Discovery of Potent Orally Active Thrombin Receptor (Protease Activated Receptor 1) Antagonists as Novel Antithrombotic Agents von Chackalamannil, Samuel, Xia, Yan, Greenlee, William J, Clasby, Martin, Doller, Darìo, Tsai, Hsingan, Asberom, Theodros, Czarniecki, Michael, Ahn, Ho-Sam, Boykow, George, Foster, Carolyn, Agans-Fantuzzi, Jacqueline, Bryant, Matthew, Lau, Janice, Chintala, Madhu

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Metabolism-Based Identification of a Potent Thrombin Receptor Antagonist von Clasby, Martin C, Chackalamannil, Samuel, Czarniecki, Michael, Doller, Dario, Eagen, Keith, Greenlee, William, Kao, Grace, Lin, Yan, Tsai, Hsingan, Xia, Yan, Ahn, Ho-Sam, Agans-Fantuzzi, Jacqueline, Boykow, George, Chintala, Madhu, Foster, Carolyn, Smith-Torhan, April, Alton, Kevin, Bryant, Matthew, Hsieh, Yunsheng, Lau, Janice, Palamanda, Jairam

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Himbacine derived thrombin receptor antagonists: Discovery of a new tricyclic core von Clasby, Martin C., Chackalamannil, Samuel, Czarniecki, Michael, Doller, Darío, Eagen, Keith, Greenlee, William J., Lin, Yan, Tagat, Jayaram R., Tsai, Hsingan, Xia, Yan, Ahn, Ho-Sam, Agans-Fantuzzi, Jacqueline, Boykow, George, Chintala, Madhu, Hsieh, Yunsheng, McPhail, Andrew T.

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Synthesis and Evaluation of Polycyclic Pyrazolo[3,4-d]pyrimidines as PDE1 and PDE5 cGMP Phosphodiesterase Inhibitors von Xia, Yan, Chackalamannil, Samuel, Czarniecki, Michael, Tsai, Hsingan, Vaccaro, Henry, Cleven, Renee, Cook, John, Fawzi, Ahmad, Watkins, Robert, Zhang, Hongtao

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Himbacine-Derived Thrombin Receptor Antagonists: C 7 -Spirocyclic Analogues of Vorapaxar von Chelliah, Mariappan V., Eagen, Keith, Guo, Zhuyan, Chackalamannil, Samuel, Xia, Yan, Tsai, Hsingan, Greenlee, William J., Ahn, Ho-Sam, Kurowski, Stan, Boykow, George, Hsieh, Yunsheng, Chintala, Madhu

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Himbacine-Derived Thrombin Receptor Antagonists: C7‑Spirocyclic Analogues of Vorapaxar von Chelliah, Mariappan V, Eagen, Keith, Guo, Zhuyan, Chackalamannil, Samuel, Xia, Yan, Tsai, Hsingan, Greenlee, William J, Ahn, Ho-Sam, Kurowski, Stan, Boykow, George, Hsieh, Yunsheng, Chintala, Madhu

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Himbacine derived thrombin receptor (PAR-1) antagonists: SAR of the pyridine ring von Xia, Yan, Chackalamannil, Samuel, Clasby, Martin, Doller, Darío, Eagen, Keith, Greenlee, William J., Tsai, Hsingan, Agans-Fantuzzi, Jacqueline, Ahn, Ho-Sam, Boykow, George C., Hsieh, Yunsheng, Lunn, Charles A., Chintala, Madhu

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Discovery and synthesis of a novel series of quinoline-based thrombin receptor (PAR-1) antagonists von Clasby, Martin C., Chackalamannil, Samuel, Czarniecki, Michael, Doller, Dario, Eagen, Keith, Greenlee, William J., Lin, Yan, Tsai, Hsingan, Xia, Yan, Ahn, Ho-Sam, Agans-Fantuzzi, Jacqueline, Boykow, George, Chintala, Madhu, Foster, Carolyn, Bryant, Matthew, Lau, Janice

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Himbacine derived thrombin receptor (PAR-1) antagonists: Structure–activity relationship of the lactone ring von Xia, Yan, Chackalamannil, Samuel, Chan, Tze-Ming, Czarniecki, Michael, Doller, Darío, Eagen, Keith, Greenlee, William J., Tsai, Hsingan, Wang, Yuguang, Ahn, Ho-Sam, Boykow, George C., McPhail, Andrew T.

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Carbocyclic Arabinofuranosyladenine (Cyclaradine): Efficacy against Genital Herpes in Guinea Pigs von Vince, Robert, Daluge, Susan, Lee, Heejoo, Shannon, William M., Arnett, Gussie, Schafer, Thomas W., Nagabhushan, Tattanahalli L., Reichert, Paul, Tsai, Hsingan

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Potent Tetracyclic Guanine Inhibitors of PDE1 and PDE5 Cyclic Guanosine Monophosphate Phosphodiesterases with Oral Antihypertensive Activity von Ahn, Ho-Sam, Bercovici, Ana, Boykow, George, Bronnenkant, Alan, Chackalamannil, Samuel, Chow, Jason, Cleven, Renee, Cook, John, Czarniecki, Michael, Domalski, Carol, Fawzi, Ahmad, Green, Michael, Gündes, Asli, Ho, Ginny, Laudicina, Malvina, Lindo, Neil, Ma, Ke, Manna, Mahua, McKittrick, Brian, Mirzai, Bita, Nechuta, Terry, Neustadt, Bernard, Puchalski, Chester, Pula, Kathryn, Silverman, Lisa, Smith, Elizabeth, Stamford, Andrew, Tedesco, Richard P, Tsai, Hsingan, Tulshian, Deen, Vaccaro, Henry, Watkins, Robert W, Weng, Xiaoyu, Witkowski, Joseph T, Xia, Yan, Zhang, Hongtao

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Highly potent and selective inhibitors of endothelin converting enzyme von Chackalamannil, Samuel, Chung, Shin, Stamford, Andrew W., McKittrick, Brian A., Wang, Yuguang, Tsai, Hsingan, Cleven, Reneé, Fawzi, Ahmad, Czarniecki, Michael

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Novel inhibitors of cholesteryl ester transfer protein von Chackalamannil, Samuel, Xia, Yan, Wang, Yuguang, Tsai, Hsingan, Czarniecki, Michael, Wang, Suke, Clemmons, Anthony, Ahn, Ho-Sam, Boykow, George

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Semisynthetic aminoglycoside antibacterials. Part 7. Synthesis of novel hexopyranosyl and hexofuranosyl derivatives of gentamine C1 and C1a von Daniels, Peter J. L., Luce, Charles E., Mallams, Alan K., Morton, James B., Saluja, Surinderjit S., Tsai, Hsingan, Weinstein, Jay, Wright, John J., Detre, George, Tanabe, Masato, Yasuda, Dennis M.

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