Myelosuppression and kinase selectivity of multikinase angiogenesis inhibitors von Kumar, R, Crouthamel, M-C, Rominger, D H, Gontarek, R R, Tummino, P J, Levin, R A, King, A G

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Genomic-sequence comparison of two unrelated isolates of the human gastric pathogen Helicobacter pylori von Alm, Richard A, Ling, Lo-See L, Moir, Donald T, King, Benjamin L, Brown, Eric D, Doig, Peter C, Smith, Douglas R, Noonan, Brian, Guild, Braydon C, deJonge, Boudewijn L, Carmel, Gilles, Tummino, Peter J, Caruso, Anthony, Uria-Nickelsen, Maria, Mills, Debra M, Ives, Cameron, Gibson, Rene, Merberg, David, Mills, Scott D, Jiang, Qin, Taylor, Diane E, Vovis, Gerald F, Trust, Trevor J

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Determination of the aggregation number of detergent micelles using steady-state fluorescence quenching von Tummino, P.J., Gafni, A.

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The in vitro Ejection of Zinc from Human Immunodeficiency Virus (HIV) Type 1 Nucleocapsid Protein by Disulfide Benzamides with Cellular Anti-HIV Activity von Tummino, Peter J., Scholten, Jeffrey D., Harvey, Patricia J., Holler, Tod P., Maloney, Lisa, Gogliotti, Rocco, Domagala, John, Hupe, Donald

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The human immunodeficiency virus type 1 (HIV-1) nucleocapsid protein zinc ejection activity of disulfide benzamides and benzisothiazolones: correlation with anti-HIV and virucidal... von TUMMINO, P. J, HARVEY, P. J, MCQUADE, T, DOMAGALA, J, GOGLIOTTI, R, SANCHEZ, J, SONG, Y, HUPE, D

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5,6-Dihydropyran-2-ones Possessing Various Sulfonyl Functionalities:  Potent Nonpeptidic Inhibitors of HIV Protease von Boyer, Frederick E, Vara Prasad, J. V. N, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hagen, Susan E, Markoski, Larry J, Tait, Bradley D, Lunney, Elizabeth A, Palovsky, Alexander, Ferguson, Donna, Graham, Neil, Holler, Tod, Hupe, Donald, Nouhan, Carolyn, Tummino, Peter J, Urumov, A, Zeikus, Eric, Zeikus, Greg, Gracheck, Stephen J, Sanders, James M, VanderRoest, Steven, Brodfuehrer, Joanne, Iyer, Krishna, Sinz, Michael, Gulnik, Sergei V, Erickson, John W

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Residence Time of Receptor−Ligand Complexes and Its Effect on Biological Function von Tummino, Peter J, Copeland, Robert A

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Synthesis of 5,6-Dihydro-4-hydroxy-2- pyrones as HIV-1 Protease Inhibitors:  The Profound Effect of Polarity on Antiviral Activity von Hagen, Susan E, Vara Prasad, J. V. N, Boyer, Frederick E, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hamilton, Harriet W, Markoski, Larry J, Steinbaugh, Bruce A, Tait, Bradley D, Lunney, Elizabeth A, Tummino, Peter J, Ferguson, Donna, Hupe, Donald, Nouhan, Carolyn, Gracheck, Stephen J, Saunders, James M, VanderRoest, Steven

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Competitive Inhibition of HIV-1 Protease by 4-Hydroxy-benzopyran-2-ones and by 4-Hydroxy-6-phenylpyran-2-ones von Tummino, P.J., Ferguson, D., Hupe, L., Hupe, D.

