Organic Photoredox-Catalyzed S‑Trifluoromethylation of Aromatic and Heteroaromatic Thiols von Bhattacharyya, Aditya, Vadde, Veeresh, Sarmah, Manash Pratim, Muthukumar, M, Mathur, Arvind, Tester, Richland

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Amide-based inhibitors of p38α MAP kinase. Part 1: Discovery of novel N-pyridyl amide lead molecules von Luedtke, Gregory R., Schinzel, Kurt, Tan, Xuefei, Tester, Richland W., Nashashibi, Imad, Xu, Yong-jin, Dugar, Sundeep, Levy, Daniel E., Jung, Joon

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Design and synthesis of piperazine-indole p38α MAP kinase inhibitors with improved pharmacokinetic profiles von Tan, Xuefei, Tester, Richland W., Luedtke, Gregory R., Chakravarty, Sarvajit, Mavunkel, Babu J., Perumattam, John J., Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E., Dugar, Sundeep

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Inhibition of Btk with CC-292 provides early pharmacodynamic assessment of activity in mice and humans von Evans, Erica K, Tester, Richland, Aslanian, Sharon, Karp, Russell, Sheets, Michael, Labenski, Matthew T, Witowski, Steven R, Lounsbury, Heather, Chaturvedi, Prasoon, Mazdiyasni, Hormoz, Zhu, Zhendong, Nacht, Mariana, Freed, Martin I, Petter, Russell C, Dubrovskiy, Alex, Singh, Juswinder, Westlin, William F

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Synthesis of diversely substituted quinazoline-2,4(1 H ,3 H )-diones by cyclization of tert -butyl (2-cyanoaryl)carbamates von Kovela, Satish, Karad, Somnath, Tatipudi, V V Ganesh, Arumugam, Karthikeyan, Somwanshi, Atul Vijay, Muthukumar, M, Mathur, Arvind, Tester, Richland

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Discovery and Synthesis of Heterobifunctional Degraders of Rearranged during Transfection (RET) Kinase von Qiao, Jennifer X., Williams, David, Gill, Patrice, Li, Ling, Norris, Derek, Tokarski, John S., Wong, Jessica, Qi, Huilin, Hafeji, Yamnah, Downes, Daniel P., Degnen, Bill, Wang, Ying-Kai, Locke, Gregory, Fang, Hua, Yu, Fei, Xu, Songmei, Naglich, Joseph, Zhang, Jun, Nanjappa, Purushothama, Dai, Chao, Chourb, Lisa, Napoline, Jonathan, Tester, Richland, Jorge, Christine, Li, Yi-Xin, Mathur, Arvind, Barbieri, Christopher, Soars, Matthew G., Venkatanarayan, Avinashnarayan, Lees, Emma, Borzilleri, Robert M., Gavai, Ashvinikumar V., Wichroski, Michael, Dhar, T. G. Murali

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In vitro and in vivo characterization of irreversible mutant-selective EGFR inhibitors that are wild-type sparing von Tjin Tham Sjin, Robert, Lee, Kwangho, Walter, Annette O, Dubrovskiy, Aleksandr, Sheets, Michael, Martin, Thia St, Labenski, Matthew T, Zhu, Zhendong, Tester, Richland, Karp, Russell, Medikonda, Aravind, Chaturvedi, Prasoon, Ren, Yixuan, Haringsma, Henry, Etter, Jeff, Raponi, Mitch, Simmons, Andrew D, Harding, Thomas C, Niu, Deqiang, Nacht, Mariana, Westlin, William F, Petter, Russell C, Allen, Andrew, Singh, Juswinder

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Clinical Development of AVL-292; A Potent, Selective Covalent Btk Inhibitor for the Treatment of B Cell Malignancies von Evans, Erica, Tester, Richland, Aslanian, Sharon, Chaturvedi, Prasoon, Mazdiyasni, Hormoz, Ponader, Sabine, Tesar, Bethany, Sheets, Michael, Nacht, Mariana, Stiede, Kathryn, Witowski, Steve, Lounsbury, Heather, Petter, Russell, Brown, Jennifer R., Burger, Jan A., Singh, Juswinder, Westlin, William F.

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Amide-based inhibitors of p38α MAP kinase. Part 2: Design, synthesis and SAR of potent N-pyrimidyl amides von Tester, Richland, Tan, Xuefei, Luedtke, Gregory R., Nashashibi, Imad, Schinzel, Kurt, Liang, Weiling, Jung, Joon, Dugar, Sundeep, Liclican, Albert, Tabora, Jocelyn, Levy, Daniel E., Do, Steven

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Amide-based inhibitors of p38a MAP kinase. Part 1: Discovery of novel N-pyridyl amide lead molecules von Luedtke, Gregory R, Schinzel, Kurt, Tan, Xuefei, Tester, Richland W, Nashashibi, Imad, Xu, Yong-Jin, Dugar, Sundeep, Levy, Daniel E, Jung, Joon

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Amide-based inhibitors of p38a MAP kinase. Part 2: Design, synthesis and SAR of potent N-pyrimidyl amides von Tester, Richland, Tan, Xuefei, Luedtke, Gregory R, Nashashibi, Imad, Schinzel, Kurt, Liang, Weiling, Jung, Joon, Dugar, Sundeep, Liclican, Albert, Tabora, Jocelyn, Levy, Daniel E, Do, Steven

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A Novel Covalent Inhibitor of Btk Inhibits B Cell Receptor Signaling and Demonstrates Efficacy in Rheumatoid Arthritis Models von Evans, Erica, Karp, Russell, Tester, Richland, Sheets, Michael, Aslanian, Sharon, Nacht, Mariana, Zhu, Zhendong, Mazdiyasni, Hormoz, Chaturvedi, Prasoon, Petter, Russell, Westlin, William, Singh, Juswinder

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Design and synthesis of piperazine-indole p38a MAP kinase inhibitors with improved pharmacokinetic profiles von Tan, Xuefei, Tester, Richland W, Luedtke, Gregory R, Chakravarty, Sarvajit, Mavunkel, Babu J, Perumattam, John J, Lu, Qing, Nashashibi, Imad, Jung, Joon, Hu, Jie, Liclican, Albert, Almirez, Ramona, Tabora, Jocelyn, Tran, Vinh, Laney, Maureen, Levy, Daniel E, Dugar, Sundeep

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O-Bridged medium sized rings via bicyclic oxonium ylides von WEST, F. G, EBERLEIN, T. H, TESTER, R. W

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Profound Catalyst Effects in the Generation and Reactivity of Carbenoid-Derived Cyclic Ylides von West, F. G., Naidu, B. N., Tester, Richland W.

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Medium ring ethers via [1,2]-shift of acetal-derived oxonium ylides von Tester, Richland W., West, F.G.

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Salts of an epidermal growth factor receptor kinase inhibitor von Witowski, Steven Richard, Tester, Richland Wayne, Lai, Mei, Lee, Kwangho

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SALTS OF AN EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR von LAI, MEI, WITOWSKI, STEVEN, RICHARD, TESTER, RICHLAND, WAYNE, LEE, KWANGHO

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SALTS OF AN EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR von LAI, MEI, TESTER, RICHLAND WAYNE, WITOWSKI, STEVEN RICHARD, LEE, KWANGHO

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SALTS OF AN EPIDERMAL GROWTH FACTOR RECEPTOR KINASE INHIBITOR von Witowski, Steven Richard, Tester, Richland Wayne, Lai, Mei, Lee, Kwangho

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