Lack of adipocyte purinergic P2Y₆ receptor greatly improves whole body glucose homeostasis von Jain, Shanu, Pydi, Sai P., Toti, Kiran S., Robaye, Bernard, Idzko, Marco, Gavrilova, Oksana, Wess, Jürgen, Jacobson, Kenneth A.

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South (S)- and North (N)-Methanocarba-7-Deazaadenosine Analogues as Inhibitors of Human Adenosine Kinase von Toti, Kiran S, Osborne, Danielle, Ciancetta, Antonella, Boison, Detlev, Jacobson, Kenneth A

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Polypharmacology of conformationally locked methanocarba nucleosides von Jacobson, Kenneth A., Tosh, Dilip K., Toti, Kiran S., Ciancetta, Antonella

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Novel alendronate-CGS21680 conjugate reduces bone resorption and induces new bone formation in post-menopausal osteoporosis and inflammatory osteolysis mouse models von Larrañaga-Vera, Ane, Toti, Kiran S, Flatow, James S, Haraczy, Alexandra J, Warnick, Eugene, Rao, Harsha, Gao, Zhan-Guo, Sussman, Sarah M, Mediero, Aranzazu, Leucht, Philipp, Jacobson, Kenneth A, Cronstein, Bruce N

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Structure-Activity Relationship and Neuroprotective Activity of 1,5-Dihydro-2 H -naphtho[1,2- b ][1,4]diazepine-2,4(3 H )-diones as P2X4 Receptor Antagonists von Toti, Kiran S, Verma, Rajkumar, McGonnigle, Michael J, Gamiotea Turro, Daylin, Wen, Zhiwei, Lewicki, Sarah A, Liang, Bruce T, Jacobson, Kenneth A

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Lack of adipocyte purinergic P2Y 6 receptor greatly improves whole body glucose homeostasis von Jain, Shanu, Pydi, Sai P, Toti, Kiran S, Robaye, Bernard, Idzko, Marco, Gavrilova, Oksana, Wess, Jürgen, Jacobson, Kenneth A

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Structure-activity relationships of pyrimidine nucleotides containing a 5′-α,β-methylene diphosphonate at the P2Y6 receptor von Oliva, Paola, Scortichini, Mirko, Dobelmann, Clemens, Jain, Shanu, Gopinatth, Varun, Toti, Kiran S., Phung, Ngan B., Junker, Anna, Jacobson, Kenneth A.

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Identification of a New Heterocyclic Scaffold for Inhibitors of the Polo-Box Domain of Polo-like Kinase 1 von Alverez, Celeste N, Park, Jung-Eun, Toti, Kiran S, Xia, Yangliu, Krausz, Kristopher W, Rai, Ganesha, Bang, Jeong K, Gonzalez, Frank J, Jacobson, Kenneth A, Lee, Kyung S

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Structure activity relationship of novel antiviral nucleosides against Enterovirus A71 von Tosh, Dilip K., Toti, Kiran S., Hurst, Brett L., Julander, Justin G., Jacobson, Kenneth A.

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Expanding the toolbox of metabolically stable lipid prodrug strategies von Toti, Kiran S, Pribut, Nicole, D'Erasmo, Michael, Dasari, Madhuri, Sharma, Savita K, Bartsch, Perry W, Burton, Samantha L, Gold, Hannah B, Bushnev, Anatoliy, Derdeyn, Cynthia A, Basson, Adriaan E, Liotta, Dennis C, Miller, Eric J

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Synthesis and Effect of Conformationally Locked Carbocyclic Guanine Nucleotides on Dynamin von Toti, Kiran S, Jimah, John R, Salmaso, Veronica, Hinshaw, Jenny E, Jacobson, Kenneth A

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Fluorescent A2A and A3 adenosine receptor antagonists as flow cytometry probes von Toti, Kiran S., Campbell, Ryan G., Lee, Hobin, Salmaso, Veronica, Suresh, R. Rama, Gao, Zhan-Guo, Jacobson, Kenneth A.

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Efficient synthesis of antifungal pyrimidines via palladium catalyzed Suzuki/Sonogashira cross-coupling reaction from Biginelli 3,4-dihydropyrimidin-2(1 H)-ones von Gholap, Atul R., Toti, Kiran S., Shirazi, Fazal, Deshpande, Mukund V., Srinivasan, Kumar V.

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Convergent synthesis of 2-thioether-substituted ()-methanocarba-adenosines as purine receptor agonists von Suresh, R. Rama, Poe, Russell B, Lin, Baorui, Lv, Kexin, Campbell, Ryan G, Gao, Zhan-Guo, Liston, Theodore E, Toti, Kiran S, Jacobson, Kenneth A

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Synthesis of an Apionucleoside Family and Discovery of a Prodrug with Anti-HIV Activity von Toti, Kiran S, Derudas, Marco, Pertusati, Fabrizio, Sinnaeve, Davy, Van den Broeck, Freya, Margamuljana, Lia, Martins, José C, Herdewijn, Piet, Balzarini, Jan, McGuigan, Christopher, Van Calenbergh, Serge

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Adenosine Kinase Expression Determines DNA Methylation in Cancer Cell Lines von Wahba, Amir E, Fedele, Denise, Gebril, Hoda, AlHarfoush, Enmar, Toti, Kiran S, Jacobson, Kenneth A, Boison, Detlev

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Synthesis and evaluation of antifungal properties of a series of the novel 2-amino-5-oxo-4-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile and its analogues von Gholap, Atul R., Toti, Kiran S., Shirazi, Fazal, Kumari, Ratna, Bhat, Manoj Kumar, Deshpande, Mukund V., Srinivasan, Kumar V.

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Allosteric Antagonism of the A2A Adenosine Receptor by a Series of Bitopic Ligands von Gao, Zhan-Guo, Toti, Kiran S., Campbell, Ryan, Suresh, R. Rama, Yang, Huijun, Jacobson, Kenneth A.

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Prevention and rescue of cardiac dysfunction by methanocarba adenosine monophosphonate derivatives von Shen, Jian-Bing, Toti, Kiran S., Chakraborty, Saibal, Kumar, T. Santhosh, Cronin, Chunxia, Liang, Bruce T., Jacobson, Kenneth A.

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Synthesis and evaluation of 5′-modified thymidines and 5-hydroxymethyl-2′-deoxyuridines as Mycobacterium tuberculosis thymidylate kinase inhibitors von Toti, Kiran S., Verbeke, Frederick, Risseeuw, Martijn D.P., Frecer, Vladimir, Munier-Lehmann, Hélène, Van Calenbergh, Serge

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