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Nonpeptidic HIV protease inhibitors possessing excellent antiviral activities and therapeutic indices. PD 178390 : A lead HIV protease inhibitor von VARA PRASAD, J. V. N, BOYER, F. E, HUMBLET, C, LUNNEY, E. A, PAVLOVSKY, A, RUBIN, J. R, FERGUSON, D, GRAHAM, N, HOLLER, T, HUPE, D, NOUHAN, C, TUMMINO, P. J, DOMAGALA, J. M, URUMOV, A, ZEIKUS, E, ZEIKUS, G, GRACHECK, S. J, SAUNDERS, J. M, VANDERROEST, S, BRODFUEHRER, J, IYER, K, SINZ, M, GULNIK, S. V, ELLSWORTH, E. L, ERICKSON, J. W, GAJDA, C, HAMILTON, H. W, HAGEN, S. E, MARKOSKI, L. J, STEINBAUGH, B. A, TAIT, B. D

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4-Hydroxy-5,6-dihydropyrones. 2. Potent Non-Peptide Inhibitors of HIV Protease von Tait, Bradley D, Hagen, Susan, Domagala, John, Ellsworth, Edmund L, Gajda, Christopher, Hamilton, Harriet W, Vara Prasad, J. V. N, Ferguson, Donna, Graham, Neil, Hupe, Donald, Nouhan, Carolyn, Tummino, Peter J, Humblet, Christine, Lunney, Elizabeth A, Pavlovsky, Alexander, Rubin, John, Gracheck, Stephen J, Baldwin, Eric T, Bhat, T. N, Erickson, John W, Gulnik, Sergei V, Liu, Beishan

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Adenine nucleotide translocase greatly increases the partition of trinitrophenyl-ATP into reduced Triton X-100 micelles von Tummino, P.J., Gafni, A.

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Novel Series of Achiral, Low Molecular Weight, and Potent HIV-1 Protease Inhibitors von Vara Prasad, J. V. N, Para, Kimberly S, Lunney, Elizabeth A, Ortwine, Daniel F, Dunbar, James B, Ferguson, Donna, Tummino, Peter J, Hupe, Donald, Tait, Bradley D

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Nonpeptidic HIV protease inhibitors: 6-alkyl-5,6-dihydropyran-2-ones possessing a novel and achiral 3-(2- t-butyl-5-methyl-4-sulfamate)phenylthio moiety von Vara Prasad, J.V.N, Markoski, Larry J, Boyer, Fred E, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hagen, Susan E, Tait, Bradley D, Lunney, Elizabeth A, Tummino, Peter J, Ferguson, Donna, Holler, Tod, Hupe, Donald, Nouhan, Carolyn, Gracheck, Stephen J, VanderRoest, Steven, Saunders, James, Iyer, K, Sinz, M

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A comparative study of succinate-supported respiration and ATP/ADP translocation in liver mitochondria from adult and old rats von Tummino, Peter J., Gafni, Ari

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Competitive Inhibition of HIV-1 Protease by Warfarin Derivatives von Tummino, P.J., Ferguson, D., Hupe, D.

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A Novel Nonpeptide HIV-1 Protease Inhibitor: Elucidation of the Binding Mode and Its Application in the Design of Related Analogs von Lunney, Elizabeth A, Hagen, Susan E, Domagala, John M, Humblet, Christine, Kosinski, Janet, Tait, Bradley D, Warmus, Joseph S, Wilson, Michael, Ferguson, Donna

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Substrate-Based Design of the First Class of Angiotensin-Converting Enzyme-Related Carboxypeptidase (ACE2) Inhibitors von Dales, Natalie A, Gould, Alexandra E, Brown, James A, Calderwood, Emily F, Guan, Bing, Minor, Charles A, Gavin, James M, Hales, Paul, Kaushik, Virendar K, Stewart, Michael, Tummino, Peter J, Vickers, Chad S, Ocain, Timothy D, Patane, Michael A

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Inhibitors of HIV protease: Unique non-peptide active site templates von Tait, Bradley D., Domagala, John, Ellsworth, Edmund L., Ferguson, Donna, Gajda, Christopher, Hupe, Donald, Lunney, Elizabeth A., Tummino, Peter J.

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A new class of anti-HIV-1 agents targeted toward the nucleocapsid protein NCp7: The 2,2′-dithiobisbenzamides von Domagala, John M., Bader, John P., Gogliotti, Rocco D., Sanchez, Joseph P., Stier, Michael A., Song, Yuntao, Vara Prasad, J.V.N., Tummino, Peter J., Scholten, Jeffrey, Harvey, Patricia, Holler, Tod, Gracheck, Steve, Hupe, Donald, Rice, William G., Schultz, Robert

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