Discovery of a Tetrahydropyrimidin-2(1H)-one Derivative (TAK-442) as a Potent, Selective, and Orally Active Factor Xa Inhibitor von Fujimoto, Takuya, Imaeda, Yasuhiro, Konishi, Noriko, Hiroe, Katsuhiko, Kawamura, Masaki, Textor, Garret P, Aertgeerts, Kathleen, Kubo, Keiji

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2-{3-[4-(Alkylsulfinyl)phenyl]-1-benzofuran-5-yl}-5-methyl-1,3,4-oxadiazole Derivatives as Novel Inhibitors of Glycogen Synthase Kinase-3β with Good Brain Permeability von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Iwashita, Hiroki, Uno, Yumiko, Onishi, Tomohiro, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D, Dougan, Douglas R, Textor, Garret P, Snell, Gyorgy P, Takizawa, Masayuki, Itoh, Fumio, Kori, Masakuni

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2-{3-[4-(Alkylsulfinyl)phenyl]-1-benzofuran-5-yl}-5-methyl-1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3beta with good brain permeability von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Iwashita, Hiroki, Uno, Yumiko, Onishi, Tomohiro, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D, Dougan, Douglas R, Textor, Garret P, Snell, Gyorgy P, Takizawa, Masayuki, Itoh, Fumio, Kori, Masakuni

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Design, synthesis and structure–activity relationships of 1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3β von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Hayase, Yoji, Kobayashi, Hiromi, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D., Dougan, Douglas R., Textor, Garret S., Snell, Gyorgy P., Itoh, Fumio

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Design, synthesis and structure-activity relationships of 1,3,4-oxadiazole derivatives as novel inhibitors of glycogen synthase kinase-3beta von Saitoh, Morihisa, Kunitomo, Jun, Kimura, Eiji, Hayase, Yoji, Kobayashi, Hiromi, Uchiyama, Noriko, Kawamoto, Tomohiro, Tanaka, Toshimasa, Mol, Clifford D, Dougan, Douglas R, Textor, Garret S, Snell, Gyorgy P, Itoh, Fumio

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