Identification of candidate substrates for poly(ADP‐ribose) polymerase‐2 (PARP2) in the absence of DNA damage using high‐density protein microarrays von Troiani, Sonia, Lupi, Rosita, Perego, Rita, Re Depaolini, Stefania, Thieffine, Sandrine, Bosotti, Roberta, Rusconi, Luisa

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Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1) von Huynh, Tram, Chen, Zhong, Pang, Suhong, Geng, Jieping, Bandiera, Tiziano, Bindi, Simona, Vianello, Paola, Roletto, Fulvia, Thieffine, Sandrine, Galvani, Arturo, Vaccaro, Wayne, Poss, Michael A., Trainor, George L., Lorenzi, Matthew V., Gottardis, Marco, Jayaraman, Lata, Purandare, Ashok V.

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Cell Division Cycle 7 Kinase Inhibitors: 1H-Pyrrolo[2,3-b]pyridines, Synthesis and Structure−Activity Relationships von Ermoli, Antonella, Bargiotti, Alberto, Brasca, Maria Gabriella, Ciavolella, Antonella, Colombo, Nicoletta, Fachin, Gabriele, Isacchi, Antonella, Menichincheri, Maria, Molinari, Antonio, Montagnoli, Alessia, Pillan, Antonio, Rainoldi, Sonia, Sirtori, Federico Riccardi, Sola, Francesco, Thieffine, Sandrine, Tibolla, Marcellino, Valsasina, Barbara, Volpi, Daniele, Santocanale, Corrado, Vanotti, Ermes

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Natural and synthetic 2-oxoglutarate derivatives are substrates for oncogenic variants of human isocitrate dehydrogenase 1 and 2 von Liu, Xiao, Reinbold, Raphael, Liu, Shuang, Herold, Ryan A., Rabe, Patrick, Duclos, Stéphanie, Yadav, Rahul B., Abboud, Martine I., Thieffine, Sandrine, Armstrong, Fraser A., Brewitz, Lennart, Schofield, Christopher J.

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Structural basis for CARM1 inhibition by indole and pyrazole inhibitors von Sack, John S, Thieffine, Sandrine, Bandiera, Tiziano, Fasolini, Marina, Duke, Gerald J, Jayaraman, Lata, Kish, Kevin F, Klei, Herbert E, Purandare, Ashok V, Rosettani, Pamela, Troiani, Sonia, Xie, Dianlin, Bertrand, Jay A

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Insights into PARP Inhibitors’ Selectivity Using Fluorescence Polarization and Surface Plasmon Resonance Binding Assays von Papeo, Gianluca, Avanzi, Nilla, Bettoni, Serena, Leone, Antonella, Paolucci, Mauro, Perego, Rita, Quartieri, Francesca, Riccardi-Sirtori, Federico, Thieffine, Sandrine, Montagnoli, Alessia, Lupi, Rosita

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Development of Biochemical Assays for the Identification of eIF4E-Specific Inhibitors von Visco, Carlo, Perrera, Claudia, Thieffine, Sandrine, Sirtori, Federico Riccardi, D’Alessio, Roberto, Magnaghi, Paola

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Abstract 691: In vitro and in vivo characterization of selective orally available Parp-1 inhibitors with demonstrated antitumor efficacy in BRCA negative cancer models von Papeo, Gianluca, Rainoldi, Sonia, Gianellini, Laura, Ciavolella, Antonella, Leone, Antonella, Lupi, Rosita, Sola, Francesco, Caprera, Francesco, Paolucci, Mauro, Thieffine, Sandrine, Perego, Rita, Albanese, Clara, Casale, Elena, Forte, Barbara, Guanci, Marco, Orsini, Paolo, Posteri, Helena, Scolaro, Alessandra, Riccardi-Sirtori, Federico, Zuccotto, Fabio, Donati, Daniele, Moll, Jurgen, Montagnoli, Alessia

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Cell Division Cycle 7 Kinase Inhibitors: 1 H -Pyrrolo[2,3- b ]pyridines, Synthesis and Structure−Activity Relationships von Ermoli, Antonella, Bargiotti, Alberto, Brasca, Maria Gabriella, Ciavolella, Antonella, Colombo, Nicoletta, Fachin, Gabriele, Isacchi, Antonella, Menichincheri, Maria, Molinari, Antonio, Montagnoli, Alessia, Pillan, Antonio, Rainoldi, Sonia, Sirtori, Federico Riccardi, Sola, Francesco, Thieffine, Sandrine, Tibolla, Marcellino, Valsasina, Barbara, Volpi, Daniele, Santocanale, Corrado, Vanotti, Ermes

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Single Protocol for the Selective Isotopic and Chemical Labeling of Protein Kinases in Insect Cells for NMR and Crystallographic Studies von Cristiani, Cinzia, Thieffine, Sandrine, Messali, Silvia, Rusconi, Luisa, Schnuchel, Arndt, Kalisz, Henryk

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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF von VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE

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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF von VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE

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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF von VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, KALISZ, HENRYK, PEREGO, RITA, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE

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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF von VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE

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formas truncadas de dbf4 humana, complexos com seus pares de interação e métodos para identificação de seus inibidores von BARBARA VALSASINA, CINZIA CRISTIANI, HENRYK KALISZ, STEFAN KNAPP, MARIA BEATRICE SACCARDO, SANDRINE THIEFFINE, RITA PEREGO

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TRUNCATED FORMS OF HUMAN DBF4, COMPLEXES WITH THEIR INTERACTING PARTNERS AND METHODS FOR IDENTIFICATION OF INHIBITORS THEREOF von VALSASINA, BARBARA, THIEFFINE, SANDRINE, CRISTIANI, CINZIA, PEREGO, RITA, KALISZ, HENRYK, KNAPP, STEFAN, SACCARDO, MARIA BEATRICE

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