Molecular Determinants of Vanilloid Sensitivity in TRPV1 von Gavva, Narender R, Klionsky, Lana, Qu, Yusheng, Shi, Licheng, Tamir, Rami, Edenson, Steve, Zhang, T J, Viswanadhan, Vellarkad N, Toth, Attila, Pearce, Larry V, Vanderah, Todd W, Porreca, Frank, Blumberg, Peter M, Lile, Jack, Sun, Yax, Wild, Ken, Louis, Jean-Claude, Treanor, James J S

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Species-Specific Pharmacology of Trichloro(Sulfanyl)ethyl Benzamides as Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists von Klionsky, Lana, Tamir, Rami, Gao, BaoXi, Wang, Weiya, Immke, David C, Nishimura, Nobuko, Gavva, Narender R

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Proton Activation Does Not Alter Antagonist Interaction with the Capsaicin-Binding Pocket of TRPV1 von Gavva, Narender R., Tamir, Rami, Klionsky, Lana, Norman, Mark H., Louis, Jean-Claude, Wild, Kenneth D., Treanor, James J.S.

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Design of Potent, Orally Available Antagonists of the Transient Receptor Potential Vanilloid 1. Structure−Activity Relationships of 2-Piperazin-1-yl-1H-benzimidazoles von Ognyanov, Vassil I, Balan, Chenera, Bannon, Anthony W, Bo, Yunxin, Dominguez, Celia, Fotsch, Christopher, Gore, Vijay K, Klionsky, Lana, Ma, Vu V, Qian, Yi-Xin, Tamir, Rami, Wang, Xianghong, Xi, Ning, Xu, Shimin, Zhu, Dawn, Gavva, Narender R, Treanor, James J. S, Norman, Mark H

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KTP/532 YAG laser treatment for allergic rhinitis von Yaniv, Eitan, Hadar, Tuvia, Shvero, Jacob, Tamir, Rami, Nageris, Ben

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The Vanilloid Receptor TRPV1 Is Tonically Activated In Vivo and Involved in Body Temperature Regulation von Gavva, Narender R, Bannon, Anthony W, Surapaneni, Sekhar, Hovland, David N., Jr, Lehto, Sonya G, Gore, Anu, Juan, Todd, Deng, Hong, Han, Bora, Klionsky, Lana, Kuang, Rongzhen, Le, April, Tamir, Rami, Wang, Jue, Youngblood, Brad, Zhu, Dawn, Norman, Mark H, Magal, Ella, Treanor, James J. S, Louis, Jean-Claude

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Design and Synthesis of Peripherally Restricted Transient Receptor Potential Vanilloid 1 (TRPV1) Antagonists von Tamayo, Nuria, Liao, Hongyu, Stec, Markian M, Wang, Xianghong, Chakrabarti, Partha, Retz, Dan, Doherty, Elizabeth M, Surapaneni, Sekhar, Tamir, Rami, Bannon, Anthony W, Gavva, Narender R, Norman, Mark H

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GDNF–Induced Activation of the Ret Protein Tyrosine Kinase Is Mediated by GDNFR-α, a Novel Receptor for GDNF von Jing, Shuqian, Wen, Duanzhi, Yu, Yanbin, Holst, Paige L, Luo, Yi, Fang, Mei, Tamir, Rami, Antonio, Laarni, Hu, Zheng, Cupples, Rod, Louis, Jean-Claude, Hu, Sylvia, Altrock, Bruce W, Fox, Gary M

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Novel Vanilloid Receptor-1 Antagonists:  2. Structure−Activity Relationships of 4-Oxopyrimidines Leading to the Selection of a Clinical Candidate von Doherty, Elizabeth M, Fotsch, Christopher, Bannon, Anthony W, Bo, Yunxin, Chen, Ning, Dominguez, Celia, Falsey, James, Gavva, Narender R, Katon, Jodie, Nixey, Thomas, Ognyanov, Vassil I, Pettus, Liping, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Zhu, Jiawang, Treanor, James J. S, Norman, Mark H

