Preliminary Structure–Activity Relationships and Biological Evaluation of Novel Antitubercular Indolecarboxamide Derivatives Against Drug-Susceptible and Drug-Resistant Mycobacteri... von Onajole, Oluseye K, Pieroni, Marco, Tipparaju, Suresh K, Lun, Shichun, Stec, Jozef, Chen, Gang, Gunosewoyo, Hendra, Guo, Haidan, Ammerman, Nicole C, Bishai, William R, Kozikowski, Alan P

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Indoleamides are active against drug-resistant Mycobacterium tuberculosis von Lun, Shichun, Guo, Haidan, Onajole, Oluseye K., Pieroni, Marco, Gunosewoyo, Hendra, Chen, Gang, Tipparaju, Suresh K., Ammerman, Nicole C., Kozikowski, Alan P., Bishai, William R.

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Targeting EphA2 in Bladder Cancer Using a Novel Antibody-Directed Nanotherapeutic von Kamoun, Walid, Swindell, Elden, Pien, Christine, Luus, Lia, Cain, Jason, Pham, Minh, Kandela, Irawati, Huang, Zhaohua Richard, Tipparaju, Suresh K., Koshkaryev, Alexander, Askoxylakis, Vasileios, Kirpotin, Dmitri B., Bloom, Troy, Mino-Kenudson, Mari, Marks, James D., Zalutskaya, Alena, Bshara, Wiam, Morrison, Carl, Drummond, Daryl C.

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Identification and Development of Novel Inhibitors of Toxoplasma gondii Enoyl Reductase von Tipparaju, Suresh K, Muench, Stephen P, Mui, Ernest J, Ruzheinikov, Sergey N, Lu, Jeffrey Z, Hutson, Samuel L, Kirisits, Michael J, Prigge, Sean T, Roberts, Craig W, Henriquez, Fiona L, Kozikowski, Alan P, Rice, David W, McLeod, Rima L

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Pyrido[1,2-a]benzimidazole-Based Agents Active Against Tuberculosis (TB), Multidrug-Resistant (MDR) TB and Extensively Drug-Resistant (XDR) TB von Pieroni, Marco, Tipparaju, Suresh K., Lun, Shichun, Song, Yang, Sturm, A. Willem, Bishai, William R., Kozikowski, Alan P.

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Indoleamides are active against drug-resistant Mycobacterium tuberculosis von Lun, Shichun, Guo, Haidan, Onajole, Oluseye K., Pieroni, Marco, Gunosewoyo, Hendra, Chen, Gang, Tipparaju, Suresh K., Ammerman, Nicole C., Kozikowski, Alan P., Bishai, William R.

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In Pursuit of Natural Product Leads: Synthesis and Biological Evaluation of 2-[3-hydroxy-2-[(3-hydroxypyridine-2-carbonyl)amino]phenyl]benzoxazole-4-carboxylic acid (A-33853) and I... von Tipparaju, Suresh K, Joyasawal, Sipak, Pieroni, Marco, Kaiser, Marcel, Brun, Reto, Kozikowski, Alan P

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Design and Synthesis of Aryl Ether Inhibitors of the Bacillus Anthracis Enoyl-ACP Reductase von Tipparaju, Suresh K., Mulhearn, Debbie C., Klein, Gary M., Chen, Yufeng, Tapadar, Subhasish, Bishop, Molly H., Yang, Shuo, Chen, Juan, Ghassemi, Mahmood, Santarsiero, Bernard D., Cook, James L., Johlfs, Mary, Mesecar, Andrew D., Johnson, Michael E., Kozikowski, Alan P.

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Structural analogs of huperzine A improve survival in guinea pigs exposed to soman von Gunosewoyo, Hendra, Tipparaju, Suresh K., Pieroni, Marco, Wang, Ying, Doctor, Bhupendra P., Nambiar, Madhusoodana P., Kozikowski, Alan P.

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Design and synthesis of 2-pyridones as novel inhibitors of the Bacillus anthracis enoyl-ACP reductase von Tipparaju, Suresh K., Joyasawal, Sipak, Forrester, Sara, Mulhearn, Debbie C., Pegan, Scott, Johnson, Michael E., Mesecar, Andrew D., Kozikowski, Alan P.

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Natural product leads for drug discovery: Isolation, synthesis and biological evaluation of 6-cyano-5-methoxyindolo[2,3- a]carbazole based ligands as antibacterial agents von Guo, Songpo, Tipparaju, Suresh K., Pegan, Scott D., Wan, Baojie, Mo, Shunyan, Orjala, Jimmy, Mesecar, Andrew D., Franzblau, Scott G., Kozikowski, Alan P.

