KAHA Ligations That Form Aspartyl Aldehyde Residues as Synthetic Handles for Protein Modification and Purification von Murar, Claudia E, Thuaud, Frédéric, Bode, Jeffrey W

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Incorporation of Acid-Labile Masking Groups for the Traceless Synthesis of C‑Terminal Peptide α‑Ketoacids von Thuaud, Frédéric, Rohrbacher, Florian, Zwicky, André, Bode, Jeffrey W

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Novel Flavaglines Displaying Improved Cytotoxicity von Thuaud, Frédéric, Ribeiro, Nigel, Gaiddon, Christian, Cresteil, Thierry, Désaubry, Laurent

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Recent advances in the biology and chemistry of the flavaglines von Ribeiro, Nigel, Thuaud, Frédéric, Nebigil, Canan, Désaubry, Laurent

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Photoprotected Peptide α-Ketoacids and Hydroxylamines for Iterative and One-Pot KAHA Ligations: Synthesis of NEDD8 von Thuaud, Frédéric, Rohrbacher, Florian, Zwicky, André, Bode, Jeffrey W.

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Chemical Synthesis of the 20kDa Heme Protein Nitrophorin4 by [alpha]-Ketoacid-Hydroxylamine (KAHA) Ligation von He, Chunmao, Kulkarni, Sameer S, Thuaud, Frédéric, Bode, Jeffrey W

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Benzofuran derivatives as anticancer inhibitors of mTOR signaling von Salomé, Christophe, Ribeiro, Nigel, Chavagnan, Thierry, Thuaud, Frédéric, Serova, Maria, de Gramont, Armand, Faivre, Sandrine, Raymond, Eric, Désaubry, Laurent

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Benzofuran derivatives as a novel class of inhibitors of mTOR signaling von Salomé, Christophe, Narbonne, Vanessa, Ribeiro, Nigel, Thuaud, Frédéric, Serova, Maria, de Gramont, Armand, Faivre, Sandrine, Raymond, Eric, Désaubry, Laurent

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eIF4F is a nexus of resistance to anti-BRAF and anti-MEK cancer therapies von Boussemart, Lise, Malka-Mahieu, Hélène, Girault, Isabelle, Allard, Delphine, Hemmingsson, Oskar, Tomasic, Gorana, Thomas, Marina, Basmadjian, Christine, Ribeiro, Nigel, Thuaud, Frédéric, Mateus, Christina, Routier, Emilie, Kamsu-Kom, Nyam, Agoussi, Sandrine, Eggermont, Alexander M., Désaubry, Laurent, Robert, Caroline, Vagner, Stéphan

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RE12 derivatives displaying Vaccinia H1-related phosphatase (VHR) inhibition in the presence of detergent and their anti-proliferative activity against HeLa cells von Thuaud, Frédéric, Kojima, Shuntaro, Hirai, Go, Oonuma, Kana, Tsuchiya, Ayako, Uchida, Takako, Tsuchimoto, Teruhisa, Sodeoka, Mikiko

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Flavaglines as Potent Anticancer and Cytoprotective Agents von Ribeiro, Nigel, Thuaud, Frédéric, Bernard, Yohann, Gaiddon, Christian, Cresteil, Thierry, Hild, Audrey, Hirsch, Etienne C, Michel, Patrick Pierre, Nebigil, Canan G, Désaubry, Laurent

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Assessment of flavaglines as potential chikungunya virus entry inhibitors von Wintachai, Phitchayapak, Thuaud, Frédéric, Basmadjian, Christine, Roytrakul, Sittiruk, Ubol, Sukathida, Désaubry, Laurent, Smith, Duncan R.

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Prohibitin Ligands in Cell Death and Survival: Mode of Action and Therapeutic Potential von Thuaud, Frédéric, Ribeiro, Nigel, Nebigil, Canan G., Désaubry, Laurent

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Synthetic Analogue of Rocaglaol Displays a Potent and Selective Cytotoxicity in Cancer Cells: Involvement of Apoptosis Inducing Factor and Caspase-12 von Thuaud, Frédéric, Bernard, Yohann, Türkeri, Gülen, Dirr, Ronan, Aubert, Geneviève, Cresteil, Thierry, Baguet, Aurélie, Tomasetto, Catherine, Svitkin, Yuri, Sonenberg, Nahum, Nebigil, Canan G, Désaubry, Laurent

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N-[3a-(4-Bromo-phen-yl)-8b-hy-droxy-6,8-dimeth-oxy-3-phenyl-2,3,3a,8b-tetra-hydro-1H-cyclo-penta-[b]benzofuran-1-yl]formamide monohydrate von Aubert, Emmanuel, Thuaud, Frédéric, Ribeiro, Nigel, Désaubry, Laurent, Espinosa, Enrique

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Synthesis of All Stereoisomers of Monomeric Spectomycin A1/A2 and Evaluation of Their Protein SUMOylation‐Inhibitory Activity von Nomura, Yusaku, Thuaud, Frédéric, Sekine, Daisuke, Ito, Akihiro, Maeda, Satoko, Koshino, Hiroyuki, Hashizume, Daisuke, Muranaka, Atsuya, Cruchter, Thomas, Uchiyama, Masanobu, Ichikawa, Satoshi, Matsuda, Akira, Yoshida, Minoru, Hirai, Go, Sodeoka, Mikiko

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Flavaglines alleviate doxorubicin cardiotoxicity: implication of Hsp27 von Bernard, Yohann, Ribeiro, Nigel, Thuaud, Frédéric, Türkeri, Gülen, Dirr, Ronan, Boulberdaa, Mounia, Nebigil, Canan G, Désaubry, Laurent

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Chemical Synthesis of the 20 kDa Heme Protein Nitrophorin 4 by α-Ketoacid-Hydroxylamine (KAHA) Ligation von He, Chunmao, Kulkarni, Sameer S., Thuaud, Frédéric, Bode, Jeffrey W.

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Assessment of flavaglines as potential chikungunya virus entry inhibitors von Wintachai, Phitchayapak, Thuaud, Frédéric, Basmadjian, Christine, Roytrakul, Sittiruk, Ubol, Sukathida, Désaubry, Laurent, Smith, Duncan R.

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Selective anticancer effects of a synthetic flavagline on human Oct4-expressing cancer stem-like cells via a p38 MAPK-dependent caspase-3-dependent pathway von Emhemmed, Fathi, Ali Azouaou, Sarah, Thuaud, Frédéric, Schini-Kerth, Valérie, Désaubry, Laurent, Muller, Christian D., Fuhrmann, Guy

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