VEGF/VEGFR signalling as a target for inhibiting angiogenesis von Kiselyov, Alex, Balakin, Konstantin V, Tkachenko, Sergey E

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Virtual and biomolecular screening converge on a selective agonist for GPR30 von Oprea, Tudor I, Prossnitz, Eric R, Bologa, Cristian G, Revankar, Chetana M, Young, Susan M, Edwards, Bruce S, Arterburn, Jeffrey B, Kiselyov, Alexander S, Parker, Matthew A, Tkachenko, Sergey E, Savchuck, Nikolay P, Sklar, Larry A

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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6 Receptor (5-HT6R) A... von Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Kysil, Volodymyr M, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M

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(3-Phenylsulfonylcycloalkano[e and d]pyrazolo[1,5-a]pyrimidin-2-yl)amines: Potent and Selective Antagonists of the Serotonin 5-HT6 Receptor von Ivachtchenko, Alexandre V, Dmitriev, Dmitri E, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Kysil, Volodymyr M, Mitkin, Oleg D, Okun, Ilya M, Tkachenko, Sergey E, Vorobiev, Anton A

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Synthesis and SAR of 3-arylsulfonyl-pyrazolo[1,5-a]pyrimidines as potent serotonin 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya

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2-Substituted 5,6-dimethyl-3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines: new series of highly potent and specific serotonin 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V, Golovina, Elena S, Kadieva, Madina G, Koryakova, Angela G, Mitkin, Oleg D, Tkachenko, Sergey E, Kysil, Volodymyr M, Okun, Ilya

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Synthesis and biological evaluation of novel γ-carboline analogues of Dimebon as potent 5-HT6 receptor antagonists von IVACHTCHENKO, Alexandre V, FROLOV, Eugene B, MITKIN, Oleg D, KYSIL, Volodymyr M, KHVAT, Alexander V, OKUN, Ilya M, TLCACHENKO, Sergey E

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Synthesis and Structure−Activity Relationship of 4-Substituted 2-(2-Acetyloxyethyl)-8-(morpholine- 4-sulfonyl)pyrrolo[3,4-c]quinoline- 1,3-diones as Potent Caspase-3 Inhibitors von Kravchenko, Dmitri V, Kuzovkova, Yulia A, Kysil, Volodymyr M, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Balakin, Konstantin V, Ivachtchenko, Alexandre V

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Synthesis of cycloalkane-annelated 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidines and their evaluation as 5-HT6 receptor antagonists von IVACHTCHENKO, Alexandre V, DMITRIEV, Dmitri E, VOROBIOV, Anton A, GOLOVINA, Elena S, DUBROVSKAYA, Elena S, KADIEVA, Madina G, KORYAKOVA, Angela G, KYSIL, Volodymyr M, MITKIN, Oleg D, TKACHENKO, Sergey E, OKUN, Ilya M

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Synthesis and biological study of 3-(phenylsulfonyl)thieno[2,3-e][1,2,3]triazolo[1,5-a]pyrimidines as potent and selective serotonin 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Koryakova, Angela G., Kovalenko, Sergiy M., Mitkin, Oleg D., Okun, Ilya M., Ravnyeyko, Irina M., Tkachenko, Sergey E., Zaremba, Oleg V.

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Pyrrolo[3,4-c]quinoline-1,3-diones as potent caspase-3 inhibitors. Synthesis and SAR of 2-substituted 4-methyl-8-(morpholine-4-sulfonyl)-pyrrolo[3,4- c]quinoline-1,3-diones von Kravchenko, Dmitri V., Kysil, Volodymyr M., Tkachenko, Sergey E., Maliarchouk, Sergey, Okun, Ilya M., Ivachtchenko, Alexandre V.

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1,3-Dioxo-4-methyl-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines as potent caspase-3 inhibitors von Kravchenko, Dmitri V, Kysil, Vladimir V, Ilyn, Alexey P, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Ivachtchenko, Alexandre V

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Exploring the chemogenomic knowledge space with annotated chemical libraries von Savchuk, Nikolay P, Balakin, Konstantin V, Tkachenko, Sergey E

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8-Sulfonyl-substituted tetrahydro-1H-pyrido[4,3-b]indoles as 5-HT6 receptor antagonists von Ivachtchenko, Alexandre V, Mitkin, Oleg D, Tkachenko, Sergey E, Okun, Ilya M, Kysil, Volodymyr M

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One-Step Assembly of Carbamoyl-Substituted Heteroannelated [1,4]Thiazepines von Ilyn, Alexey P, Loseva, Marina V, Vvedensky, Vladimir Y, Putsykina, Elena B, Tkachenko, Sergey E, Kravchenko, Dmitri V, Khvat, Alexandr V, Krasavin, Mikhail Y, Ivachtchenko, Alexandre V

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Small-molecule modulators of Hh and Wnt signaling pathways von Kiselyov, Alex S, Tkachenko, Sergey E, Balakin, Konstantin V, Ivachtchenko, Alexandre V

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Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5- a ]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT 6 Receptor (5-HT 6... von Ivachtchenko, Alexandre V., Golovina, Elena S., Kadieva, Madina G., Kysil, Volodymyr M., Mitkin, Oleg D., Tkachenko, Sergey E., Okun, Ilya M.

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Property-Based Design of GPCR-Targeted Library von Balakin, Konstantin V, Tkachenko, Sergey E, Lang, Stanley A, Okun, Ilya, Ivashchenko, Andrey A, Savchuk, Nikolay P

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Synthesis and caspase-3 inhibitory activity of 8-sulfonyl-1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4-c]quinolines von Kravchenko, Dmitri V, Kysil, Volodymyr M, Tkachenko, Sergey E, Maliarchouk, Sergey, Okun, Ilya M, Ivachtchenko, Alexandre V

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Structure-Based versus Property-Based Approaches in the Design of G-Protein-Coupled Receptor-Targeted Libraries von Balakin, Konstantin V, Lang, Stanley A, Skorenko, Andrey V, Tkachenko, Sergey E, Ivashchenko, Andrey A, Savchuk, Nikolay P

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