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Technology Transfer and Process Development of Danicopan to Enable Process Validation von Liu, Yangmu Chloe, Tipparaju, Suresh K., Tracey, Michael R., Carr, Robert, Damarancha, Anil, Hashimoto, Akihiro, Hubbs, Stephen, Keyes, Chad, Lucas, John, Nandialath, Vidya, Stevens, Mark, Thottakara, Mareena

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Development of a Scalable Process for the Synthesis of Cyclopropyl-Methyl-Proline with Complex Stereochemistry: A Key Building Block of Factor D Inhibitors von Hashimoto, Akihiro, Ferretti, Antonio C., Tipparaju, Suresh K., Burt, Justin L., Soman, Ashish, Phadke, Avinash, Chandran, Prabu, Lahoti, Anand M., Bilidegalu N, Devaraju, Mani, Anbazhagan, Datta, Swarup, Rai, Sankappa, Huddar, Sameerana, Kumara, Prasanna, Raju, Tirumani, AN, Guruprasad, Ganapathy, Suman, Chukka, Tanish

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Antitumour activity and tolerability of an EphA2-targeted nanotherapeutic in multiple mouse models von Kamoun, Walid S., Kirpotin, Dmitri B., Huang, Zhaohua Richard, Tipparaju, Suresh K., Noble, Charles O., Hayes, Mark E., Luus, Lia, Koshkaryev, Alexander, Kim, Jaeyeon, Olivier, Ken, Kornaga, Tad, Oyama, Shinji, Askoxylakis, Vasileios, Pien, Christine, Kuesters, Geoffrey, Dumont, Nancy, Lugovskoy, Alexey A., Schihl, Sarah A., Wilton, John H., Geddie, Melissa L., Suchy, James, Grabow, Stephanie, Kohli, Neeraj, Reynolds, C. Patrick, Blaydes, Rachel, Zhou, Yu, Sawyer, Andrew J., Marks, James D., Drummond, Daryl C.

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Abstract 4711: Immunomodulatory effects of an EphA2-targeted docetaxel antibody-directed nanotherapeutic and synergistic combination with PD-1 inhibitor von Sawyer, Andrew J., Dugast, Anne-Sophie, Luus, Lia, Huang, Zhaohua Richard, Tipparaju, Suresh K., Kirpotin, Dmitri B., Drummond, Daryl C., Kamoun, Walid S.

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Abstract 3096: Mechanisms of synergy of carboplatin and an EphA2-targeted docetaxel antibody-directed nanotherapeutic von Kamoun, Walid S., Sawyer, Andrew J., Pien, Christine, Koshkaryev, Alexander, Luus, Lia, Merrigan, Samantha, Sun, Gang, Kozin, Sergey, Huang, Zhaohua Richard, Tipparaju, Suresh K., Kirpotin, Dmitri B., Xu, Hannah, Askoxylakis, Vasileios, Reynolds, Patrick C., Drummond, Daryl C.

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INHIBITING ATAXIA TELANGIECTASIA AND RAD3-RELATED PROTEIN (ATR) von Geng, Bolin, Kirpotin, Dmitri B, Koshkaryev, Alexander, Drummond, Daryl C, Alkan, Ozan, Tipparaju, Suresh K

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OXAZOLIDINONE COMPOUNDS, LIPOSOME COMPOSITIONS COMPRISING OXAZOLIDINONE COMPOUNDS AND METHOD OF USE THEREOF von Noble, Charles O, Koshkaryev, Alexander, Kirpotin, Dmitri B, Drummond, Daryl C, Tipparaju, Suresh K

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OXAZOLIDINONE COMPOUNDS, LIPOSOME COMPOSITIONS COMPRISING OXAZOLIDINONE COMPOUNDS AND METHOD OF USE THEREOF von Noble, Charles O, Koshkaryev, Alexander, Kirpotin, Dmitri B, Drummond, Daryl C, Tipparaju, Suresh K

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INHIBITING ATAXIA TELANGIECTASIA AND RAD3-RELATED PROTEIN (ATR) von ALKAN, Ozan, KIRPOTIN, Dmitri B, DRUMMOND, Daryl C, GENG, Bolin, KOSHKARYEV, Alexander, TIPPARAJU, Suresh K

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