao, Jian, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Discovery, design and synthesis of a selective S1P3 receptor allosteric agonist von Guerrero, Miguel, Poddutoori, Ramulu, Urbano, Mariangela, Peng, Xuemei, Spicer, Timothy P., Chase, Peter S., Hodder, Peter S., Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Discovery, design and synthesis of novel potent and selective sphingosine-1-phosphate 4 receptor (S1P4-R) agonists von Guerrero, Miguel, Urbano, Mariangela, Zhao, Jian, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Antagonists of the kappa opioid receptor von Urbano, Mariangela, Guerrero, Miguel, Rosen, Hugh, Roberts, Edward

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Modulators of the Sphingosine 1-phosphate receptor 1 von Urbano, Mariangela, Guerrero, Miguel, Rosen, Hugh, Roberts, Edward

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Discovery, synthesis and SAR analysis of novel selective small molecule S1P₄-R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chemot... von Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Identification of a potent and selective σ1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells von Rossi, Daniela, Pedrali, Alice, Urbano, Mariangela, Gaggeri, Raffaella, Serra, Massimo, Fernández, Leyden, Fernández, Michael, Caballero, Julio, Ronsisvalle, Simone, Prezzavento, Orazio, Schepmann, Dirk, Wuensch, Bernhard, Peviani, Marco, Curti, Daniela, Azzolina, Ornella, Collina, Simona

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Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140) von Guerrero, Miguel, Urbano, Mariangela, Kim, Eun-Kyong, Gamo, Ana M, Riley, Sean, Abgaryan, Lusine, Leaf, Nora, Van Orden, Lori Jean, Brown, Steven J, Xie, Jennifer Y, Porreca, Frank, Cameron, Michael D, Rosen, Hugh, Roberts, Edward

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SAR analysis of novel non-peptidic NPBWR1 (GPR7) antagonists von Guerrero, Miguel, Urbano, Mariangela, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Discovery, synthesis and SAR analysis of novel selective small molecule S1P 4-R agonists based on a (2 Z,5 Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one che... von Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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SAR analysis of innovative selective small molecule antagonists of sphingosine-1-phosphate 4 (S1P4) receptor von Urbano, Mariangela, Guerrero, Miguel, Zhao, Jian, Velaparthi, Subash, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Discovery, design and synthesis of a selective S1P(3) receptor allosteric agonist von Guerrero, Miguel, Poddutoori, Ramulu, Urbano, Mariangela, Peng, Xuemei, Spicer, Timothy P, Chase, Peter S, Hodder, Peter S, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Design, synthesis and SAR analysis of novel selective σ1 ligands (Part 2) von ROSSI, Daniela, URBANO, Mariangela, WUENSCH, Bernard, AZZOLINA, Ornella, COLLINA, Simona, PEDRALI, Alice, SERRA, Massimo, ZAMPIERI, Daniele, GRAZIA MAMOLO, Maria, LAGGNER, Christian, ZANETTE, Caterina, FLORIO, Chiara, SCHEPMANN, Dirk

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Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7) von Urbano, Mariangela, Guerrero, Miguel, Zhao, Jian, Velaparthi, Subash, Adrian Saldanha, S., Chase, Peter, Wang, Zhiwei, Civelli, Olivier, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Design, synthesis, and SAR analysis of novel selective σ1 ligands von Collina, Simona, Loddo, Guya, Urbano, Mariangela, Linati, Laura, Callegari, Athos, Ortuso, Francesco, Alcaro, Stefano, Laggner, Christian, Langer, Thierry, Prezzavento, Orazio, Ronsisvalle, Giuseppe, Azzolina, Ornella

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Discovery, synthesis and SAR analysis of novel selective small molecule S1P sub(4-R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolid i n-4-one... von Urbano, Mariangela, Guerrero, Miguel, Velaparthi, Subash, Crisp, Melissa, Chase, Peter, Hodder, Peter, Schaeffer, Marie-Therese, Brown, Steven, Rosen, Hugh, Roberts, Edward

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Substituted benzylaminoalkylindoles with preference for the σ2 binding site von GRAZIA MAMOLO, Maria, ZAMPIERI, Daniele, ZANETTE, Caterina, FLORIO, Chiara, COLLINA, Simona, URBANO, Mariangela, AZZOLINA, Ornella, VIO, Luciano

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Identification of a potent and selective Ief sub(1 receptor agonist potentiating NGF-induced neurite outgrowth in PC12 cells) von Rossi, Daniela, Pedrali, Alice, Urbano, Mariangela, Gaggeri, Raffaella, Serra, Massimo, Fernandez, Leyden, Fernandez, Michael, Caballero, Julio, Ronsisvalle, Simone, Prezzavento, Orazio, Schepmann, Dirk, Wuensch, Bernhard, Peviani, Marco, Curti, Daniela, Azzolina, Ornella, Collina, Simona

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