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Novel Vanilloid Receptor-1 Antagonists:  3. The Identification of a Second-Generation Clinical Candidate with Improved Physicochemical and Pharmacokinetic Properties von Wang, Hui-Ling, Katon, Jodie, Balan, Chenera, Bannon, Anthony W, Bernard, Charles, Doherty, Elizabeth M, Dominguez, Celia, Gavva, Narender R, Gore, Vijay, Ma, Vu, Nishimura, Nobuko, Surapaneni, Sekhar, Tang, Phi, Tamir, Rami, Thiel, Oliver, Treanor, James J. S, Norman, Mark H

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Discovery of Potent, Orally Available Vanilloid Receptor-1 Antagonists. Structure−Activity Relationship of N-Aryl Cinnamides von Doherty, Elizabeth M, Fotsch, Christopher, Bo, Yunxin, Chakrabarti, Partha P, Chen, Ning, Gavva, Narender, Han, Nianhe, Kelly, Michael G, Kincaid, John, Klionsky, Lana, Liu, Qingyian, Ognyanov, Vassil I, Tamir, Rami, Wang, Xianghong, Zhu, Jiawang, Norman, Mark H, Treanor, James J. S

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Abstract 2058: Translational regulation of SPARC by the microRNAs mir29a, b, and c von Trieu, Vuong, Hwang, Larn, Lin, Xiaoqin, Tamir, Rami, Motamed, Kouros, Desai, Neil

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Novel Vanilloid Receptor-1 Antagonists:  1. Conformationally Restricted Analogues of trans-Cinnamides von Norman, Mark H, Zhu, Jiawang, Fotsch, Christopher, Bo, Yunxin, Chen, Ning, Chakrabarti, Partha, Doherty, Elizabeth M, Gavva, Narender R, Nishimura, Nobuko, Nixey, Thomas, Ognyanov, Vassil I, Rzasa, Robert M, Stec, Markian, Surapaneni, Sekhar, Tamir, Rami, Viswanadhan, Vellarkad N, Treanor, James J. S

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Structure–activity relationship (SAR) investigations of substituted imidazole analogs as TRPV1 antagonists von Gore, Vijay K., Ma, Vu V., Tamir, Rami, Gavva, Narender R., Treanor, James J.S., Norman, Mark H.

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Generation of suppressor cells in atopic patients during immunotherapy that modulate IgE synthesis von Tamir, Rami, Castracane, John M., Rocklin, Ross E.

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Substituted aryl pyrimidines as potent and soluble TRPV1 antagonists von Stec, Markian M., Bo, Yunxin, Chakrabarti, Partha P., Liao, Lillian, Ncube, Mqhele, Tamayo, Nuria, Tamir, Rami, Gavva, Narender R., Treanor, James J.S., Norman, Mark H.

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Trisubstituted pyrimidines as transient receptor potential vanilloid 1 (TRPV1) antagonists with improved solubility von Wang, Xianghong, Chakrabarti, Partha P., Ognyanov, Vassil I., Pettus, Liping H., Tamir, Rami, Tan, Helming, Tang, Phi, Treanor, James J.S., Gavva, Narender R., Norman, Mark H.

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Synthesis and evaluation of thiazole carboxamides as vanilloid receptor 1 (TRPV1) antagonists von Xi, Ning, Bo, Yunxin, Doherty, Elizabeth M., Fotsch, Christopher, Gavva, Narender R., Han, Nianhe, Hungate, Randall W., Klionsky, Lana, Liu, Qingyian, Tamir, Rami, Xu, Shimin, Treanor, James J.S., Norman, Mark H.

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Species-specific pharmacology of Trichloro antagonists von Klionsky, Lana, Tamir, Rami, Gao, BaoXi, Wang, Weiya, Immke, David C, Nishimura, Nobuko, Gavva, Narender R

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4-Aminopyrimidine tetrahydronaphthols: A series of novel vanilloid receptor-1 antagonists with improved solubility properties von Doherty, Elizabeth M., Retz, Daniel, Gavva, Narender R., Tamir, Rami, Treanor, James J.S., Norman, Mark H.

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